ZA201305992B - 5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives - Google Patents

5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives

Info

Publication number
ZA201305992B
ZA201305992B ZA2013/05992A ZA201305992A ZA201305992B ZA 201305992 B ZA201305992 B ZA 201305992B ZA 2013/05992 A ZA2013/05992 A ZA 2013/05992A ZA 201305992 A ZA201305992 A ZA 201305992A ZA 201305992 B ZA201305992 B ZA 201305992B
Authority
ZA
South Africa
Prior art keywords
oxopyrimidine
fluoro
carboxylate derivatives
carboxylate
derivatives
Prior art date
Application number
ZA2013/05992A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA201305992(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of ZA201305992B publication Critical patent/ZA201305992B/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA2013/05992A 2009-08-07 2013-08-14 5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives ZA201305992B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07
PCT/US2010/044585 WO2011017544A1 (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
ZA201305992B true ZA201305992B (en) 2014-10-29

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA2013/05992A ZA201305992B (en) 2009-08-07 2013-08-14 5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives

Country Status (28)

Country Link
US (1) US8318758B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP2462133B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP5818791B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR101792286B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN102548979B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (1) AU2010279408B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR112012002807B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (1) CA2769251C (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CL (1) CL2012000314A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CO (1) CO6491089A2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CR (1) CR20120033A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK2462133T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EA (1) EA022930B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EC (1) ECSP12011651A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2506169T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HN (1) HN2012000261A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL217954A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IN (1) IN2012DN00695A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MX2012001623A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NI (1) NI201200019A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NZ (1) NZ597638A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PE (1) PE20120689A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PL (1) PL2462133T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
PT (1) PT2462133E (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RS (1) RS53658B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
UA (1) UA106086C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO2011017544A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ZA (1) ZA201305992B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT2462134E (pt) * 2009-08-07 2014-07-28 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
UA117743C2 (uk) 2012-12-28 2018-09-25 Адама Махтешім Лтд. N-(заміщені)-5-фтор-4-іміно-3-метил-2-оксо-3,4-дигідропіримідин-1(2h)-карбоксамідні похідні
RU2656101C2 (ru) 2012-12-28 2018-05-31 Адама Мактешим Лтд. Производные 1-(замещенный бензоил)-5-фтор-4-имино-3-метил-3,4-дигидропиримидин-2(1h)-она
DK2938194T3 (da) * 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
NZ708981A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN106068268A (zh) 2013-12-31 2016-11-02 阿达玛马克西姆股份有限公司 5‑氟‑4‑亚氨基‑3‑(烷基/取代烷基)‑1‑(芳基磺酰基)‑3,4‑二氢嘧啶‑2(1h)‑酮及其制备方法
JP6608366B2 (ja) 2013-12-31 2019-11-20 アダマ・マクテシム・リミテッド 真菌防除のための相乗的殺真菌性混合物および組成物
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
MX380092B (es) 2015-11-06 2025-03-11 Samumed Llc Tratamiento de la osteoartritis.
MY199242A (en) 2016-06-01 2023-10-22 Samumed Llc Process for preparing n-(5-(3-(7-(3-fluorophenyl)-3h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide
CN118515619A (zh) 2017-07-17 2024-08-20 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
DE69712331T2 (de) * 1996-03-11 2002-11-28 Syngenta Participations Ag, Basel Pyrimidin-4-on derivate als pestizidesmittel
WO2004037159A2 (en) * 2002-10-23 2004-05-06 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
RU2470927C2 (ru) * 2007-04-27 2012-12-27 Дайити Санкио Компани,Лимитед Производные с азотсодержащим шестичленным ароматическим кольцом и содержащие их фармацевтические продукты
KR20110042204A (ko) 2008-08-01 2011-04-25 다우 아그로사이언시즈 엘엘씨 살진균제로서의 5-플루오로시토신의 용도

Also Published As

Publication number Publication date
BR112012002807A2 (pt) 2015-10-13
NI201200019A (es) 2012-05-22
MX2012001623A (es) 2012-04-11
DK2462133T3 (en) 2015-01-05
CL2012000314A1 (es) 2012-10-05
ECSP12011651A (es) 2012-03-30
JP5818791B2 (ja) 2015-11-18
CA2769251A1 (en) 2011-02-10
KR20120043069A (ko) 2012-05-03
EP2462133A1 (en) 2012-06-13
ES2506169T3 (es) 2014-10-13
HK1172892A1 (en) 2013-05-03
EA201270255A1 (ru) 2012-07-30
EP2462133A4 (en) 2013-01-16
CR20120033A (es) 2012-03-22
CA2769251C (en) 2018-05-15
BR112012002807B1 (pt) 2018-07-10
EA022930B1 (ru) 2016-03-31
PL2462133T3 (pl) 2015-03-31
WO2011017544A1 (en) 2011-02-10
IL217954A0 (en) 2012-03-29
IN2012DN00695A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2015-06-19
CO6491089A2 (es) 2012-07-31
US8318758B2 (en) 2012-11-27
IL217954A (en) 2016-02-29
JP2013501726A (ja) 2013-01-17
CN102548979A (zh) 2012-07-04
AU2010279408A1 (en) 2012-02-09
NZ597638A (en) 2014-06-27
RS53658B1 (en) 2015-04-30
CN102548979B (zh) 2015-05-13
UA106086C2 (uk) 2014-07-25
PT2462133E (pt) 2014-12-26
EP2462133B1 (en) 2014-09-24
BR112012002807A8 (pt) 2017-07-11
KR101792286B1 (ko) 2017-10-31
US20110034491A1 (en) 2011-02-10
HN2012000261A (es) 2015-01-05
PE20120689A1 (es) 2012-06-06
AU2010279408B2 (en) 2015-09-10

Similar Documents

Publication Publication Date Title
ZA201200895B (en) Aminopyrazole derivative
ZA201203205B (en) Benzimidazole-imidazole derivatives
IL217956A0 (en) N1-sulfonyl-5-fluoropyrimidinone derivatives
IL217953A0 (en) 5-fluoropyrimidinone derivatives
IL216007A0 (en) Isoxazole-pyridine derivatives
ZA201305992B (en) 5-fluoro-2-oxopyrimidine-1(2h)-carboxylate derivatives
IL215109A0 (en) Isoxazole-pyridazine derivatives
ZA201106855B (en) Oxasiazole derivatives
IL214941A0 (en) Isoxazole-pyrazole derivatives
ZA201104991B (en) Deoxyactagardine derivatives
IL217950A0 (en) N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
IL217952A0 (en) N1-acyl-5-fluoropyrimidinone derivatives
ZA201109370B (en) Pyrazinooxazepine derivatives
ZA201104279B (en) Tetrahydronaphthalen-2-ol derivatives
GB0912499D0 (en) Indopyl-pyridone derivatives