WO2007009726A3 - Procede de production de compositions pharmaceutiques contenant du glimepiride - Google Patents

Procede de production de compositions pharmaceutiques contenant du glimepiride Download PDF

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Publication number
WO2007009726A3
WO2007009726A3 PCT/EP2006/007016 EP2006007016W WO2007009726A3 WO 2007009726 A3 WO2007009726 A3 WO 2007009726A3 EP 2006007016 W EP2006007016 W EP 2006007016W WO 2007009726 A3 WO2007009726 A3 WO 2007009726A3
Authority
WO
WIPO (PCT)
Prior art keywords
pharmaceutical compositions
compositions containing
producing pharmaceutical
containing glimepiride
glimepiride
Prior art date
Application number
PCT/EP2006/007016
Other languages
German (de)
English (en)
Other versions
WO2007009726A2 (fr
Inventor
Prurushottam S Singnurkar
Prashant Kumar Tewari
Claudia Koritke
Georg Stark
Original Assignee
Alfred E Tiefenbacher Gmbh & C
Usv Ltd
Prurushottam S Singnurkar
Prashant Kumar Tewari
Claudia Koritke
Georg Stark
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alfred E Tiefenbacher Gmbh & C, Usv Ltd, Prurushottam S Singnurkar, Prashant Kumar Tewari, Claudia Koritke, Georg Stark filed Critical Alfred E Tiefenbacher Gmbh & C
Priority to EP06762653A priority Critical patent/EP1904033B1/fr
Priority to DE502006004804T priority patent/DE502006004804D1/de
Priority to AT06762653T priority patent/ATE442132T1/de
Publication of WO2007009726A2 publication Critical patent/WO2007009726A2/fr
Publication of WO2007009726A3 publication Critical patent/WO2007009726A3/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/2027Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La présente invention concerne un procédé de production de compositions pharmaceutiques orales solides contenant du glimépiride. Les compositions produites par ledit procédé sont caractérisées par une stabilité élevée.
PCT/EP2006/007016 2005-07-20 2006-07-17 Procede de production de compositions pharmaceutiques contenant du glimepiride WO2007009726A2 (fr)

Priority Applications (3)

Application Number Priority Date Filing Date Title
EP06762653A EP1904033B1 (fr) 2005-07-20 2006-07-17 Procede de production de compositions pharmaceutiques contenant du glimepiride
DE502006004804T DE502006004804D1 (de) 2005-07-20 2006-07-17 Verfahren zur herstellung von glimepirid enthaltenden pharmazeutischen zusammensetzungen
AT06762653T ATE442132T1 (de) 2005-07-20 2006-07-17 Verfahren zur herstellung von glimepirid enthaltenden pharmazeutischen zusammensetzungen

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102005034484A DE102005034484A1 (de) 2005-07-20 2005-07-20 Verfahren zur Herstellung von Glimepirid enthaltenden pharmazeutischen Zusammensetzungen
DE102005034484.4 2005-07-20

Publications (2)

Publication Number Publication Date
WO2007009726A2 WO2007009726A2 (fr) 2007-01-25
WO2007009726A3 true WO2007009726A3 (fr) 2007-08-23

Family

ID=37650158

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2006/007016 WO2007009726A2 (fr) 2005-07-20 2006-07-17 Procede de production de compositions pharmaceutiques contenant du glimepiride

Country Status (5)

Country Link
EP (1) EP1904033B1 (fr)
AT (1) ATE442132T1 (fr)
DE (2) DE102005034484A1 (fr)
ES (1) ES2333362T3 (fr)
WO (1) WO2007009726A2 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2228066A1 (fr) * 2009-03-03 2010-09-15 LEK Pharmaceuticals d.d. Compositions pharmaceutiques d'un ingrédient pharmaceutique à base de sulphonylurée avec d'excellentes propriétés de dissolution

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19860698A1 (de) * 1998-12-30 2000-07-06 Hexal Ag Neue pharmazeutische Zusammensetzung
US20030147952A1 (en) * 2002-02-01 2003-08-07 Depomed, Inc. Manufacture of oral dosage forms delivering both immediate-release and sustained-release drugs
US20040147564A1 (en) * 2003-01-29 2004-07-29 Rao Vinay U. Combinations of glimepiride and the thiazolidinedione for treatment of diabetes

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3465247B2 (ja) * 1992-12-28 2003-11-10 アベンティス ファーマ株式会社 動脈硬化症の予防および治療剤

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19860698A1 (de) * 1998-12-30 2000-07-06 Hexal Ag Neue pharmazeutische Zusammensetzung
US20030147952A1 (en) * 2002-02-01 2003-08-07 Depomed, Inc. Manufacture of oral dosage forms delivering both immediate-release and sustained-release drugs
US20040147564A1 (en) * 2003-01-29 2004-07-29 Rao Vinay U. Combinations of glimepiride and the thiazolidinedione for treatment of diabetes

Also Published As

Publication number Publication date
ES2333362T3 (es) 2010-02-19
ATE442132T1 (de) 2009-09-15
DE502006004804D1 (de) 2009-10-22
EP1904033B1 (fr) 2009-09-09
DE102005034484A1 (de) 2007-02-01
WO2007009726A2 (fr) 2007-01-25
EP1904033A2 (fr) 2008-04-02

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