WO2015027848A1 - Méthode pour administrer une formulation comportant du peramivir et/ou un dérivé correspondant - Google Patents
Méthode pour administrer une formulation comportant du peramivir et/ou un dérivé correspondant Download PDFInfo
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- WO2015027848A1 WO2015027848A1 PCT/CN2014/084836 CN2014084836W WO2015027848A1 WO 2015027848 A1 WO2015027848 A1 WO 2015027848A1 CN 2014084836 W CN2014084836 W CN 2014084836W WO 2015027848 A1 WO2015027848 A1 WO 2015027848A1
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- WIPO (PCT)
- Prior art keywords
- administration
- peramivir
- derivatives
- administration method
- inhalation
- Prior art date
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- 230000008520 organization Effects 0.000 description 1
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- 238000009520 phase I clinical trial Methods 0.000 description 1
- COLNVLDHVKWLRT-UHFFFAOYSA-N phenylalanine Natural products OC(=O)C(N)CC1=CC=CC=C1 COLNVLDHVKWLRT-UHFFFAOYSA-N 0.000 description 1
- 239000000244 polyoxyethylene sorbitan monooleate Substances 0.000 description 1
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- 229920000053 polysorbate 80 Polymers 0.000 description 1
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- 238000000926 separation method Methods 0.000 description 1
- SQVRNKJHWKZAKO-OQPLDHBCSA-N sialic acid Chemical compound CC(=O)N[C@@H]1[C@@H](O)C[C@@](O)(C(O)=O)OC1[C@H](O)[C@H](O)CO SQVRNKJHWKZAKO-OQPLDHBCSA-N 0.000 description 1
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- 239000011780 sodium chloride Substances 0.000 description 1
- 229960002668 sodium chloride Drugs 0.000 description 1
- 239000001509 sodium citrate Substances 0.000 description 1
- NLJMYIDDQXHKNR-UHFFFAOYSA-K sodium citrate Chemical compound O.O.[Na+].[Na+].[Na+].[O-]C(=O)CC(O)(CC([O-])=O)C([O-])=O NLJMYIDDQXHKNR-UHFFFAOYSA-K 0.000 description 1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0075—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a dry powder inhaler [DPI], e.g. comprising micronized drug mixed with lactose carrier particles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0078—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a nebulizer such as a jet nebulizer, ultrasonic nebulizer, e.g. in the form of aqueous drug solutions or dispersions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Pulmonology (AREA)
- Epidemiology (AREA)
- Otolaryngology (AREA)
- Virology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Dispersion Chemistry (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
L'invention concerne une méthode pour administrer une formulation comportant du péramivir et/ou un dérivé correspondant ; cette méthode permettant de traiter des refroidissements causés par un virus de la grippe ; et l'administration se faisant par l'intermédiaire de plus d'un ou de deux éléments parmi les éléments suivants : poudre sèche, insufflateur de poudre, inhalateur à doses quantifiées ou nébuliseur.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN201310376626.8 | 2013-08-26 | ||
| CN2013103766268A CN103446051A (zh) | 2013-08-26 | 2013-08-26 | 含有帕拉米韦和/或其衍生物制剂的给药方法 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| WO2015027848A1 true WO2015027848A1 (fr) | 2015-03-05 |
Family
ID=49729173
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PCT/CN2014/084836 WO2015027848A1 (fr) | 2013-08-26 | 2014-08-20 | Méthode pour administrer une formulation comportant du peramivir et/ou un dérivé correspondant |
Country Status (2)
| Country | Link |
|---|---|
| CN (1) | CN103446051A (fr) |
| WO (1) | WO2015027848A1 (fr) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3932400A4 (fr) * | 2019-02-25 | 2022-09-21 | Guangzhou Nanxin Pharmaceutical Co., Ltd. | Inhalant de type solution de péramivir et son procédé de préparation |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN106420621A (zh) * | 2016-10-09 | 2017-02-22 | 默栢瑞成都生物技术有限公司 | 帕拉米韦粉剂的制备方法 |
| CN111067879B (zh) * | 2020-01-20 | 2022-08-09 | 珠海瑞思普利医药科技有限公司 | 一种抗肿瘤组合物吸入粉雾剂及其制备方法 |
| CN111265499B (zh) * | 2020-02-17 | 2022-11-15 | 江苏艾立康医药科技有限公司 | 一种洛匹那韦吸入气雾剂及其制备方法 |
| CN113491678B (zh) * | 2020-04-07 | 2023-01-20 | 知和(山东)大药厂有限公司 | 一种盐酸阿比朵尔吸入剂及其制备方法 |
| CN111358773B (zh) * | 2020-04-10 | 2021-03-30 | 广州南鑫药业有限公司 | 一种帕拉米韦干粉吸入剂及其制备方法 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009143011A1 (fr) * | 2008-05-20 | 2009-11-26 | Novartis Ag | Compositions antivirales, procédés de fabrication et d’utilisation de ces compositions, et système de délivrance pulmonaire de ces compositions |
| WO2011035128A1 (fr) * | 2009-09-17 | 2011-03-24 | Mutual Pharmaceutical Company, Inc. | Procédé de traitement de l'asthme avec des agents antiviraux |
-
2013
- 2013-08-26 CN CN2013103766268A patent/CN103446051A/zh active Pending
-
2014
- 2014-08-20 WO PCT/CN2014/084836 patent/WO2015027848A1/fr active Application Filing
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2009143011A1 (fr) * | 2008-05-20 | 2009-11-26 | Novartis Ag | Compositions antivirales, procédés de fabrication et d’utilisation de ces compositions, et système de délivrance pulmonaire de ces compositions |
| WO2011035128A1 (fr) * | 2009-09-17 | 2011-03-24 | Mutual Pharmaceutical Company, Inc. | Procédé de traitement de l'asthme avec des agents antiviraux |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3932400A4 (fr) * | 2019-02-25 | 2022-09-21 | Guangzhou Nanxin Pharmaceutical Co., Ltd. | Inhalant de type solution de péramivir et son procédé de préparation |
Also Published As
| Publication number | Publication date |
|---|---|
| CN103446051A (zh) | 2013-12-18 |
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