ZA200600756B - 2-methoxymethyl-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octane tartrate salts - Google Patents
2-methoxymethyl-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octane tartrate salts Download PDFInfo
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- ZA200600756B ZA200600756B ZA200600756A ZA200600756A ZA200600756B ZA 200600756 B ZA200600756 B ZA 200600756B ZA 200600756 A ZA200600756 A ZA 200600756A ZA 200600756 A ZA200600756 A ZA 200600756A ZA 200600756 B ZA200600756 B ZA 200600756B
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- 235000015424 sodium Nutrition 0.000 description 1
- 239000007858 starting material Substances 0.000 description 1
- 230000035882 stress Effects 0.000 description 1
- 238000007920 subcutaneous administration Methods 0.000 description 1
- 239000004094 surface-active agent Substances 0.000 description 1
- 208000024891 symptom Diseases 0.000 description 1
- 210000003568 synaptosome Anatomy 0.000 description 1
- 238000003786 synthesis reaction Methods 0.000 description 1
- 239000000454 talc Substances 0.000 description 1
- 229910052623 talc Inorganic materials 0.000 description 1
- 150000003892 tartrate salts Chemical class 0.000 description 1
- 238000012360 testing method Methods 0.000 description 1
- 150000004685 tetrahydrates Chemical class 0.000 description 1
- 231100001274 therapeutic index Toxicity 0.000 description 1
- 238000004448 titration Methods 0.000 description 1
- 230000000699 topical effect Effects 0.000 description 1
- 231100000331 toxic Toxicity 0.000 description 1
- 230000002588 toxic effect Effects 0.000 description 1
- 231100000419 toxicity Toxicity 0.000 description 1
- 230000001988 toxicity Effects 0.000 description 1
- CYRMSUTZVYGINF-UHFFFAOYSA-N trichlorofluoromethane Chemical compound FC(Cl)(Cl)Cl CYRMSUTZVYGINF-UHFFFAOYSA-N 0.000 description 1
- 229940029284 trichlorofluoromethane Drugs 0.000 description 1
- 150000004684 trihydrates Chemical class 0.000 description 1
- 229910052722 tritium Inorganic materials 0.000 description 1
- 239000003981 vehicle Substances 0.000 description 1
- 239000011345 viscous material Substances 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200301117 | 2003-07-31 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200600756B true ZA200600756B (en) | 2007-05-30 |
Family
ID=36701727
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200600756A ZA200600756B (en) | 2003-07-31 | 2004-07-29 | 2-methoxymethyl-3-(3,4-dichlorophenyl)-8-azabicyclo[3.2.1]octane tartrate salts |
Country Status (22)
| Country | Link |
|---|---|
| US (1) | US7700619B2 (sl) |
| EP (1) | EP1651223B1 (sl) |
| JP (1) | JP4711961B2 (sl) |
| CN (1) | CN100427484C (sl) |
| AR (1) | AR045141A1 (sl) |
| AT (1) | ATE355060T1 (sl) |
| AU (1) | AU2004260837C1 (sl) |
| BR (1) | BRPI0413035A (sl) |
| CA (1) | CA2534295A1 (sl) |
| DE (1) | DE602004005048T2 (sl) |
| DK (1) | DK1651223T3 (sl) |
| ES (1) | ES2281827T3 (sl) |
| MY (1) | MY140105A (sl) |
| NZ (1) | NZ544957A (sl) |
| PL (1) | PL1651223T3 (sl) |
| PT (1) | PT1651223E (sl) |
| RU (1) | RU2348631C2 (sl) |
| SI (1) | SI1651223T1 (sl) |
| TW (1) | TW200507844A (sl) |
| UA (1) | UA86025C2 (sl) |
| WO (1) | WO2005011694A1 (sl) |
| ZA (1) | ZA200600756B (sl) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080200498A1 (en) * | 2005-07-12 | 2008-08-21 | Angelo Ceci | Pharmaceutical Composition For The Treatment Of Disorders Of Sexual Desire |
