ZA200405859B - Pyrrolopyrimidines as phosphodiesterase VII inhibitors. - Google Patents
Pyrrolopyrimidines as phosphodiesterase VII inhibitors. Download PDFInfo
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- ZA200405859B ZA200405859B ZA200405859A ZA200405859A ZA200405859B ZA 200405859 B ZA200405859 B ZA 200405859B ZA 200405859 A ZA200405859 A ZA 200405859A ZA 200405859 A ZA200405859 A ZA 200405859A ZA 200405859 B ZA200405859 B ZA 200405859B
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Classifications
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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DE10163991A DE10163991A1 (de) | 2001-12-24 | 2001-12-24 | Pyrrolo-pyrimidine |
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EP (1) | EP1458722B1 (fr) |
JP (1) | JP2005520801A (fr) |
KR (1) | KR20040071252A (fr) |
CN (1) | CN1608067A (fr) |
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AT (1) | ATE411316T1 (fr) |
AU (1) | AU2002367090B2 (fr) |
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RU (1) | RU2004122924A (fr) |
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ZA (1) | ZA200405859B (fr) |
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DE10226420A1 (de) * | 2002-06-13 | 2004-01-15 | Eucro European Contract Research Gmbh & Co Kg | Verfahren zur Behandlung der Artherosklerose |
CN100374441C (zh) * | 2003-06-06 | 2008-03-12 | 天津倍方科技发展有限公司 | 二氢吡咯[2,3-d]嘧啶-4-酮衍生物,其制备方法及其制药用途 |
JP4783731B2 (ja) * | 2003-08-29 | 2011-09-28 | ヴァーナリス(ケンブリッジ)リミテッド | ピリミドチオフェン化合物 |
WO2005063251A1 (fr) * | 2003-12-17 | 2005-07-14 | Pfizer Products Inc. | Tuteur modifie utile pour liberer des medicaments le long du support du tuteur |
PE20060272A1 (es) * | 2004-05-24 | 2006-05-22 | Glaxo Group Ltd | (2r,3r,4s,5r,2'r,3'r,4's,5's)-2,2'-{trans-1,4-ciclohexanodiilbis-[imino(2-{[2-(1-metil-1h-imidazol-4-il)etil]amino}-9h-purin-6,9-diil)]}bis[5-(2-etil-2h-tetrazol-5-il)tetrahidro-3,4-furanodiol] como agonista a2a |
DE102005022977A1 (de) * | 2005-05-19 | 2006-12-07 | Merck Patent Gmbh | Phenylchinazolinderivate |
GB0514809D0 (en) | 2005-07-19 | 2005-08-24 | Glaxo Group Ltd | Compounds |
EP2258359A3 (fr) | 2005-08-26 | 2011-04-06 | Braincells, Inc. | Neurogenèse par modulation des récepteurs muscariniques avec sabcomeline |
CA2620333A1 (fr) | 2005-08-26 | 2007-03-01 | Braincells, Inc. | Neurogenese par modulation du recepteur muscarinique |
EP1940389A2 (fr) | 2005-10-21 | 2008-07-09 | Braincells, Inc. | Modulation de la neurogenese par inhibition de la pde |
EP1942879A1 (fr) | 2005-10-31 | 2008-07-16 | Braincells, Inc. | Modulation de la neurogenese dont la mediation est assuree par recepteur gaba |
US20100216734A1 (en) | 2006-03-08 | 2010-08-26 | Braincells, Inc. | Modulation of neurogenesis by nootropic agents |
JP2009536667A (ja) | 2006-05-09 | 2009-10-15 | ブレインセルス,インコーポレイティド | 5ht受容体介在性の神経新生 |
JP2009536669A (ja) | 2006-05-09 | 2009-10-15 | ブレインセルス,インコーポレイティド | アンジオテンシン調節による神経新生 |
BRPI0716604A2 (pt) | 2006-09-08 | 2013-04-09 | Braincells Inc | combinaÇÕes contendo um derivado de 4-acilaminopiridina |
