WO2005095404A3 - 6-(2-fluorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel - Google Patents

6-(2-fluorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel Download PDF

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Publication number
WO2005095404A3
WO2005095404A3 PCT/EP2005/003208 EP2005003208W WO2005095404A3 WO 2005095404 A3 WO2005095404 A3 WO 2005095404A3 EP 2005003208 W EP2005003208 W EP 2005003208W WO 2005095404 A3 WO2005095404 A3 WO 2005095404A3
Authority
WO
WIPO (PCT)
Prior art keywords
halogen
alkyl
membered
triazolopyrimidines
fluorophenyl
Prior art date
Application number
PCT/EP2005/003208
Other languages
English (en)
French (fr)
Other versions
WO2005095404A2 (de
Inventor
Carsten Blettner
Markus Gewehr
Wassilios Grammenos
Thomas Grote
Udo Huenger
Bernd Mueller
Matthias Niedenbrueck
Joachim Rheinheimer
Peter Schaefer
Frank Schieweck
Anja Schwoegler
Oliver Wagner
Michael Rack
Barbara Nave
Maria Scherer
Siegfried Strathmann
Ulrich Schoefl
Reinhard Stierl
Original Assignee
Basf Ag
Carsten Blettner
Markus Gewehr
Wassilios Grammenos
Thomas Grote
Udo Huenger
Bernd Mueller
Matthias Niedenbrueck
Joachim Rheinheimer
Peter Schaefer
Frank Schieweck
Anja Schwoegler
Oliver Wagner
Michael Rack
Barbara Nave
Maria Scherer
Siegfried Strathmann
Ulrich Schoefl
Reinhard Stierl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag, Carsten Blettner, Markus Gewehr, Wassilios Grammenos, Thomas Grote, Udo Huenger, Bernd Mueller, Matthias Niedenbrueck, Joachim Rheinheimer, Peter Schaefer, Frank Schieweck, Anja Schwoegler, Oliver Wagner, Michael Rack, Barbara Nave, Maria Scherer, Siegfried Strathmann, Ulrich Schoefl, Reinhard Stierl filed Critical Basf Ag
Priority to US10/594,738 priority Critical patent/US20070208038A1/en
Priority to JP2007505464A priority patent/JP2007530618A/ja
Priority to BRPI0508717-1A priority patent/BRPI0508717A/pt
Priority to EP05716387A priority patent/EP1732927A2/de
Publication of WO2005095404A2 publication Critical patent/WO2005095404A2/de
Publication of WO2005095404A3 publication Critical patent/WO2005095404A3/de
Priority to IL177661A priority patent/IL177661A0/en

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Catching Or Destruction (AREA)

Abstract

Die vorliegende Anmeldung offenbart 6-(2-Fluorphenyl)-triazolopyrimidine der Formel I in der die Substituenten folgende Bedeutung haben: R1C4-C8-Alkyl, C4-C8-Halogenalkyl, substituiertes C3-C8-Cycloalkyl, C3-C8- Halogencycloalkyl, C5-C8-Alkenyl, C2-C8-Halogenalkenyl, C3-C6-Cycloalkenyl, C3-C6-Halogencyclo­alkenyl, C2-C8-Alkinyl, C2-C8-Halogenalkinyl oder Phenyl, Naphthyl, oder ein fünf­oder sechsgliedriger gesättigter, partiell ungesättigter oder aromatischer Hetero­cyclus, enthaltend ein bis vier Heteroatome aus der Gruppe O, N oder S, R2 Wasserstoff, C1-C3-Alkyl oder eine der bei R1 genannten Gruppen, R1 und R2 können auch zusammen mit dem Stickstoffatom, an das sie gebunden sind, ein fünf- oder sechsgliedriges Heterocyclyl oder Heteroaryl bilden, welches über N gebunden ist und ein bis drei weitere Heteroatome aus der Gruppe O, N und S als Ringglied enthalten,wobei ggf. durch Methyigruppen substituiertes Piperidin-1-yl ausgenommen blei­bt; R1 und/oder R2 können gemäß der Beschreibung substituiert sein; L1 Chlor oder Fluor; L2 Wasserstoff,wenn L1 Fluor bedeutet, zusätzlich Fluor, X Alkyl. Desweiteren werden Verfahren zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Schadpilzen sowie die enthaltende Mittel offenbart.
PCT/EP2005/003208 2004-03-30 2005-03-26 6-(2-fluorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel WO2005095404A2 (de)

Priority Applications (5)

Application Number Priority Date Filing Date Title
US10/594,738 US20070208038A1 (en) 2004-03-30 2005-03-26 6-(2-Fluorophenyl)-Triazolopyrimidines, Method for Producing Them, Their use for Controlling Parasitic Fungi and Agents Containing the Same
JP2007505464A JP2007530618A (ja) 2004-03-30 2005-03-26 ６−（２−フルオロフェニル）−トリアゾロピリミジン、その製造方法、寄生性真菌を抑制するためのその使用、および上記化合物を含有する薬剤
BRPI0508717-1A BRPI0508717A (pt) 2004-03-30 2005-03-26 compostos, processo para preparar os mesmos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
EP05716387A EP1732927A2 (de) 2004-03-30 2005-03-26 6-(2-fluorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
IL177661A IL177661A0 (en) 2004-03-30 2006-08-23 6-(2-fluorophenyl)-triazolopyrimidines, method for producing them, their use for controlling parasitic fungi and agents containing the same

