YU176590A - Novi n-aril i n-heteroarilamid i karbamid derivati kao inhibitori acil koenzima a: holesterol acil transferaza (acat) - Google Patents

Novi n-aril i n-heteroarilamid i karbamid derivati kao inhibitori acil koenzima a: holesterol acil transferaza (acat)

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Publication number
YU176590A
YU176590A YU176590A YU176590A YU176590A YU 176590 A YU176590 A YU 176590A YU 176590 A YU176590 A YU 176590A YU 176590 A YU176590 A YU 176590A YU 176590 A YU176590 A YU 176590A
Authority
YU
Yugoslavia
Prior art keywords
heteroarylamide
acat
inhibitors
aryl
acyl
Prior art date
Application number
YU176590A
Other languages
English (en)
Inventor
P.A. Mccartny
F.J. Walker
E.S. Hamanaka
G. Chang
T. Truong
Original Assignee
Pfizer Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc. filed Critical Pfizer Inc.
Publication of YU176590A publication Critical patent/YU176590A/sh

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Opisani su novi N-aril- i N-heteroarilamid i karbamid derivati, jedinjenja formule I njihove farmaceutski prihvatljive soli, u kojoj Q i R1 su kao što je ovde gore definisano, i nove karboksilne kiseline i kiselinski halidni intermedijeri koji se upotrebljavaju za sinteze tih jedinjenja. Jedinjenja formule I su inhibitori acil koenzima A. holesterol aciltransferaza (ACAT) i ista se upotrebljavaju kao hipolipidemička i antiarterosklerotička sredstva.
YU176590A 1989-09-15 1990-09-14 Novi n-aril i n-heteroarilamid i karbamid derivati kao inhibitori acil koenzima a: holesterol acil transferaza (acat) YU176590A (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US50403389A 1989-09-15 1989-09-15

Publications (1)

Publication Number Publication Date
YU176590A true YU176590A (sh) 1993-05-28

Family

ID=47291544

Family Applications (1)

Application Number Title Priority Date Filing Date
YU176590A YU176590A (sh) 1989-09-15 1990-09-14 Novi n-aril i n-heteroarilamid i karbamid derivati kao inhibitori acil koenzima a: holesterol acil transferaza (acat)

Country Status (1)

Country Link
YU (1) YU176590A (sh)

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