YU46177B - Postupak za dobijanje 2-okso-1-//(supstituisanih sulfonil) amino/karbonil/azetidina - Google Patents

Postupak za dobijanje 2-okso-1-//(supstituisanih sulfonil) amino/karbonil/azetidina

Info

Publication number
YU46177B
YU46177B YU165986A YU165986A YU46177B YU 46177 B YU46177 B YU 46177B YU 165986 A YU165986 A YU 165986A YU 165986 A YU165986 A YU 165986A YU 46177 B YU46177 B YU 46177B
Authority
YU
Yugoslavia
Prior art keywords
amino
azetidine
oxo
carbonyl
preparation
Prior art date
Application number
YU165986A
Other languages
English (en)
Serbo-Croatian (sh)
Other versions
YU165986A (en
Inventor
H. Breuer
U. Treuner
W. Koster
R. Zahler
Original Assignee
E.R. Squibb & Sons Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by E.R. Squibb & Sons Inc. filed Critical E.R. Squibb & Sons Inc.
Publication of YU165986A publication Critical patent/YU165986A/xx
Publication of YU46177B publication Critical patent/YU46177B/sh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
YU165986A 1985-09-26 1986-09-26 Postupak za dobijanje 2-okso-1-//(supstituisanih sulfonil) amino/karbonil/azetidina YU46177B (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US78047985A 1985-09-26 1985-09-26

Publications (2)

Publication Number Publication Date
YU165986A YU165986A (en) 1988-06-30
YU46177B true YU46177B (sh) 1993-05-28

Family

ID=25119699

Family Applications (1)

Application Number Title Priority Date Filing Date
YU165986A YU46177B (sh) 1985-09-26 1986-09-26 Postupak za dobijanje 2-okso-1-//(supstituisanih sulfonil) amino/karbonil/azetidina

Country Status (31)

