WO2010018474A3 - Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques - Google Patents

Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques Download PDF

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Publication number
WO2010018474A3
WO2010018474A3 PCT/IB2009/053131 IB2009053131W WO2010018474A3 WO 2010018474 A3 WO2010018474 A3 WO 2010018474A3 IB 2009053131 W IB2009053131 W IB 2009053131W WO 2010018474 A3 WO2010018474 A3 WO 2010018474A3
Authority
WO
WIPO (PCT)
Prior art keywords
preparation
biological uses
novel
glucopyranose derivatives
novel glucopyranose
Prior art date
Application number
PCT/IB2009/053131
Other languages
English (en)
Other versions
WO2010018474A2 (fr
Inventor
Robert Vachy
Original Assignee
Robert Vachy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Robert Vachy filed Critical Robert Vachy
Priority to EP09786642A priority Critical patent/EP2321329A2/fr
Priority to CN2009801354392A priority patent/CN102149723A/zh
Priority to CA2734191A priority patent/CA2734191A1/fr
Priority to US12/737,748 priority patent/US20110136748A1/en
Priority to JP2011522570A priority patent/JP2011530579A/ja
Publication of WO2010018474A2 publication Critical patent/WO2010018474A2/fr
Publication of WO2010018474A3 publication Critical patent/WO2010018474A3/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
    • C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
    • C07H13/08—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals directly attached to carbocyclic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

L'invention a pour objet un nouvel ester, le 3,5-di-tertiobutyl-4-hyclroxybenzoate de 3,4,5-trihydroxy-6-méthoxy tétrahydropyran-2-yl méthyl défini par la formule (I) suivante : L'invention concerne également le procédé de préparation du composé de formule (I) et l'utilisation dudit composé (I) pour la préparation d'un médicament destiné au traitement et/ou à la prévention des infections par des virus à enveloppe.
PCT/IB2009/053131 2008-08-12 2009-07-20 Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques WO2010018474A2 (fr)

Priority Applications (5)

Application Number Priority Date Filing Date Title
EP09786642A EP2321329A2 (fr) 2008-08-12 2009-07-20 Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques
CN2009801354392A CN102149723A (zh) 2008-08-12 2009-07-20 新型吡喃葡萄糖衍生物、其制备和其生物学应用
CA2734191A CA2734191A1 (fr) 2008-08-12 2009-07-20 Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques
US12/737,748 US20110136748A1 (en) 2008-08-12 2009-07-20 Novel glucopyranose derivatives, preparation thereof, and biological uses thereof
JP2011522570A JP2011530579A (ja) 2008-08-12 2009-07-20 新規グルコース誘導体、その製剤および生物学的用途

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR08/04572 2008-08-12
FR0804572A FR2934998B1 (fr) 2008-08-12 2008-08-12 Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques

Publications (2)

Publication Number Publication Date
WO2010018474A2 WO2010018474A2 (fr) 2010-02-18
WO2010018474A3 true WO2010018474A3 (fr) 2010-04-29

Family

ID=40524524

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IB2009/053131 WO2010018474A2 (fr) 2008-08-12 2009-07-20 Nouveaux derives de glucopyranose, leur preparation et leurs applications biologiques

Country Status (7)

Country Link
US (1) US20110136748A1 (fr)
EP (1) EP2321329A2 (fr)
JP (1) JP2011530579A (fr)
CN (1) CN102149723A (fr)
CA (1) CA2734191A1 (fr)
FR (1) FR2934998B1 (fr)
WO (1) WO2010018474A2 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9278989B2 (en) 2012-03-08 2016-03-08 Kyushu University Sugar-derived gelator
CN111658631A (zh) * 2020-06-11 2020-09-15 广东盛普生命科技有限公司 没食子酸及其衍生物和结构类似物在制备抗冠状病毒药物方面的应用

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4870157A (en) * 1985-07-09 1989-09-26 Olin Corporation Selected 4-acyl-2,6-dialkylphenol adducts of saccharides and their use as stabilizers of organic materials against oxidative degradation
FR2887249A1 (fr) * 2005-06-21 2006-12-22 Rdw Pharma Soc Par Actions Sim Compose d-glucopyranose 1-[3,5-bis(1,1-dimenthylethyl)-4- hydroxybenzoate] et ses derives, leur preparation et leurs utilisations

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4833155A (en) * 1986-11-25 1989-05-23 Syntex (U.S.A.) Inc. 3-(ω-(3,5,-di-t-butyl-4-hydroxyphenyl)-alkanoyl)pyrroles, and anti-inflammatory uses thereof
US5312837A (en) * 1991-01-29 1994-05-17 Genelabs Technologies, Inc. Method of treating viral infections with aryl macrocyclic compounds

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4870157A (en) * 1985-07-09 1989-09-26 Olin Corporation Selected 4-acyl-2,6-dialkylphenol adducts of saccharides and their use as stabilizers of organic materials against oxidative degradation
FR2887249A1 (fr) * 2005-06-21 2006-12-22 Rdw Pharma Soc Par Actions Sim Compose d-glucopyranose 1-[3,5-bis(1,1-dimenthylethyl)-4- hydroxybenzoate] et ses derives, leur preparation et leurs utilisations

Also Published As

Publication number Publication date
FR2934998B1 (fr) 2010-09-03
FR2934998A1 (fr) 2010-02-19
US20110136748A1 (en) 2011-06-09
WO2010018474A2 (fr) 2010-02-18
CN102149723A (zh) 2011-08-10
EP2321329A2 (fr) 2011-05-18
JP2011530579A (ja) 2011-12-22
CA2734191A1 (fr) 2010-02-18

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