ZA200701332B - Prodrugs containing novel bio-cleavable linkers - Google Patents

Prodrugs containing novel bio-cleavable linkers

Info

Publication number
ZA200701332B
ZA200701332B ZA200701332A ZA200701332A ZA200701332B ZA 200701332 B ZA200701332 B ZA 200701332B ZA 200701332 A ZA200701332 A ZA 200701332A ZA 200701332 A ZA200701332 A ZA 200701332A ZA 200701332 B ZA200701332 B ZA 200701332B
Authority
ZA
South Africa
Prior art keywords
cleavable linkers
containing novel
prodrugs containing
novel bio
bio
Prior art date
Application number
ZA200701332A
Other languages
English (en)
Inventor
Satyam Apparao
Original Assignee
Nicholas Piramal India Ltd
Satyam Apparao
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nicholas Piramal India Ltd, Satyam Apparao filed Critical Nicholas Piramal India Ltd
Publication of ZA200701332B publication Critical patent/ZA200701332B/xx

Links

ZA200701332A 2004-08-26 2007-02-14 Prodrugs containing novel bio-cleavable linkers ZA200701332B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US60463204P 2004-08-26 2004-08-26

Publications (1)

Publication Number Publication Date
ZA200701332B true ZA200701332B (en) 2008-12-31

Family

ID=38890139

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200701332A ZA200701332B (en) 2004-08-26 2007-02-14 Prodrugs containing novel bio-cleavable linkers

Country Status (2)

Country Link
CN (1) CN101039701A (zh)
ZA (1) ZA200701332B (zh)

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* Cited by examiner, † Cited by third party
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CN101701061B (zh) * 2009-10-30 2011-09-28 北京化工大学 维生素c为亲水片断的药物输送材料及其制备方法
JP2013523777A (ja) * 2010-04-02 2013-06-17 ティーエスアールエル インコーポレイテッド ノイラミニダーゼ阻害剤
CA2800497C (en) * 2010-05-10 2019-03-12 The Regents Of The University Of California Methods for preparing ratiometric combinatorial nanoparticules
CN102335190B (zh) * 2011-07-18 2013-01-23 华东师范大学 还原降解释药可控的巯嘌呤纳米胶束前药及其应用
WO2013073480A1 (ja) * 2011-11-18 2013-05-23 日油株式会社 細胞内動態を改善したカチオン性脂質
CN105658651A (zh) * 2012-09-21 2016-06-08 巴兹尔·里格斯 用于治疗炎症相关的病症、疼痛和发热、皮肤病症、癌症及其癌症前期状况的组合物
MX368258B (es) 2013-03-15 2019-09-25 Zymeworks Inc Compuestos citotoxicos y antimitoticos y metodos de uso de los mismos.
CN104327018B (zh) * 2013-12-01 2016-07-13 复旦大学 一种含二硫键可聚合紫杉醇单体及其合成方法
MX2016008444A (es) * 2013-12-27 2017-01-11 Zymeworks Inc Sistemas de enlace que contienen sulfonamida para conjugados de farmacos.
EP3194421B1 (en) 2014-09-17 2021-11-03 Zymeworks Inc. Cytotoxic and anti-mitotic compounds, and methods of using the same
CN105732643A (zh) * 2016-04-18 2016-07-06 苏州大学 一种偶联物、其制备方法及在制备ido酶抑制剂和非甾体抗炎药物中的应用
CN106831805B (zh) * 2017-03-21 2019-03-15 莎穆(上海)生物科技有限公司 一种喜树碱-阿霉素前药及其制备方法和应用
CN109207531B (zh) * 2017-07-03 2022-04-19 上海医药工业研究院 甲砜霉素与氟苯尼考关键中间体的生物制备方法
CN113645968A (zh) * 2019-03-18 2021-11-12 西达赛奈医疗中心 治疗胃肠疾病和障碍的组合物和方法
CN110256313B (zh) * 2019-05-15 2021-01-29 江苏省原子医学研究所 一种光敏剂前药化合物及其制备方法和应用
CN111202850A (zh) * 2019-11-05 2020-05-29 中国药科大学 一种喜树碱前药及其制备方法和应用
CN111053761B (zh) * 2020-01-16 2022-05-03 杭州旦承医药科技有限公司 一种吸入用双膦酸类药物及其制备方法及其在慢性阻塞性肺疾病的用途
IL296152A (en) * 2020-03-23 2022-11-01 John M H Gregg Antiviral compounds and methods of their administration
CN114848835B (zh) * 2022-03-22 2023-08-25 暨南大学 塞来昔布的聚乙二醇修饰及连接叶酸基团的靶向药物分子及制备方法

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Publication number Publication date
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