| WO2007028769A1 (en) * | 2005-09-05 | 2007-03-15 | Neurosearch A/S | Monoamine neurotransmitter re-uptake inhibitor for neuroprotection |
| EP1779851A1 (en) | 2005-10-31 | 2007-05-02 | Boehringer Ingelheim Pharma GmbH & Co.KG | Treatment of diabetes |
| GB0703998D0 (en) * | 2007-03-01 | 2007-04-11 | Glaxo Group Ltd | Novel salt |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8923209D0 (en) * | 1989-10-14 | 1989-11-29 | Wyeth John & Brother Ltd | Heterocyclic compounds |
| CN1077574C (zh) * | 1996-02-22 | 2002-01-09 | 神经研究公司 | 托烷衍生物,其制备和应用 |
| AU2002365288A1 (en) * | 2001-11-30 | 2003-06-10 | Neurosearch A/S | Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases |
-
2004
- 2004-07-28 AR ARP040102679A patent/AR045141A1/es not_active Application Discontinuation
- 2004-07-29 TW TW093122661A patent/TW200507844A/zh unknown
- 2004-07-29 ZA ZA200600756A patent/ZA200600756B/en unknown
- 2004-07-29 UA UAA200600268A patent/UA86025C2/ru unknown
- 2004-07-29 DE DE602004005048T patent/DE602004005048T2/de active Active
- 2004-07-29 NZ NZ544957A patent/NZ544957A/en unknown
- 2004-07-29 SI SI200430267T patent/SI1651223T1/sl unknown
- 2004-07-29 DK DK04766360T patent/DK1651223T3/da active
- 2004-07-29 WO PCT/EP2004/051651 patent/WO2005011694A1/en active IP Right Grant
- 2004-07-29 RU RU2005141065/04A patent/RU2348631C2/ru not_active IP Right Cessation
- 2004-07-29 ES ES04766360T patent/ES2281827T3/es active Active
- 2004-07-29 EP EP04766360A patent/EP1651223B1/en active Active
- 2004-07-29 CN CNB2004800198958A patent/CN100427484C/zh not_active Expired - Fee Related
- 2004-07-29 BR BRPI0413035-9A patent/BRPI0413035A/pt not_active Application Discontinuation
- 2004-07-29 US US10/566,384 patent/US7700619B2/en not_active Expired - Fee Related
- 2004-07-29 CA CA002534295A patent/CA2534295A1/en not_active Abandoned
- 2004-07-29 AU AU2004260837A patent/AU2004260837C1/en not_active Ceased
- 2004-07-29 JP JP2006521585A patent/JP4711961B2/ja not_active Expired - Fee Related
- 2004-07-29 AT AT04766360T patent/ATE355060T1/de not_active IP Right Cessation
- 2004-07-29 PT PT04766360T patent/PT1651223E/pt unknown
- 2004-07-29 PL PL04766360T patent/PL1651223T3/pl unknown
- 2004-07-30 MY MYPI20043081A patent/MY140105A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP2007509030A (ja) | 2007-04-12 |
| AU2004260837A1 (en) | 2005-02-10 |
| PL1651223T3 (pl) | 2007-07-31 |
| ATE355060T1 (de) | 2006-03-15 |
| US20070043075A1 (en) | 2007-02-22 |
| MY140105A (en) | 2009-11-30 |
| WO2005011694A1 (en) | 2005-02-10 |
| ES2281827T3 (es) | 2007-10-01 |
| TW200507844A (en) | 2005-03-01 |
| EP1651223B1 (en) | 2007-02-28 |
| AR045141A1 (es) | 2005-10-19 |
| RU2005141065A (ru) | 2006-08-10 |
| SI1651223T1 (sl) | 2007-08-31 |
| UA86025C2 (en) | 2009-03-25 |
| RU2348631C2 (ru) | 2009-03-10 |
| CN100427484C (zh) | 2008-10-22 |
| DK1651223T3 (da) | 2007-06-11 |
| CA2534295A1 (en) | 2005-02-10 |
| CN1822837A (zh) | 2006-08-23 |
| AU2004260837C1 (en) | 2010-08-19 |
| DE602004005048T2 (de) | 2007-08-16 |
| EP1651223A1 (en) | 2006-05-03 |
| NZ544957A (en) | 2009-02-28 |
| DE602004005048D1 (de) | 2007-04-12 |
| JP4711961B2 (ja) | 2011-06-29 |
| PT1651223E (pt) | 2007-03-30 |
| BRPI0413035A (pt) | 2006-10-03 |
| US7700619B2 (en) | 2010-04-20 |
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