ZA200100038B - Oxazolidinones to treat eye infections. - Google Patents
Oxazolidinones to treat eye infections. Download PDFInfo
- Publication number
- ZA200100038B ZA200100038B ZA200100038A ZA200100038A ZA200100038B ZA 200100038 B ZA200100038 B ZA 200100038B ZA 200100038 A ZA200100038 A ZA 200100038A ZA 200100038 A ZA200100038 A ZA 200100038A ZA 200100038 B ZA200100038 B ZA 200100038B
- Authority
- ZA
- South Africa
- Prior art keywords
- treating
- infection according
- ophthalmic infection
- ophthalmic
- oxazolidinone
- Prior art date
Links
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title claims description 35
- 208000001860 Eye Infections Diseases 0.000 title description 3
- 208000011323 eye infectious disease Diseases 0.000 title description 3
- 208000015181 infectious disease Diseases 0.000 claims description 37
- 238000000034 method Methods 0.000 claims description 26
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- 239000000203 mixture Substances 0.000 claims description 22
- 239000000243 solution Substances 0.000 claims description 19
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 10
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- 125000004105 2-pyridyl group Chemical group N1=C([*])C([H])=C([H])C([H])=C1[H] 0.000 claims description 4
- 125000000175 2-thienyl group Chemical group S1C([*])=C([H])C([H])=C1[H] 0.000 claims description 4
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Classifications
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Ophthalmology & Optometry (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9276598P | 1998-07-14 | 1998-07-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200100038B true ZA200100038B (en) | 2002-01-02 |
Family
ID=22235050
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200100038A ZA200100038B (en) | 1998-07-14 | 2001-01-02 | Oxazolidinones to treat eye infections. |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US6337329B1 (ja) |
| EP (1) | EP1096934B1 (ja) |
| JP (1) | JP2002520359A (ja) |
| KR (1) | KR20010079530A (ja) |
| CN (1) | CN1305374A (ja) |
| AT (1) | ATE304886T1 (ja) |
| AU (1) | AU740781B2 (ja) |
| BG (1) | BG64666B1 (ja) |
| BR (1) | BR9912004A (ja) |
| CA (1) | CA2334811A1 (ja) |
| DE (1) | DE69927380T2 (ja) |
| DK (1) | DK1096934T3 (ja) |
| EA (1) | EA003274B1 (ja) |
| EE (1) | EE200100026A (ja) |
| ES (1) | ES2249020T3 (ja) |
| HU (1) | HUP0102836A3 (ja) |
| ID (1) | ID27276A (ja) |
| IL (1) | IL140769A0 (ja) |
| NO (1) | NO20010202D0 (ja) |
| NZ (1) | NZ509375A (ja) |
| PL (1) | PL345544A1 (ja) |
| PT (1) | PT1096934E (ja) |
| SG (1) | SG125079A1 (ja) |
| SK (1) | SK20332000A3 (ja) |
| TR (1) | TR200100066T2 (ja) |
| WO (1) | WO2000003710A1 (ja) |
| ZA (1) | ZA200100038B (ja) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR020660A1 (es) * | 1998-09-30 | 2002-05-22 | Alcon Lab Inc | Composiciones antibioticas para el tratamiento de ojos, oidos y nariz |
| JP2003529544A (ja) * | 1999-09-13 | 2003-10-07 | インサイト・ビジョン・インコーポレイテッド | 眼感染症の予防たのための局所処置 |
| US6562820B2 (en) * | 2000-07-05 | 2003-05-13 | Pharmacia & Upjohn Company | Method for treatment and prevention of mastitis |
| PE20020300A1 (es) * | 2000-08-22 | 2002-05-10 | Pharmacia Corp | Composicion de solucion de un farmaco antibiotico a base de oxazolidinona con mejoramiento de la carga de farmaco |
| PE20020578A1 (es) * | 2000-10-10 | 2002-08-14 | Upjohn Co | Una composicion de antibiotico topico para el tratamiento de infecciones oculares |
