WO2002008248A1 - Procede de production de derive de peptides - Google Patents

Procede de production de derive de peptides Download PDF

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Publication number
WO2002008248A1
WO2002008248A1 PCT/JP2001/006295 JP0106295W WO0208248A1 WO 2002008248 A1 WO2002008248 A1 WO 2002008248A1 JP 0106295 W JP0106295 W JP 0106295W WO 0208248 A1 WO0208248 A1 WO 0208248A1
Authority
WO
WIPO (PCT)
Prior art keywords
peptide derivative
hydrogen atom
producing
producing peptide
methyl group
Prior art date
Application number
PCT/JP2001/006295
Other languages
English (en)
Japanese (ja)
Inventor
Tsutomu Sato
Hirohito Shimizu
Original Assignee
Chugai Seiyaku Kabushiki Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Seiyaku Kabushiki Kaisha filed Critical Chugai Seiyaku Kabushiki Kaisha
Priority to AU2001272769A priority Critical patent/AU2001272769A1/en
Publication of WO2002008248A1 publication Critical patent/WO2002008248A1/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic

Abstract

La présente invention concerne un procédé de production d'un composé de formule générale (VI), dans laquelle R1 représente un atome d'hydrogène, un groupe alkyle aliphatique, linéaire ou ramifié, comprenant 1 à 4 atomes de carbone, R2 représente un atome d'hydrogène ou un groupe méthyle, R3 représente un atome d'hydrogène ou un groupe méthyle, et R4 représente un atome d'halogène. Le procédé peut être avantageusement utilisé pour la production commerciale d'un nouveau dérivé de peptides.
PCT/JP2001/006295 2000-07-21 2001-07-19 Procede de production de derive de peptides WO2002008248A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2001272769A AU2001272769A1 (en) 2000-07-21 2001-07-19 Method for producing peptide derivative

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000-219977 2000-07-21
JP2000219977A JP2005097119A (ja) 2000-07-21 2000-07-21 ペプチド誘導体の製造方法

Publications (1)

Publication Number Publication Date
WO2002008248A1 true WO2002008248A1 (fr) 2002-01-31

Family

ID=18714662

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2001/006295 WO2002008248A1 (fr) 2000-07-21 2001-07-19 Procede de production de derive de peptides

Country Status (3)

Country Link
JP (1) JP2005097119A (fr)
AU (1) AU2001272769A1 (fr)
WO (1) WO2002008248A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1312612A1 (fr) * 2000-08-24 2003-05-21 Chugai Seiyaku Kabushiki Kaisha Derive de peptide cyclique

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5555917B2 (ja) * 2010-02-22 2014-07-23 公益財団法人名古屋産業科学研究所 脂肪族第一級アミンのモノメチル化方法

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6357562A (ja) * 1986-08-27 1988-03-12 Kao Corp 新規なアシル化エチレンジアミン誘導体とその製造方法および用途
WO1990006914A1 (fr) * 1988-12-22 1990-06-28 The Upjohn Company N-alcoylation d'acides amines proteges par un groupement n-alpha-boc
WO1994008676A1 (fr) * 1992-10-22 1994-04-28 Kabushiki Kaisha Ace Denken Machine a sous du type a ecran d'affichage

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6357562A (ja) * 1986-08-27 1988-03-12 Kao Corp 新規なアシル化エチレンジアミン誘導体とその製造方法および用途
WO1990006914A1 (fr) * 1988-12-22 1990-06-28 The Upjohn Company N-alcoylation d'acides amines proteges par un groupement n-alpha-boc
WO1994008676A1 (fr) * 1992-10-22 1994-04-28 Kabushiki Kaisha Ace Denken Machine a sous du type a ecran d'affichage

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
NIPPON SEIKAGAKUKAI ED.: "Shin eikagaku jikken kouza 1, tanpakushitsu VI; Gousei oyobi hatsugen", 15 June 1992, TOKYO KAGAKU DOUJIN *

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1312612A1 (fr) * 2000-08-24 2003-05-21 Chugai Seiyaku Kabushiki Kaisha Derive de peptide cyclique
EP1312612A4 (fr) * 2000-08-24 2004-09-22 Chugai Pharmaceutical Co Ltd Derive de peptide cyclique
US7018981B2 (en) 2000-08-24 2006-03-28 Chugai Seiyaku Kabushiki Kaisha Cyclic motilin receptor antagonists

Also Published As

Publication number Publication date
JP2005097119A (ja) 2005-04-14
AU2001272769A1 (en) 2002-02-05

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