ZA200007448B - Inhibitors of transcription factor NF-kB. - Google Patents
Inhibitors of transcription factor NF-kB. Download PDFInfo
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- ZA200007448B ZA200007448B ZA200007448A ZA200007448A ZA200007448B ZA 200007448 B ZA200007448 B ZA 200007448B ZA 200007448 A ZA200007448 A ZA 200007448A ZA 200007448 A ZA200007448 A ZA 200007448A ZA 200007448 B ZA200007448 B ZA 200007448B
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- benzalindanone
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
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- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4462—Non condensed piperidines, e.g. piperocaine only substituted in position 3
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Dermatology (AREA)
- Virology (AREA)
- Pulmonology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Oncology (AREA)
- Hospice & Palliative Care (AREA)
- Toxicology (AREA)
- Transplantation (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9001698P | 1998-06-19 | 1998-06-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200007448B true ZA200007448B (en) | 2001-12-12 |
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| Application Number | Title | Priority Date | Filing Date |
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| ZA200007448A ZA200007448B (en) | 1998-06-19 | 2000-12-13 | Inhibitors of transcription factor NF-kB. |
Country Status (17)
| Country | Link |
|---|---|
| EP (1) | EP1085872A4 (zh) |
| JP (1) | JP2002518333A (zh) |
| KR (1) | KR20010052990A (zh) |
| CN (1) | CN1306428A (zh) |
| AR (1) | AR019871A1 (zh) |
| AU (1) | AU4699699A (zh) |
| BR (1) | BR9911151A (zh) |
| CA (1) | CA2335293A1 (zh) |
| CO (1) | CO5080752A1 (zh) |
| CZ (1) | CZ20004760A3 (zh) |
| HU (1) | HUP0102492A2 (zh) |
| IL (1) | IL140324A0 (zh) |
| NO (1) | NO20006452L (zh) |
| PL (1) | PL345577A1 (zh) |
| TR (1) | TR200003779T2 (zh) |
| WO (1) | WO1999065495A1 (zh) |
| ZA (1) | ZA200007448B (zh) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002509431A (ja) | 1996-12-23 | 2002-03-26 | イミュネックス・コーポレーション | ＮＦ−κＢのレセプター活性化因子−レセプターはＴＮＦレセプタースーパーファミリーの一員である− |
| US6316408B1 (en) | 1997-04-16 | 2001-11-13 | Amgen Inc. | Methods of use for osetoprotegerin binding protein receptors |
| AU762574B2 (en) | 1998-05-14 | 2003-06-26 | Immunex Corporation | Method of inhibiting osteoclast activity |
| EP1250137B1 (en) * | 2000-01-24 | 2007-08-15 | Genzyme Corporation | Jak/stat pathway inhibitors and the use thereof for the treatment of primary generalized osteoarthritis |
| US20060148732A1 (en) * | 2000-11-17 | 2006-07-06 | Gutterman Jordan U | Inhibition of NF-kappaB by triterpene compositions |
| US7425580B2 (en) | 2004-05-19 | 2008-09-16 | Wyeth | (Diaryl-methyl)-malononitriles and their use as estrogen receptor ligands |
| JP2009526855A (ja) | 2006-02-16 | 2009-07-23 | ミレニアム・ファーマシューティカルズ・インコーポレイテッド | アルファカルボリンおよびその使用 |
| WO2010038465A1 (ja) | 2008-10-02 | 2010-04-08 | 旭化成ファーマ株式会社 | ８位置換イソキノリン誘導体及びその用途 |
| US9127016B2 (en) | 2009-03-20 | 2015-09-08 | University of Pittsburgh—of the Commonwealth System of Higher Education | Small molecule inhibitors of Dusp6 and uses therefor |
| EP2461806A4 (en) * | 2009-07-31 | 2012-12-26 | Us Health | SMALL ANTI-ANGIOGENIC MOLECULES AND METHODS OF USE |
| WO2012109527A2 (en) | 2011-02-10 | 2012-08-16 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Class of hdac inhibitors expands the renal progenitor cells population and improves the rate of recovery from acute kidney injury |
| WO2014071000A1 (en) | 2012-10-31 | 2014-05-08 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Class of hdac inhibitors expands the renal progenitor cells population and improves the rate of recovery from acute kidney injury |
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1998
- 1998-06-18 HU HU0102492A patent/HUP0102492A2/hu unknown
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1999
- 1999-06-17 CO CO99037918A patent/CO5080752A1/es unknown
- 1999-06-18 TR TR2000/03779T patent/TR200003779T2/xx unknown
- 1999-06-18 IL IL14032499A patent/IL140324A0/xx unknown
- 1999-06-18 AU AU46996/99A patent/AU4699699A/en not_active Abandoned
- 1999-06-18 CA CA002335293A patent/CA2335293A1/en not_active Abandoned
- 1999-06-18 BR BR9911151-9A patent/BR9911151A/pt not_active Application Discontinuation
- 1999-06-18 JP JP2000554375A patent/JP2002518333A/ja not_active Withdrawn
- 1999-06-18 PL PL99345577A patent/PL345577A1/xx not_active Application Discontinuation
- 1999-06-18 CN CN99807572A patent/CN1306428A/zh active Pending
- 1999-06-18 KR KR1020007014385A patent/KR20010052990A/ko not_active Application Discontinuation
- 1999-06-18 WO PCT/US1999/013897 patent/WO1999065495A1/en not_active Application Discontinuation
- 1999-06-18 AR ARP990102952A patent/AR019871A1/es unknown
- 1999-06-18 CZ CZ20004760A patent/CZ20004760A3/cs unknown
- 1999-06-18 EP EP99930459A patent/EP1085872A4/en not_active Withdrawn
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2000
- 2000-12-13 ZA ZA200007448A patent/ZA200007448B/en unknown
- 2000-12-18 NO NO20006452A patent/NO20006452L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NO20006452L (no) | 2001-02-16 |
| BR9911151A (pt) | 2001-03-06 |
| CN1306428A (zh) | 2001-08-01 |
| CA2335293A1 (en) | 1999-12-23 |
| HUP0102492A2 (hu) | 2001-11-28 |
| EP1085872A1 (en) | 2001-03-28 |
| TR200003779T2 (tr) | 2001-06-21 |
| EP1085872A4 (en) | 2003-04-16 |
| AU4699699A (en) | 2000-01-05 |
| IL140324A0 (en) | 2002-02-10 |
| WO1999065495A1 (en) | 1999-12-23 |
| JP2002518333A (ja) | 2002-06-25 |
| KR20010052990A (ko) | 2001-06-25 |
| PL345577A1 (en) | 2001-12-17 |
| CZ20004760A3 (cs) | 2001-08-15 |
| AR019871A1 (es) | 2002-03-20 |
| NO20006452D0 (no) | 2000-12-18 |
| CO5080752A1 (es) | 2001-09-25 |
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