ZA200100038B - Oxazolidinones to treat eye infections. - Google Patents
Oxazolidinones to treat eye infections. Download PDFInfo
- Publication number
- ZA200100038B ZA200100038B ZA200100038A ZA200100038A ZA200100038B ZA 200100038 B ZA200100038 B ZA 200100038B ZA 200100038 A ZA200100038 A ZA 200100038A ZA 200100038 A ZA200100038 A ZA 200100038A ZA 200100038 B ZA200100038 B ZA 200100038B
- Authority
- ZA
- South Africa
- Prior art keywords
- treating
- infection according
- ophthalmic infection
- ophthalmic
- oxazolidinone
- Prior art date
Links
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title claims description 35
- 208000001860 Eye Infections Diseases 0.000 title description 3
- 208000011323 eye infectious disease Diseases 0.000 title description 3
- 208000015181 infectious disease Diseases 0.000 claims description 37
- 238000000034 method Methods 0.000 claims description 26
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- 239000000203 mixture Substances 0.000 claims description 22
- 239000000243 solution Substances 0.000 claims description 19
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims description 10
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- 125000004105 2-pyridyl group Chemical group N1=C([*])C([H])=C([H])C([H])=C1[H] 0.000 claims description 4
- 125000000175 2-thienyl group Chemical group S1C([*])=C([H])C([H])=C1[H] 0.000 claims description 4
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Classifications
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9276598P | 1998-07-14 | 1998-07-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200100038B true ZA200100038B (en) | 2002-01-02 |
Family
ID=22235050
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200100038A ZA200100038B (en) | 1998-07-14 | 2001-01-02 | Oxazolidinones to treat eye infections. |
Country Status (27)
| Country | Link |
|---|---|
| US (2) | US6337329B1 (de) |
| EP (1) | EP1096934B1 (de) |
| JP (1) | JP2002520359A (de) |
| KR (1) | KR20010079530A (de) |
| CN (1) | CN1305374A (de) |
| AT (1) | ATE304886T1 (de) |
| AU (1) | AU740781B2 (de) |
| BG (1) | BG64666B1 (de) |
| BR (1) | BR9912004A (de) |
| CA (1) | CA2334811A1 (de) |
| DE (1) | DE69927380T2 (de) |
| DK (1) | DK1096934T3 (de) |
| EA (1) | EA003274B1 (de) |
| EE (1) | EE200100026A (de) |
| ES (1) | ES2249020T3 (de) |
| HU (1) | HUP0102836A3 (de) |
| ID (1) | ID27276A (de) |
| IL (1) | IL140769A0 (de) |
| NO (1) | NO20010202D0 (de) |
| NZ (1) | NZ509375A (de) |
| PL (1) | PL345544A1 (de) |
| PT (1) | PT1096934E (de) |
| SG (1) | SG125079A1 (de) |
| SK (1) | SK20332000A3 (de) |
| TR (1) | TR200100066T2 (de) |
| WO (1) | WO2000003710A1 (de) |
| ZA (1) | ZA200100038B (de) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR020660A1 (es) * | 1998-09-30 | 2002-05-22 | Alcon Lab Inc | Composiciones antibioticas para el tratamiento de ojos, oidos y nariz |
| ATE337002T1 (de) * | 1999-09-13 | 2006-09-15 | Insite Vision Inc | Topische behandlung zur vorbeugung von augeninfektionen |
| US6562820B2 (en) | 2000-07-05 | 2003-05-13 | Pharmacia & Upjohn Company | Method for treatment and prevention of mastitis |
| PE20020300A1 (es) * | 2000-08-22 | 2002-05-10 | Pharmacia Corp | Composicion de solucion de un farmaco antibiotico a base de oxazolidinona con mejoramiento de la carga de farmaco |
| AR031135A1 (es) * | 2000-10-10 | 2003-09-10 | Upjohn Co | Composiciones de antibiotico topico para el tratamiento de infecciones oculares |