Country Link
JP (1) JPS6284082A (cs)
KR (1) KR900001013B1 (cs)
CN (1) CN86106980A (cs)
AT (1) ATA257986A (cs)
AU (1) AU600912B2 (cs)
BE (1) BE905502A (cs)
CA (1) CA1308719C (cs)
CH (1) CH670828A5 (cs)
DD (1) DD250121A5 (cs)
DE (1) DE3632876A1 (cs)
DK (1) DK460386A (cs)
EG (1) EG18314A (cs)
ES (1) ES2001995A6 (cs)
FI (1) FI863890A7 (cs)
FR (1) FR2587700B1 (cs)
GB (1) GB2181130B (cs)
GR (1) GR862449B (cs)
HU (1) HU198044B (cs)
IE (1) IE59686B1 (cs)
IL (1) IL80160A (cs)
IT (1) IT1214533B (cs)
LU (1) LU86611A1 (cs)
NL (1) NL8602446A (cs)
NO (1) NO863837L (cs)
NZ (1) NZ217704A (cs)
PH (1) PH23315A (cs)
PL (1) PL151546B1 (cs)
PT (1) PT83440B (cs)
SE (1) SE8604089L (cs)
YU (1) YU46177B (cs)
ZA (1) ZA867373B (cs)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0308416A1 (en) * 1986-05-23 1989-03-29 The Upjohn Company N-1 substituted sulfonylaminocarbonyl, c-4 substituted monobactams
ATE66225T1 (de) * 1987-02-11 1991-08-15 Upjohn Co Neue n-1 substituierte beta-lactame als antibiotika.
US5006650A (en) * 1987-02-11 1991-04-09 The Upjohn Company Novel N-1 substituted beta-lactams as antibiotics
EP0357604A1 (en) * 1987-02-27 1990-03-14 The Upjohn Company Antibiotic beta-lactams containing a pyridone carboxylic acid or acid derivative
CA1317298C (en) * 1987-03-03 1993-05-04 Upjohn Company (The) Antibiotic sulfonylaminocarbonyl activated .beta.-lactams
US4762922A (en) * 1987-07-01 1988-08-09 Squibb Corporation 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4772693A (en) * 1987-07-01 1988-09-20 E. R. Squibb & Sons, Inc. 2-oxo-1-((Substituted sulfonyl)amino)-carbonyl)azetidines
US5015737A (en) * 1987-07-22 1991-05-14 The Upjohn Company Therapeutically useful beta-lactams
EP0368908A1 (en) * 1987-07-22 1990-05-23 The Upjohn Company THERAPEUTICALLY USEFUL $g(b)-LACTAMS
US4777252A (en) * 1987-08-13 1988-10-11 E. R. Squibb & Sons, Inc. 2-oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
US4889930A (en) * 1987-12-21 1989-12-26 E. R. Squibb & Sons, Inc. Process for making 2-oxo-1-((substituted sulfonyl)amino)carbonzyl)azetidines and intermediates used therein
US4871841A (en) * 1987-12-23 1989-10-03 E. R. Squibb & Sons, Inc. 2-Oxo-1-[[(substituted sulfonyl)amino]-carbonyl]azetidines
JPH01290674A (ja) * 1988-04-04 1989-11-22 E R Squibb & Sons Inc アゼチジニル誘導体
US4959470A (en) * 1988-08-17 1990-09-25 E. R. Squibb & Sons, Inc. 2-oxo-[[(substituted sulfonyl)-amino]carbonyl]-azetidines
ES2133376T3 (es) * 1992-12-23 1999-09-16 Novartis Ag Derivados de imidazol y su uso como agentes agroquimicos.
DE69405535T2 (de) * 1994-03-11 1998-04-02 Agfa Gevaert Nv Photographisches Material, das einen neuen Typ eines Hydrazides enthält
JP4792974B2 (ja) * 2003-12-25 2011-10-12 小野薬品工業株式会社 アゼチジン環化合物およびその医薬
GB201111704D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Novel compounds
GB201111705D0 (en) 2011-07-07 2011-08-24 Takeda Pharmaceutical Compounds and their use
JO3115B1 (ar) 2011-08-22 2017-09-20 Takeda Pharmaceuticals Co مركبات بيريدازينون واستخدامها كمثبطات daao
UA111861C2 (uk) 2011-11-15 2016-06-24 Такеда Фармасьютікал Компані Лімітед Ароматична гетероциклічна сполука дигідрокси
GB201222711D0 (en) 2012-12-17 2013-01-30 Takeda Pharmaceutical Novel compounds
CN106986820B (zh) * 2017-02-24 2019-05-21 浙江工商大学 多功能的羟基吡啶酮衍生物及其水合物的制备法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ199981A (en) * 1981-04-09 1985-08-16 Squibb & Sons Inc 2-oxo-1-(((substituted sulphonyl)amino)carbonyl)azetidines
CA1272726C (en) * 1982-01-04 1990-08-14 2-oxo-1-(aminocarbonylaminosulfonyl- aminocarbonyl)azetidines
US4939253A (en) * 1982-08-04 1990-07-03 E. R. Squibb & Sons, Inc. 2-oxoazetidin-1-yloxy acetic acids and analogs
US4801705A (en) * 1986-06-23 1989-01-31 E. R. Squibb & Sons, Inc. 2-oxo-1-(((substituted sulfonyl)amino)-carbonyl)azetidines