US20100184806A1 (en) | 2006-09-19 | 2010-07-22 | Braincells, Inc. | Modulation of neurogenesis by ppar agents |
RU2449790C2 (ru) * | 2007-03-27 | 2012-05-10 | Омерос Корпорейшен | Использование ингибиторов pde7 для лечения нарушений движения |
US8637528B2 (en) * | 2007-03-27 | 2014-01-28 | Omeros Corporation | Use of PDE7 inhibitors for the treatment of movement disorders |
WO2010093191A2 (fr) * | 2009-02-13 | 2010-08-19 | Lg Life Sciences Ltd. | Nouveaux composés efficaces en tant qu'inhibiteurs de xanthine oxydase, leur procédé de préparation et composition pharmaceutique les contenant |
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-
2001
- 2001-12-24 DE DE10163991A patent/DE10163991A1/de not_active Withdrawn
-
2002
- 2002-11-08 KR KR10-2004-7010053A patent/KR20040071252A/ko not_active Application Discontinuation
- 2002-11-08 CN CNA028260341A patent/CN1608067A/zh active Pending
- 2002-11-08 MX MXPA04006235A patent/MXPA04006235A/es not_active Application Discontinuation
- 2002-11-08 AU AU2002367090A patent/AU2002367090B2/en not_active Ceased
- 2002-11-08 RU RU2004122924/04A patent/RU2004122924A/ru not_active Application Discontinuation
- 2002-11-08 CA CA2471538A patent/CA2471538C/fr not_active Expired - Fee Related
- 2002-11-08 DE DE50212917T patent/DE50212917D1/de not_active Expired - Lifetime
- 2002-11-08 BR BR0215308-4A patent/BR0215308A/pt not_active IP Right Cessation
- 2002-11-08 PL PL02369728A patent/PL369728A1/xx unknown
- 2002-11-08 JP JP2003556412A patent/JP2005520801A/ja active Pending
- 2002-11-08 US US10/500,040 patent/US7498334B2/en not_active Expired - Fee Related
- 2002-11-08 WO PCT/EP2002/012533 patent/WO2003055882A1/fr active Application Filing
- 2002-11-08 HU HU0402216A patent/HUP0402216A2/hu unknown
- 2002-11-08 AT AT02805744T patent/ATE411316T1/de not_active IP Right Cessation
- 2002-11-08 ES ES02805744T patent/ES2314132T3/es not_active Expired - Lifetime
- 2002-11-08 EP EP02805744A patent/EP1458722B1/fr not_active Expired - Lifetime
- 2002-12-20 AR ARP020105061A patent/AR037972A1/es not_active Application Discontinuation
-
2004
- 2004-07-22 ZA ZA200405859A patent/ZA200405859B/en unknown
Also Published As
Publication number | Publication date |
---|---|
KR20040071252A (ko) | 2004-08-11 |
CA2471538A1 (fr) | 2003-07-10 |
BR0215308A (pt) | 2004-12-21 |
AR037972A1 (es) | 2004-12-22 |
DE50212917D1 (de) | 2008-11-27 |
CA2471538C (fr) | 2011-03-22 |
ATE411316T1 (de) | 2008-10-15 |
US7498334B2 (en) | 2009-03-03 |
JP2005520801A (ja) | 2005-07-14 |
DE10163991A1 (de) | 2003-07-03 |
WO2003055882A1 (fr) | 2003-07-10 |
US20050059686A1 (en) | 2005-03-17 |
CN1608067A (zh) | 2005-04-20 |
AU2002367090A1 (en) | 2003-07-15 |
EP1458722B1 (fr) | 2008-10-15 |
MXPA04006235A (es) | 2004-11-01 |
RU2004122924A (ru) | 2005-05-27 |
HUP0402216A2 (hu) | 2005-02-28 |
AU2002367090B2 (en) | 2008-11-13 |
ES2314132T3 (es) | 2009-03-16 |
PL369728A1 (en) | 2005-05-02 |
EP1458722A1 (fr) | 2004-09-22 |
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