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102004016082.1 2004-03-30
DE102004016082 2004-03-30

Publications (2)

Publication Number Publication Date
WO2005095404A2 WO2005095404A2 (de) 2005-10-13
WO2005095404A3 true WO2005095404A3 (de) 2006-04-06

Family

ID=34962287

Family Applications (2)

Application Number Title Priority Date Filing Date
PCT/EP2005/003208 WO2005095404A2 (de) 2004-03-30 2005-03-26 6-(2-fluorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
PCT/EP2005/004187 WO2005095405A2 (de) 2004-03-30 2005-03-29 6-(2,6-dichlorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel

Family Applications After (1)

Application Number Title Priority Date Filing Date
PCT/EP2005/004187 WO2005095405A2 (de) 2004-03-30 2005-03-29 6-(2,6-dichlorphenyl)-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel

Country Status (7)

Country Link
US (2) US20070208038A1 (de)
EP (2) EP1732927A2 (de)
JP (2) JP2007530618A (de)
CN (2) CN1938313A (de)
BR (2) BRPI0508717A (de)
IL (2) IL177512A0 (de)
WO (2) WO2005095404A2 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007113136A1 (de) * 2006-03-30 2007-10-11 Basf Aktiengesellschaft Verwendung von substituierten riazolopyrimidinen zur bekämpfung von phyto pathogenen schadpilzen

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2765875A1 (fr) * 1997-07-14 1999-01-15 American Cyanamid Co 5-alkyl-triazolopyrimidines fongicides
US5994360A (en) * 1997-07-14 1999-11-30 American Cyanamid Company Fungicidal 5-alkyl-triazolopyrimidines
JP2002308879A (ja) * 2001-04-13 2002-10-23 Nippon Soda Co Ltd ５−ハロアルキル−アゾロピリミジン化合物、製造方法及び有害生物防除剤
WO2002083677A1 (en) * 2001-04-11 2002-10-24 Basf Aktiengesellschaft 6-(2-chloro-6-fluoro-phenyl)-triazolopyrimidines
WO2003008415A1 (en) * 2001-07-18 2003-01-30 Basf Aktiengesellschaft 6-(2,6-difluorophenyl)-triazolopyrimidines as fungicides
WO2004087705A1 (de) * 2003-03-31 2004-10-14 Basf Aktiengesellschaft 7-alkenylamino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6117876A (en) * 1997-04-14 2000-09-12 American Cyanamid Company Fungicidal trifluorophenyl-triazolopyrimidines
NZ523807A (en) * 2000-06-30 2004-09-24 Wyeth Corp Substituted-triazolopyrimidines as anticancer agents
AU2002221831A1 (en) * 2000-11-13 2002-05-21 Basf Aktiengesellschaft 7-(r)-amino-triazolopyrimidines, the production thereof and use of the same for combating phytopathogenic fungi
AU2003232227A1 (en) * 2002-05-03 2003-11-17 Basf Aktiengesellschaft Fungicidal triazolopyrimidines, method for the production thereof, use thereof for controlling harmful fungi and agents containing said fungicidal triazolopyrimidines
UA80304C2 (en) * 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
JP2006522046A (ja) * 2003-04-02 2006-09-28 ビーエーエスエフ　アクチェンゲゼルシャフト ７−（アルキニルアミノ）トリアゾロピリミジン、その製造および有害な真菌の防除におけるその使用、ならびにそれらを含有する製剤

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2765875A1 (fr) * 1997-07-14 1999-01-15 American Cyanamid Co 5-alkyl-triazolopyrimidines fongicides
US5994360A (en) * 1997-07-14 1999-11-30 American Cyanamid Company Fungicidal 5-alkyl-triazolopyrimidines
WO2002083677A1 (en) * 2001-04-11 2002-10-24 Basf Aktiengesellschaft 6-(2-chloro-6-fluoro-phenyl)-triazolopyrimidines
JP2002308879A (ja) * 2001-04-13 2002-10-23 Nippon Soda Co Ltd ５−ハロアルキル−アゾロピリミジン化合物、製造方法及び有害生物防除剤
WO2003008415A1 (en) * 2001-07-18 2003-01-30 Basf Aktiengesellschaft 6-(2,6-difluorophenyl)-triazolopyrimidines as fungicides
WO2004087705A1 (de) * 2003-03-31 2004-10-14 Basf Aktiengesellschaft 7-alkenylamino-triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
PATENT ABSTRACTS OF JAPAN vol. 2003, no. 02 5 February 2003 (2003-02-05) *

Also Published As

Publication number Publication date
EP1732927A2 (de) 2006-12-20
CN1938313A (zh) 2007-03-28
IL177661A0 (en) 2006-12-31
US20070208038A1 (en) 2007-09-06
WO2005095405A2 (de) 2005-10-13
US20070142404A1 (en) 2007-06-21
JP2007530618A (ja) 2007-11-01
JP2007530634A (ja) 2007-11-01
BRPI0508717A (pt) 2007-08-07
WO2005095404A2 (de) 2005-10-13
EP1735316A2 (de) 2006-12-27
BRPI0508728A (pt) 2007-08-14
IL177512A0 (en) 2006-12-10
CN1938312A (zh) 2007-03-28
WO2005095405A3 (de) 2005-12-22

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