ZA200804610B - Aminophenylsulfonamide derivatives as HIV protease inhibitor - Google Patents

Aminophenylsulfonamide derivatives as HIV protease inhibitor

Info

Publication number
ZA200804610B
ZA200804610B ZA200804610A ZA200804610A ZA200804610B ZA 200804610 B ZA200804610 B ZA 200804610B ZA 200804610 A ZA200804610 A ZA 200804610A ZA 200804610 A ZA200804610 A ZA 200804610A ZA 200804610 B ZA200804610 B ZA 200804610B
Authority
ZA
South Africa
Prior art keywords
aminophenylsulfonamide
derivatives
protease inhibitor
hiv protease
hiv
Prior art date
Application number
ZA200804610A
Other languages
English (en)
Inventor
Kock Herman Augustinus De
Tim Hugo Maria Jonckers
Stefaan Julien Last
Paul Jozef Gabrriel Maria Boonants
Dominique Louis Nestor Ghislain Surleraux
Piet Tom Bert Paul Wigerinck
Original Assignee
Tibotec Pharm Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35822401&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ZA200804610(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Tibotec Pharm Ltd filed Critical Tibotec Pharm Ltd
Publication of ZA200804610B publication Critical patent/ZA200804610B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA200804610A 2005-11-28 2008-05-27 Aminophenylsulfonamide derivatives as HIV protease inhibitor ZA200804610B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP05111393 2005-11-28

Publications (1)

Publication Number Publication Date
ZA200804610B true ZA200804610B (en) 2009-11-25

Family

ID=35822401

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200804610A ZA200804610B (en) 2005-11-28 2008-05-27 Aminophenylsulfonamide derivatives as HIV protease inhibitor

Country Status (12)

Country Link
US (1) US7803836B2 (pt)
EP (1) EP1960381B1 (pt)
JP (1) JP5210876B2 (pt)
CN (1) CN101304987B (pt)
AR (1) AR058238A1 (pt)
AU (1) AU2006316399B2 (pt)
BR (1) BRPI0619005A2 (pt)
CA (1) CA2628540C (pt)
EA (1) EA016060B1 (pt)
TW (1) TWI432438B (pt)
WO (1) WO2007060249A1 (pt)
ZA (1) ZA200804610B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI482775B (zh) 2008-09-01 2015-05-01 Tibotec Pharm Ltd 用於製備（３ｒ，３ａｓ，６ａｒ）－六氫呋喃并〔２，３－ｂ〕呋喃－３－基（１ｓ，２ｒ）－３－〔〔（４－胺基苯基）磺醯基〕（異丁基）胺基〕－１－苯甲基－２－羥基丙基胺基甲酸酯之方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5723490A (en) * 1992-09-08 1998-03-03 Vertex Pharmaceuticals Incorporated THF-containing sulfonamide inhibitors of aspartyl protease
US6436989B1 (en) 1997-12-24 2002-08-20 Vertex Pharmaceuticals, Incorporated Prodrugs of aspartyl protease inhibitors
ID25551A (id) 1997-12-24 2000-10-12 Vertex Pharma Bahan baku obat penghambat protease aspartil
AU2012199A (en) 1997-12-24 1999-07-19 Vertex Pharmaceuticals Incorporated Prodrugs of aspartyl protease inhibitors
AU2010299A (en) 1997-12-24 1999-07-19 Vertex Pharmaceuticals Incorporated Prodrugs os aspartyl protease inhibitors
WO1999065870A2 (en) * 1998-06-19 1999-12-23 Vertex Pharmaceuticals Incorporated Sulfonamide inhibitors of aspartyl protease
AU4828199A (en) * 1998-06-23 2000-01-10 Board Of Trustees Of The University Of Illinois, The Multi-drug resistant retroviral protease inhibitors and associated methods
AR037797A1 (es) 2001-12-12 2004-12-01 Tibotec Pharm Ltd Combinacion de inhibidores de proteasa dependientes del citocromo p450
US7157489B2 (en) * 2002-03-12 2007-01-02 The Board Of Trustees Of The University Of Illinois HIV protease inhibitors
AU2003231766A1 (en) 2002-04-26 2003-11-10 Gilead Sciences, Inc. Non nucleoside reverse transcriptase inhibitors
AU2004309122B2 (en) 2003-12-23 2011-07-21 Janssen Sciences Ireland Unlimited Company Process for the preparation of (3R,3aS,6AR)-hexahydrofuro [2,3-b] furan-3-yl (1S,2R)-3-[[(4-aminophenyl) sulfonyl] (isobutyl) amino]-1-benzyl-2-hydroxypropylcarbamate

Also Published As

Publication number Publication date
AU2006316399B2 (en) 2012-04-12
EA016060B1 (ru) 2012-01-30
EP1960381B1 (en) 2015-06-17
US20080306061A1 (en) 2008-12-11
CN101304987A (zh) 2008-11-12
CA2628540A1 (en) 2007-05-31
EA200801477A1 (ru) 2009-02-27
EP1960381A1 (en) 2008-08-27
US7803836B2 (en) 2010-09-28
CN101304987B (zh) 2013-11-06
TWI432438B (zh) 2014-04-01
AU2006316399A1 (en) 2007-05-31
WO2007060249A1 (en) 2007-05-31
JP2009517370A (ja) 2009-04-30
TW200738731A (en) 2007-10-16
JP5210876B2 (ja) 2013-06-12
BRPI0619005A2 (pt) 2013-01-08
AR058238A1 (es) 2008-01-23
CA2628540C (en) 2015-09-08

Similar Documents

Publication Publication Date Title
IL179056A0 (en) An hiv protease inhibitor
ZA200707650B (en) Azolylacylguanidines as ß-secretase inhibitors
EP1981519A4 (en) PROTEASE INHIBITION
SI1948666T1 (sl) Hiv integrazni inhibitorji
ZA200710951B (en) Piperidinyl-substituted isoquinolone derivatives as Rhokinase inhibitors
EP1839669A4 (en) NEW ANGIOGENESEHEMMER
EP1881825A4 (en) INHIBITORS OF HIV INTEGRASE
HK1127345A1 (en) Azapeptide derivatives as hiv protease inhibitors
IL183850A0 (en) Hiv protease inhibitors
HK1180311A1 (zh) 抗病毒雙趺喃衍生物用作 蛋白酶抑制劑和其中間產物
HK1127351A1 (zh) 抗病毒蛋白酶抑制劑
AP2007004282A0 (en) Derivatives of A 1-phenyltriazole as antiparasiticagents
EP1910363A4 (en) INHIBITORS OF HIV INTEGRASE
EP1855672A4 (en) HIV PROTEASE INHIBITORS
GB0513841D0 (en) Cysteine protease inhibitors
AU2007337830A8 (en) Benzenesulfonamide derivatives as HIV protease inhibitors
ZA200804607B (en) Substituted aminophenylsulfonamide compounds as HIV protease inhibitor
EP2134336A4 (en) HIV PROTEASE INHIBITORS DERIVED FROM BENZOFURAN
ZA200800672B (en) Introcatechol derivatives as COMT inhibitors
EP1910356A4 (en) HIV integrase
ZA200706305B (en) HIV protease inhibitors
GB0513839D0 (en) Cysteine protease inhibitors
GB0513840D0 (en) Cysteine protease inhibitors
ZA200804610B (en) Aminophenylsulfonamide derivatives as HIV protease inhibitor
ZA200705383B (en) Benzoyl-tetrahydropyridine as GlyT-1 inhibitors