ZA807078B - Secondary amines,their preparation and use in pharamaceutical compositions - Google Patents

Secondary amines,their preparation and use in pharamaceutical compositions

Info

Publication number
ZA807078B
ZA807078B ZA00807078A ZA807078A ZA807078B ZA 807078 B ZA807078 B ZA 807078B ZA 00807078 A ZA00807078 A ZA 00807078A ZA 807078 A ZA807078 A ZA 807078A ZA 807078 B ZA807078 B ZA 807078B
Authority
ZA
South Africa
Prior art keywords
sup
preparation
secondary amines
hydrogen
pharamaceutical compositions
Prior art date
Application number
ZA00807078A
Other languages
English (en)
Inventor
M Ferris
Original Assignee
Beecham Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group Ltd filed Critical Beecham Group Ltd
Publication of ZA807078B publication Critical patent/ZA807078B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/80Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/79Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D307/81Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/78Benzo [b] furans; Hydrogenated benzo [b] furans
    • C07D307/86Benzo [b] furans; Hydrogenated benzo [b] furans with an oxygen atom directly attached in position 7

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Furan Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA00807078A 1979-11-15 1980-11-14 Secondary amines,their preparation and use in pharamaceutical compositions ZA807078B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7939536 1979-11-15

Publications (1)

Publication Number Publication Date
ZA807078B true ZA807078B (en) 1981-10-28

Family

ID=10509209

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00807078A ZA807078B (en) 1979-11-15 1980-11-14 Secondary amines,their preparation and use in pharamaceutical compositions

Country Status (13)

Country Link
US (1) US4341793A (fr)
EP (1) EP0029320B1 (fr)
JP (1) JPS5683484A (fr)
AT (1) ATE14222T1 (fr)
AU (1) AU540343B2 (fr)
CA (1) CA1161053A (fr)
DE (1) DE3070865D1 (fr)
DK (1) DK489180A (fr)
ES (2) ES8202808A1 (fr)
IE (1) IE50475B1 (fr)
IL (1) IL61496A0 (fr)
NZ (1) NZ195551A (fr)
ZA (1) ZA807078B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0070133B1 (fr) * 1981-07-11 1986-05-14 Beecham Group Plc Phényléthanolamines secondaires, procédés pour leur préparation et leur application pharmaceutique
CA1219865A (fr) * 1982-05-14 1987-03-31 Leo Alig Derives de phenethanolamine d'aziridine
CA1258454A (fr) * 1982-08-10 1989-08-15 Leo Alig Phenethanolamines
EP0139921B1 (fr) * 1983-08-17 1987-03-25 Beecham Group Plc Dérivés de 2-phényléthylamine
US5151439A (en) * 1990-05-04 1992-09-29 American Cyanamid Company Substituted 5-(2-((2-aryl-2-hydroxyethyl)amino)propyl)-1,3-benzodioxoles
US5106867A (en) * 1990-05-04 1992-04-21 American Cyanamid Company Method of increasing lean meat in edible animals
US5245053A (en) * 1990-05-04 1993-09-14 American Cyanamid Company Substituted 5-(2-(2-aryl-2-hydroxyethyl)-amino)propyl)-1,3-benzodioxoles
US5061727A (en) * 1990-05-04 1991-10-29 American Cyanamid Company Substituted 5-(2-((2-aryl-2-hydroxyethyl)amino)propyl)-1,3-benzodioxoles
AT395849B (de) * 1991-04-04 1993-03-25 Noe Christian R Pharmakologisch aktive in position 3 substituierte alpha-aminomethyl-2benzofuranmethanole
CA2164009A1 (fr) * 1993-06-14 1994-12-22 Robert L. Dow Amines secondaires, agents antidiabetiques et anti-obesite
US5563171A (en) * 1993-11-05 1996-10-08 American Cyanamid Company Treatment of glaucoma and ocular hypertension with β3-adrenergic agonists
US5578638A (en) * 1993-11-05 1996-11-26 American Cyanamid Company Treatment of glaucoma and ocular hypertension with β3 -adrenergic agonists
US5627200A (en) * 1994-09-26 1997-05-06 Pfizer Inc β3 -Adrenoceptor agonists and antagonists for the treatment of intestinal motility disorders, depression, prostate disease and dyslipidemia
EP0801060A1 (fr) * 1996-04-09 1997-10-15 Pfizer Inc. Des agonistes bèta-3 adrénergiques hétérocycliques
FR2758460B1 (fr) * 1997-01-21 1999-12-31 Sanofi Sa Utilisation des agonistes des recepteurs beta-3 adrenergiques pour la preparation de medicaments cicatrisants
AU2005243239C1 (en) * 2004-05-03 2013-10-24 Janssen Pharmaceutica N.V. Indole, benzofuran and benzothiophene derivatives as selective androgen receptor modulators (SARMS)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE663926A (fr) * 1964-05-20
DE2500157C2 (de) * 1975-01-03 1983-09-15 Hoechst Ag, 6230 Frankfurt N-Acyl-4-(2-aminoäthyl)-benzoesäuren, deren Salze und Ester, Verfahren zu deren Herstellung und deren Verwendung
DK268779A (da) * 1978-07-03 1980-01-04 Lilly Co Eli Fremgangsmaade til fremstilling af phenethanolaminer

Also Published As

Publication number Publication date
IL61496A0 (en) 1980-12-31
US4341793A (en) 1982-07-27
AU6435480A (en) 1981-05-21
NZ195551A (en) 1984-11-09
EP0029320A3 (en) 1981-08-05
DK489180A (da) 1981-05-16
DE3070865D1 (en) 1985-08-14
ATE14222T1 (de) 1985-07-15
ES496880A0 (es) 1982-02-16
IE802371L (en) 1981-05-15
AU540343B2 (en) 1984-11-15
EP0029320B1 (fr) 1985-07-10
ES507410A0 (es) 1982-09-01
JPS5683484A (en) 1981-07-08
EP0029320A2 (fr) 1981-05-27
CA1161053A (fr) 1984-01-24
IE50475B1 (en) 1986-04-30
ES8207165A1 (es) 1982-09-01
ES8202808A1 (es) 1982-02-16

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