ZA200605148B - Antimicrobial preservatives to achieve multi-dose formulation using beta-cyclodextrins for liquid dosage forms - Google Patents
Antimicrobial preservatives to achieve multi-dose formulation using beta-cyclodextrins for liquid dosage forms Download PDFInfo
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- ZA200605148B ZA200605148B ZA200605148A ZA200605148A ZA200605148B ZA 200605148 B ZA200605148 B ZA 200605148B ZA 200605148 A ZA200605148 A ZA 200605148A ZA 200605148 A ZA200605148 A ZA 200605148A ZA 200605148 B ZA200605148 B ZA 200605148B
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- ZA
- South Africa
- Prior art keywords
- cyclodextrin
- preservative
- compound
- formula
- cresol
- Prior art date
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Classifications
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- A61K31/716—Glucans
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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- A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
- A61K47/6949—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes
- A61K47/6951—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit inclusion complexes, e.g. clathrates, cavitates or fullerenes using cyclodextrin
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P31/10—Antimycotics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
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- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
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US54089704P | 2004-01-30 | 2004-01-30 |
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Family Applications (1)
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ZA200605148A ZA200605148B (en) | 2004-01-30 | 2006-06-22 | Antimicrobial preservatives to achieve multi-dose formulation using beta-cyclodextrins for liquid dosage forms |
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US (1) | US8183230B2 (ko) |
EP (1) | EP1713504B1 (ko) |
JP (1) | JP5021318B2 (ko) |
KR (1) | KR100834232B1 (ko) |
CN (1) | CN101090735A (ko) |
AR (2) | AR047469A1 (ko) |
AU (1) | AU2005216709B2 (ko) |
BR (1) | BRPI0506496B8 (ko) |
CA (1) | CA2554346C (ko) |
CO (1) | CO5700794A2 (ko) |
CY (1) | CY1119188T1 (ko) |
DK (1) | DK1713504T3 (ko) |
ES (1) | ES2638113T3 (ko) |
HU (1) | HUE034099T2 (ko) |
IL (1) | IL176676A0 (ko) |
LT (1) | LT1713504T (ko) |
NO (1) | NO20063858L (ko) |
NZ (1) | NZ548236A (ko) |
PL (1) | PL1713504T3 (ko) |
PT (1) | PT1713504T (ko) |
RU (1) | RU2332997C2 (ko) |
SI (1) | SI1713504T1 (ko) |
TW (1) | TW200524632A (ko) |
WO (1) | WO2005082416A2 (ko) |
ZA (1) | ZA200605148B (ko) |
Families Citing this family (9)
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AU2013273764B2 (en) * | 2011-11-29 | 2016-05-05 | Zoetis Services Llc | Pharmaceutical compositions |
CN107261152B (zh) | 2011-11-29 | 2022-03-04 | 优奥斯私人有限公司 | 包含环糊精和疏水性药物的可注射药物组合物的防腐方法 |
EP3865120A1 (en) * | 2013-07-19 | 2021-08-18 | Boehringer Ingelheim Vetmedica GmbH | Preserved etherified cyclodextrin derivatives containing liquid aqueous pharmaceutical composition |
NL2015865B1 (en) | 2015-11-27 | 2017-06-13 | Le Vet B V | Maropitant Formulation. |
CN110730662A (zh) | 2017-04-10 | 2020-01-24 | 才思治疗公司 | 用于治疗共核蛋白病的nk1-拮抗剂组合和方法 |
US11266633B2 (en) | 2017-06-30 | 2022-03-08 | Chase Therapeutics Corporation | NK-1 antagonist compositions and methods for use in treating depression |
US10959962B2 (en) * | 2019-02-15 | 2021-03-30 | Saol International Development Ltd. | Injectable phenol formulations and methods of their use |
EP3725298A1 (en) | 2019-04-16 | 2020-10-21 | Faes Farma, S.A. | Stable and preserved pharmaceutical compositions of bilastine |
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- 2005-01-17 CN CNA2005800032849A patent/CN101090735A/zh active Pending
- 2005-01-17 EP EP05702263.4A patent/EP1713504B1/en active Active
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