WO2011074851A3 - Préparation pharmaceutique - Google Patents

Préparation pharmaceutique Download PDF

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Publication number
WO2011074851A3
WO2011074851A3 PCT/KR2010/008925 KR2010008925W WO2011074851A3 WO 2011074851 A3 WO2011074851 A3 WO 2011074851A3 KR 2010008925 W KR2010008925 W KR 2010008925W WO 2011074851 A3 WO2011074851 A3 WO 2011074851A3
Authority
WO
WIPO (PCT)
Prior art keywords
preparation
active ingredient
inner core
coating layer
pharmaceutical preparation
Prior art date
Application number
PCT/KR2010/008925
Other languages
English (en)
Korean (ko)
Other versions
WO2011074851A2 (fr
Inventor
이범진
풍 트란하렌
Original Assignee
㈜유라팜
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ㈜유라팜 filed Critical ㈜유라팜
Publication of WO2011074851A2 publication Critical patent/WO2011074851A2/fr
Publication of WO2011074851A3 publication Critical patent/WO2011074851A3/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/27Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • A61K9/2846Poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/286Polysaccharides, e.g. gums; Cyclodextrin
    • A61K9/2866Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Abstract

La présente invention concerne une préparation pharmaceutique comprenant : un noyau interne incluant un acidulant et du bambutérol ou l'un de ses sels de qualité pharmaceutique au titre de principe actif ; et une couche de revêtement destinée au revêtement de la surface du noyau interne, la couche de revêtement incluant à la fois un polymère pH-dépendant et un polymère pH-indépendant. Lorsque la préparation selon la présente invention est administrée par voie orale, la préparation libère le principe actif après l'écoulement d'un temps de retard prédéterminé après son passage de l'estomac à l'intestin d'un patient, ce qui permet d'obtenir des effets thérapeutiques pendant la période où les symptômes asthmatiques deviennent sévères.
PCT/KR2010/008925 2009-12-14 2010-12-14 Préparation pharmaceutique WO2011074851A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
KR1020090123838A KR101152977B1 (ko) 2009-12-14 2009-12-14 약제학적 제제
KR10-2009-0123838 2009-12-14

Publications (2)

Publication Number Publication Date
WO2011074851A2 WO2011074851A2 (fr) 2011-06-23
WO2011074851A3 true WO2011074851A3 (fr) 2011-11-03

Family

ID=44167850

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/KR2010/008925 WO2011074851A2 (fr) 2009-12-14 2010-12-14 Préparation pharmaceutique

Country Status (2)

Country Link
KR (1) KR101152977B1 (fr)
WO (1) WO2011074851A2 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103288670B (zh) * 2013-05-16 2014-11-05 南京医科大学第一附属医院 多羟基二苯甲酮衍生物及其应用
CN107668351A (zh) * 2017-10-20 2018-02-09 浙江耀飞生物科技有限公司 一种肠溶型复合饲料酸化剂

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5788987A (en) * 1997-01-29 1998-08-04 Poli Industria Chimica Spa Methods for treating early morning pathologies
WO2003057278A2 (fr) * 2002-01-04 2003-07-17 Ivax Research, Inc. Systeme d'apport de medicament destine a l'apport continu de glipizide
US6635680B2 (en) * 1999-09-02 2003-10-21 Nostrum Pharmaceuticals, Inc. Controlled release pellet formulation
KR20050112599A (ko) * 2004-05-27 2005-12-01 한국화학연구원 서방형 약물 전달 시스템
KR20050114921A (ko) * 2004-06-02 2005-12-07 씨제이 주식회사 방출제어형 약제학적 조성물
KR100762846B1 (ko) * 2003-09-29 2007-10-04 씨제이 주식회사 서방성 제제
KR20080026754A (ko) * 2006-09-21 2008-03-26 주식회사 삼양사 생물학적 활성성분을 함유하는 방출 제어형 입자, 및 이의제조방법

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5788987A (en) * 1997-01-29 1998-08-04 Poli Industria Chimica Spa Methods for treating early morning pathologies
US6635680B2 (en) * 1999-09-02 2003-10-21 Nostrum Pharmaceuticals, Inc. Controlled release pellet formulation
WO2003057278A2 (fr) * 2002-01-04 2003-07-17 Ivax Research, Inc. Systeme d'apport de medicament destine a l'apport continu de glipizide
KR100762846B1 (ko) * 2003-09-29 2007-10-04 씨제이 주식회사 서방성 제제
KR20050112599A (ko) * 2004-05-27 2005-12-01 한국화학연구원 서방형 약물 전달 시스템
KR20050114921A (ko) * 2004-06-02 2005-12-07 씨제이 주식회사 방출제어형 약제학적 조성물
KR20080026754A (ko) * 2006-09-21 2008-03-26 주식회사 삼양사 생물학적 활성성분을 함유하는 방출 제어형 입자, 및 이의제조방법

Also Published As

Publication number Publication date
KR101152977B1 (ko) 2012-06-11
KR20110067302A (ko) 2011-06-22
WO2011074851A2 (fr) 2011-06-23

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