ZA200608624B

ZA200608624B - Pharmaceutical salts of 3-0(3',3'-dimethylsuccinyl) betulinic acid

Pharmaceutical salts of 3-0(3',3'-dimethylsuccinyl) betulinic acid Download PDF

Info

Publication number: ZA200608624B
Authority: ZA; South Africa
Prior art keywords: pharmaceutical composition; dsb; salt; administered; agent
Prior art date: 2004-03-17

Application number

ZA200608624A

Other languages

English (en)

Inventor

Power Martin Dale

Martin David Eugene

Original Assignee

Panacos Pharmaceuticals Inc

Priority date

2004-03-17

Filing date

2005-03-17

Publication date

2008-05-28

2005-03-17 Application filed by Panacos Pharmaceuticals Inc filed Critical Panacos Pharmaceuticals Inc

2008-05-28 Publication of ZA200608624B publication Critical patent/ZA200608624B/en

Links

150000003839 salts Chemical class 0.000 title claims description 79
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PZXJOHSZQAEJFE-UHFFFAOYSA-N dihydrobetulinic acid Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C)CCC5(C(O)=O)CCC(C(C)C)C5C4CCC3C21C PZXJOHSZQAEJFE-UHFFFAOYSA-N 0.000 title claims description 19
QGJZLNKBHJESQX-UHFFFAOYSA-N 3-Epi-Betulin-Saeure Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C)CCC5(C(O)=O)CCC(C(=C)C)C5C4CCC3C21C QGJZLNKBHJESQX-UHFFFAOYSA-N 0.000 title claims description 18
CLOUCVRNYSHRCF-UHFFFAOYSA-N 3beta-Hydroxy-20(29)-Lupen-3,27-oic acid Natural products C1CC(O)C(C)(C)C2CCC3(C)C4(C(O)=O)CCC5(C)CCC(C(=C)C)C5C4CCC3C21C CLOUCVRNYSHRCF-UHFFFAOYSA-N 0.000 title claims description 18
QGJZLNKBHJESQX-FZFNOLFKSA-N betulinic acid Chemical compound C1C[C@H](O)C(C)(C)[C@@H]2CC[C@@]3(C)[C@]4(C)CC[C@@]5(C(O)=O)CC[C@@H](C(=C)C)[C@@H]5[C@H]4CC[C@@H]3[C@]21C QGJZLNKBHJESQX-FZFNOLFKSA-N 0.000 title claims description 18
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