Also Published As

Publication number Publication date
AU6315686A (en) 1987-04-02
PL261575A1 (en) 1988-07-21
GR862449B (en) 1987-01-27
GB2181130A (en) 1987-04-15
EG18314A (en) 1993-02-28
PL151546B1 (en) 1990-09-28
CH670828A5 (cs) 1989-07-14
PT83440A (pt) 1986-10-01
DE3632876A1 (de) 1987-04-02
SE8604089D0 (sv) 1986-09-26
DD250121A5 (de) 1987-09-30
SE8604089L (sv) 1987-03-27
KR870003101A (ko) 1987-04-15
HUT44535A (en) 1988-03-28
NO863837D0 (no) 1986-09-26
GB2181130B (en) 1989-09-20
LU86611A1 (fr) 1987-04-02
IL80160A (en) 1991-04-15
PH23315A (en) 1989-07-14
BE905502A (fr) 1987-01-16
GB8623151D0 (en) 1986-10-29
IL80160A0 (en) 1986-12-31
NL8602446A (nl) 1987-04-16
ZA867373B (en) 1987-05-27
IT8621834A0 (it) 1986-09-26
NZ217704A (en) 1989-02-24
CA1308719C (en) 1992-10-13
CN86106980A (zh) 1987-04-08
DK460386D0 (da) 1986-09-26
FR2587700B1 (fr) 1988-09-16
DK460386A (da) 1987-03-27
AU600912B2 (en) 1990-08-30
ES2001995A6 (es) 1988-07-01
PT83440B (pt) 1989-05-12
JPS6284082A (ja) 1987-04-17
YU165986A (en) 1988-06-30
FI863890A7 (fi) 1987-03-27
IE862547L (en) 1987-03-26
FI863890A0 (fi) 1986-09-26
KR900001013B1 (ko) 1990-02-24
ATA257986A (de) 1994-07-15
FR2587700A1 (fr) 1987-03-27
HU198044B (en) 1989-07-28
IT1214533B (it) 1990-01-18
NO863837L (no) 1987-03-27
IE59686B1 (en) 1994-03-23

Similar Documents

Publication Publication Date Title
YU46177B (sh) Postupak za dobijanje 2-okso-1-//(supstituisanih sulfonil) amino/karbonil/azetidina
YU46916B (sh) Postupak za dobijanje kalcijum nezavisnih camp inhibitora fosfodiesteraze
ES2054826T3 (es) Peptidos con actividad inhibidora de colagenasa.
WO2005007625A3 (en) Heterocyclic amides with anti-tuberculosis activity
GB2091723B (en) Derivatives of 2-oxoazetidine-1-sulphonic acid
AU6516986A (en) New 3-oxadiazole and 3-carboxylic acid ester beta-carboline derivatives, their production and their use as drugs
DE68906200D1 (de) Kondensierte pyrazol-3-oxo-propannitril-derivate und verfahren zu deren herstellung.
DE68924556D1 (de) N-(N-(Tetrahydropyrido[2,3-d]pyrimidinylmethyl)-aminomethylbenzoyl)glutaminsäure-Derivate.
EP0533951A4 (en) Novel oxazinone derivative
BG60267B2 (bg) Метод за получаване на производни на амидоксим
TW238304B (en) A process for the preparation of 1-substituted-5(4H)-tetrazolinones
ATE204880T1 (de) N-acyldipeptide, und pharmazeutische präparate davon
HRP20000609B1 (en) Process for the synthesis of hiv protease inhibitors
IT1213555B (it) 2 metiltiometildiidropiridine, un processo per laloro preparazione e composizioni farmaceutiche che le contengono.
ATE47135T1 (de) Antikonvulsive mittel.
ES8801650A1 (es) Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico.
FR2350341A1 (fr) Nouveaux derives de piperidine et leur methode de preparation
DE3781783D1 (de) N-alkyl-derivate von 2-amino-6,7-dimethoxytetralin, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzungen mit antihypertensiver wirkung.
DE3682360D1 (de) 2-propadienylpenicillin-derivate und zwischenprodukte.
SE8403349L (sv) Hetercykliska ettiksyraestrar
DE3679257D1 (de) 4-cyanopiperidine-derivate, herstellung und anwendung.
ES471702A1 (es) Procedimiento para la preparacion de derivados de amida de acido
DK248287D0 (da) Fremgangsmaade til fremstilling af chephalosporinderivater
DE69409799D1 (de) Herstellung von symmetrischen und unsymmetrischen disubstituierten n-cyandithioiminocarbonaten
TH13390A (cs)