| US7125568B2 (en) | 2001-08-23 | 2006-10-24 | Sung Michael T | Lipophilic drug compositions |
| US20030069235A1 (en) * | 2001-09-14 | 2003-04-10 | J. Greg Slatter | Treatment for ocular infections |
| JP2005521691A (ja) * | 2002-02-22 | 2005-07-21 | ファルマシア・コーポレーション | シクロデキストリン化合物及び塩化セチルピリジニウムを含有する眼科用抗菌性薬物製剤 |
| TW201043267A (en) * | 2009-03-19 | 2010-12-16 | Intervet Int Bv | In situ constituting a vaccine for administration to a predetermined herd of animals |
| CN101766628B (zh) * | 2010-01-20 | 2012-07-04 | 广东宏盈科技有限公司 | 一种眼科外用抗细菌感染药物 |
| EP2895161B1 (de) * | 2012-09-13 | 2017-05-03 | Starpharma Pty Limited | Verfahren zur behandlung oder prophylaxe von infektionen des auges |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5164510A (en) * | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
| US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
| AU667198B2 (en) * | 1991-11-01 | 1996-03-14 | Pharmacia & Upjohn Company | Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents |
| US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
| JP3698724B2 (ja) | 1993-11-22 | 2005-09-21 | ファルマシア・アンド・アップジョン・カンパニー | 置換−ヒドロキシアセチルピペラジンフェニルオキサゾリジノンのエステル |
| DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
| DE4425612A1 (de) | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
| WO1997045137A1 (en) * | 1996-05-31 | 1997-12-04 | The Scripps Research Institute | Methods and compositions useful for inhibition of angiogenesis |
-
1999
- 1999-07-07 AU AU49530/99A patent/AU740781B2/en not_active Ceased
- 1999-07-07 IL IL14076999A patent/IL140769A0/xx unknown
- 1999-07-07 WO PCT/US1999/012367 patent/WO2000003710A1/en not_active Application Discontinuation
- 1999-07-07 BR BR9912004-6A patent/BR9912004A/pt not_active Application Discontinuation
- 1999-07-07 SK SK2033-2000A patent/SK20332000A3/sk unknown
- 1999-07-07 ES ES99933483T patent/ES2249020T3/es not_active Expired - Lifetime
- 1999-07-07 EE EEP200100026A patent/EE200100026A/xx unknown
- 1999-07-07 ID IDW20002687A patent/ID27276A/id unknown
- 1999-07-07 EP EP99933483A patent/EP1096934B1/de not_active Expired - Lifetime
- 1999-07-07 CN CN99807427A patent/CN1305374A/zh active Pending
- 1999-07-07 NZ NZ509375A patent/NZ509375A/en unknown
- 1999-07-07 JP JP2000559845A patent/JP2002520359A/ja not_active Withdrawn
- 1999-07-07 KR KR1020017000567A patent/KR20010079530A/ko not_active Application Discontinuation
- 1999-07-07 AT AT99933483T patent/ATE304886T1/de not_active IP Right Cessation
- 1999-07-07 DK DK99933483T patent/DK1096934T3/da active
- 1999-07-07 CA CA002334811A patent/CA2334811A1/en not_active Abandoned
- 1999-07-07 US US09/349,430 patent/US6337329B1/en not_active Expired - Fee Related
- 1999-07-07 DE DE69927380T patent/DE69927380T2/de not_active Expired - Fee Related
- 1999-07-07 TR TR2001/00066T patent/TR200100066T2/xx unknown
- 1999-07-07 EA EA200100133A patent/EA003274B1/ru unknown
- 1999-07-07 SG SG200300091A patent/SG125079A1/en unknown
- 1999-07-07 PL PL99345544A patent/PL345544A1/xx unknown
- 1999-07-07 HU HU0102836A patent/HUP0102836A3/hu unknown
- 1999-07-07 PT PT99933483T patent/PT1096934E/pt unknown
-
2001
- 2001-01-02 ZA ZA200100038A patent/ZA200100038B/en unknown
- 2001-01-10 BG BG105142A patent/BG64666B1/bg unknown
- 2001-01-12 NO NO20010202A patent/NO20010202D0/no not_active Application Discontinuation
- 2001-09-19 US US09/955,679 patent/US6740652B2/en not_active Expired - Fee Related
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