WO2006041841A1 - Phenyl derivatives and methods of use - Google Patents

Phenyl derivatives and methods of use Download PDF

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Publication number
WO2006041841A1
WO2006041841A1 PCT/US2005/035677 US2005035677W WO2006041841A1 WO 2006041841 A1 WO2006041841 A1 WO 2006041841A1 US 2005035677 W US2005035677 W US 2005035677W WO 2006041841 A1 WO2006041841 A1 WO 2006041841A1
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Prior art keywords
compounds
methods
disorders
immune
phenyl derivatives
Prior art date
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PCT/US2005/035677
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English (en)
French (fr)
Inventor
Roland E. Dolle
Karin Worm
Q. Jean Zhou
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Adolor Corp
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Adolor Corp
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Publication date
Application filed by Adolor Corp filed Critical Adolor Corp
Priority to MX2007003826A priority Critical patent/MX2007003826A/es
Priority to BRPI0516544-0A priority patent/BRPI0516544A/pt
Priority to AU2005294459A priority patent/AU2005294459A1/en
Priority to JP2007535753A priority patent/JP2008515897A/ja
Priority to EP05810259A priority patent/EP1817277A4/en
Priority to CN2005800340695A priority patent/CN101035758B/zh
Priority to CA002583297A priority patent/CA2583297A1/en
Publication of WO2006041841A1 publication Critical patent/WO2006041841A1/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

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    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
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PCT/US2005/035677 2004-10-05 2005-10-04 Phenyl derivatives and methods of use Ceased WO2006041841A1 (en)

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MX2007003826A MX2007003826A (es) 2004-10-05 2005-10-04 Derivados de fenilo y metodos de uso.
BRPI0516544-0A BRPI0516544A (pt) 2004-10-05 2005-10-04 composto, composição farmacêutica, método de aglutinação de receptores de canabinóides em um paciente e métodos para proteção, indução de apoptose e modulação do apetite
AU2005294459A AU2005294459A1 (en) 2004-10-05 2005-10-04 Phenyl derivatives and methods of use
JP2007535753A JP2008515897A (ja) 2004-10-05 2005-10-04 フェニル誘導体及びそれを使用する方法
EP05810259A EP1817277A4 (en) 2004-10-05 2005-10-04 PHENYL DERIVATIVES AND METHOD OF USE
CN2005800340695A CN101035758B (zh) 2004-10-05 2005-10-04 苯基衍生物及其应用方法
CA002583297A CA2583297A1 (en) 2004-10-05 2005-10-04 Phenyl derivatives and methods of use

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US12016829B2 (en) 2019-10-11 2024-06-25 Pike Therapeutics Inc. Pharmaceutical composition and method for treating seizure disorders
US12097293B2 (en) 2019-10-14 2024-09-24 Pike Therapeutics Inc. Transdermal delivery of cannabidiol
US12121617B2 (en) 2019-10-14 2024-10-22 Pike Therapeutics Inc. Transdermal delivery of cannabidiol
US12186280B2 (en) 2019-10-11 2025-01-07 Pike Therapeutics Inc. Pharmaceutical composition and method for treating seizure disorders
US12268699B2 (en) 2019-10-14 2025-04-08 Pike Therapeutics Inc. Transdermal delivery of tetrahydrocannabinol
US12409132B2 (en) 2019-10-03 2025-09-09 Pike Therapeutics Usa, Inc. Transdermal delivery of dronabinol
US12409131B2 (en) 2019-10-03 2025-09-09 Pike Therapeutics Usa, Inc. Transdermal delivery of dronabinol

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WO2008109027A2 (en) * 2007-03-02 2008-09-12 University Of Tennessee Research Foundation, The Tri-aryl/heteroaroaromatic cannabinoids and use thereof
CN101815513B (zh) * 2007-08-07 2012-11-14 斯泰伦博斯大学 含有对乙酰氨基苯酚的眼用制剂
EP2211619A1 (en) * 2007-10-18 2010-08-04 Merck Sharp & Dohme Corp. Substituted 1,2,4-oxadiazoles and analogs thereof as cb2 receptor modulators, useful in the treatment of pain, respiratory and non-respiratory diseases
WO2009140078A1 (en) * 2008-05-16 2009-11-19 The Procter & Gamble Company Treatment of lower urinary tract dysfunction with cb2-receptor-selective agonists
KR20110130489A (ko) * 2009-03-23 2011-12-05 스미또모 가가꾸 가부시끼가이샤 시클로프로판카르복실산에스테르의 제조 방법
US9855225B2 (en) * 2011-08-18 2018-01-02 Temple University Office Of Technology Transfer Cannabinoid receptor treatments
CN103288684B (zh) * 2013-05-03 2014-12-10 西安交通大学 一种具有抗肿瘤活性的联苯脲化合物及其制备方法
US9585867B2 (en) 2015-08-06 2017-03-07 Charles Everett Ankner Cannabinod formulation for the sedation of a human or animal
US12364668B2 (en) 2017-11-15 2025-07-22 The Regents Of The University Of California Treatment of opioid use disorder, opioid withdrawal symptoms, and chronic pain
EP3838967A1 (en) * 2019-12-16 2021-06-23 Spago Nanomedical AB Immobilization of phenolic compounds
JP7687721B2 (ja) * 2020-12-25 2025-06-03 エムティックスバイオ カンパニ－ リミテッド 新規なアミノアルカン酸にビフェニル基を導入した誘導体化合物およびそれを含む抗炎症用組成物
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Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12409132B2 (en) 2019-10-03 2025-09-09 Pike Therapeutics Usa, Inc. Transdermal delivery of dronabinol
US12409131B2 (en) 2019-10-03 2025-09-09 Pike Therapeutics Usa, Inc. Transdermal delivery of dronabinol
US12016829B2 (en) 2019-10-11 2024-06-25 Pike Therapeutics Inc. Pharmaceutical composition and method for treating seizure disorders
US12186280B2 (en) 2019-10-11 2025-01-07 Pike Therapeutics Inc. Pharmaceutical composition and method for treating seizure disorders
US12097293B2 (en) 2019-10-14 2024-09-24 Pike Therapeutics Inc. Transdermal delivery of cannabidiol
US12121617B2 (en) 2019-10-14 2024-10-22 Pike Therapeutics Inc. Transdermal delivery of cannabidiol
US12268699B2 (en) 2019-10-14 2025-04-08 Pike Therapeutics Inc. Transdermal delivery of tetrahydrocannabinol

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CA2583297A1 (en) 2006-04-20
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BRPI0516544A (pt) 2008-09-09
EP1817277A4 (en) 2010-03-10

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