| US7125568B2 (en) | 2001-08-23 | 2006-10-24 | Sung Michael T | Lipophilic drug compositions |
| US20030069235A1 (en) * | 2001-09-14 | 2003-04-10 | J. Greg Slatter | Treatment for ocular infections |
| MXPA04008173A (es) * | 2002-02-22 | 2004-11-26 | Pharmacia Corp | Formulaciones de farmaco antibiotico oftalmico que contienen un compuesto de ciclodextrina y cloruro de cetil piridinio. |
| TW201043267A (en) * | 2009-03-19 | 2010-12-16 | Intervet Int Bv | In situ constituting a vaccine for administration to a predetermined herd of animals |
| CN101766628B (zh) * | 2010-01-20 | 2012-07-04 | 广东宏盈科技有限公司 | 一种眼科外用抗细菌感染药物 |
| WO2014043576A1 (en) * | 2012-09-13 | 2014-03-20 | Starpharma Pty Limited | Method of treatment or prophylaxis of infections of the eye |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5164510A (en) | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
| US5231188A (en) | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
| KR100257418B1 (ko) * | 1991-11-01 | 2000-05-15 | 로렌스 티. 마이젠헬더 | 치환된 아릴-및 헤테로아릴-페닐옥사졸리디논 |
| US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
| DK0730591T3 (da) | 1993-11-22 | 2000-01-31 | Upjohn Co | Estere af substituerede hydroxyacetyl-piperazin-phenyl-oxazolidinoner |
| DE4425612A1 (de) * | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
| DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
| HUP9901628A3 (en) * | 1996-05-31 | 2002-11-28 | Scripps Research Inst | Methods and compositions useful for inhibition of alfa v beta5 mediated angiogenesis |
-
1999
- 1999-07-07 US US09/349,430 patent/US6337329B1/en not_active Expired - Fee Related
- 1999-07-07 CA CA002334811A patent/CA2334811A1/en not_active Abandoned
- 1999-07-07 PL PL99345544A patent/PL345544A1/xx unknown
- 1999-07-07 AT AT99933483T patent/ATE304886T1/de not_active IP Right Cessation
- 1999-07-07 ID IDW20002687A patent/ID27276A/id unknown
- 1999-07-07 DE DE69927380T patent/DE69927380T2/de not_active Expired - Fee Related
- 1999-07-07 TR TR2001/00066T patent/TR200100066T2/xx unknown
- 1999-07-07 NZ NZ509375A patent/NZ509375A/en unknown
- 1999-07-07 EP EP99933483A patent/EP1096934B1/en not_active Expired - Lifetime
- 1999-07-07 SK SK2033-2000A patent/SK20332000A3/sk unknown
- 1999-07-07 KR KR1020017000567A patent/KR20010079530A/ko not_active Application Discontinuation
- 1999-07-07 BR BR9912004-6A patent/BR9912004A/pt not_active Application Discontinuation
- 1999-07-07 IL IL14076999A patent/IL140769A0/xx unknown
- 1999-07-07 CN CN99807427A patent/CN1305374A/zh active Pending
- 1999-07-07 DK DK99933483T patent/DK1096934T3/da active
- 1999-07-07 AU AU49530/99A patent/AU740781B2/en not_active Ceased
- 1999-07-07 SG SG200300091A patent/SG125079A1/en unknown
- 1999-07-07 HU HU0102836A patent/HUP0102836A3/hu unknown
- 1999-07-07 EA EA200100133A patent/EA003274B1/ru unknown
- 1999-07-07 JP JP2000559845A patent/JP2002520359A/ja not_active Withdrawn
- 1999-07-07 EE EEP200100026A patent/EE200100026A/xx unknown
- 1999-07-07 PT PT99933483T patent/PT1096934E/pt unknown
- 1999-07-07 ES ES99933483T patent/ES2249020T3/es not_active Expired - Lifetime
- 1999-07-07 WO PCT/US1999/012367 patent/WO2000003710A1/en not_active Application Discontinuation
-
2001
- 2001-01-02 ZA ZA200100038A patent/ZA200100038B/en unknown
- 2001-01-10 BG BG105142A patent/BG64666B1/bg unknown
- 2001-01-12 NO NO20010202A patent/NO20010202D0/no not_active Application Discontinuation
- 2001-09-19 US US09/955,679 patent/US6740652B2/en not_active Expired - Fee Related
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