WO1996015115A1 - Composes de pyrazole herbicides - Google Patents

Composes de pyrazole herbicides Download PDF

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Publication number
WO1996015115A1
WO1996015115A1 PCT/GB1995/002458 GB9502458W WO9615115A1 WO 1996015115 A1 WO1996015115 A1 WO 1996015115A1 GB 9502458 W GB9502458 W GB 9502458W WO 9615115 A1 WO9615115 A1 WO 9615115A1
Authority
WO
WIPO (PCT)
Prior art keywords
compound
reaction
compounds
general formula
alkyl
Prior art date
Application number
PCT/GB1995/002458
Other languages
English (en)
Inventor
Ewan James Turner Chrystal
Susan Patricia Barnett
Kevin Beautement
Original Assignee
Zeneca Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zeneca Limited filed Critical Zeneca Limited
Priority to AU36599/95A priority Critical patent/AU3659995A/en
Publication of WO1996015115A1 publication Critical patent/WO1996015115A1/fr

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/18—One oxygen or sulfur atom
    • C07D231/20—One oxygen atom attached in position 3 or 5
    • C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

L'invention porte sur des composés de la formule générale (I). Dans cette formule, R1 est un hydrogène ou un alkyle, un alcényle, un alcynyle, un benzyle, un cycloalkyle ou un cycloalcényle, n'importe lequel d'entre eux pouvant éventuellement être substitué. R2 est un alkyle, un alcényle ou un alcynyle, n'importe lequel d'entre eux pouvant éventuellement être substitué, ou un halo, un OR5, un SO¿mR?5, un O(alkyle)CO¿2R?5 ou un O(alkyle)COR5, m étant égal à 0, 1 ou 2. R3 est un hydrogène, un halogène, un cyano, un alkyle, un alcényle ou un alcynyle, n'importe lequel d'entre eux pouvant éventuellement être substitué, ou un SO¿2?Z, COR?5, CO¿2R5 ou un OR5. R4 et un hydrogène, un alkyle, un alcényle ou un alcynyle, n'importe lequel d'entre eux pouvant éventuellement être substitué, ou un cyano, un nitro, un halogène, un NR?5R6, un OR5¿, un SO¿pR?5, un CO¿2R?5, un CONR?5R6, un NR5SO¿2R6, un COR5, un C(NOR5)R6, un OSO¿p?R?5, un NR5COR6¿, un O(alkyle)COR5, un O(alkyle)CO¿2R?5 ou un SO¿2?Z. Chaque X est indépendamment un halogène, un cyano, un nitro, un alkyle, un alcényle, ou un alcynyle, n'importe lequel d'entre eux pouvant éventuellement être substitué, un OR?5, un NR5R6, un NR5SO¿2R6, un OSO¿pR?5, un SO¿pR?5, un CO¿2R?5, un COR?5, un NR5COR6, un R5OR6¿, un CONR5R6, un SO¿2?Z ou un hétérocyclyle ou, selon un autre mode de réalisation, deux groupes X ou un seul groupe X et R?4¿ peuvent former ensemble un autre cycle; Z étant un halogène, p étant égal à 0, 1 ou 2 et n à 0, 1, 2 ou 3. Y est un halogène, un cyano ou un alcoxy éventuellement substitué. R5 et R6 sont chacun d'entre eux indépendamment un hydrogène, un alkyle, un alcényle, un alcynyle, n'importe lequel pouvant éventuellement être substitué. Lesdits composés sont actifs en tant qu'herbicides et efficaces lorsqu'ils sont appliqués avant ou après la levée de la plante.
PCT/GB1995/002458 1994-11-10 1995-10-18 Composes de pyrazole herbicides WO1996015115A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU36599/95A AU3659995A (en) 1994-11-10 1995-10-18 Herbicidal pyrazole compounds

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9422667.7 1994-11-10
GB9422667A GB9422667D0 (en) 1994-11-10 1994-11-10 Herbicides

Publications (1)

Publication Number Publication Date
WO1996015115A1 true WO1996015115A1 (fr) 1996-05-23

Family

ID=10764155

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/GB1995/002458 WO1996015115A1 (fr) 1994-11-10 1995-10-18 Composes de pyrazole herbicides

Country Status (5)

Country Link
AU (1) AU3659995A (fr)
GB (1) GB9422667D0 (fr)
IL (1) IL115712A0 (fr)
WO (1) WO1996015115A1 (fr)
ZA (1) ZA959001B (fr)

Cited By (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997000246A1 (fr) * 1995-06-15 1997-01-03 Novartis Ag Nouveaux herbicides
WO1997012884A1 (fr) * 1995-10-04 1997-04-10 Fmc Corporation Derives de la 6-heterocyclyl-indazole, comme herbicides
WO1997015559A1 (fr) * 1995-10-26 1997-05-01 Basf Aktiengesellschaft 4,5-di(trifluoromethyl)pyrazoles substitues et leur utilisation comme herbicides et pour la dessiccation/defoliation de plantes
WO1997018195A1 (fr) * 1995-11-15 1997-05-22 Basf Aktiengesellschaft 1-methyl-3-phenylpyrazoles substitues et leur utilisation comme herbicides et pour la dessiccation/defoliation de plantes
WO1997040018A1 (fr) * 1996-04-18 1997-10-30 Bayer Aktiengesellschaft 3-cyanoarylpyrazoles et leur utilisation comme herbicides
WO1997046535A1 (fr) * 1996-06-03 1997-12-11 Bayer Aktiengesellschaft 3-cyanoaryl-pyrazoles et leur utilisation comme herbicides
WO1998020000A2 (fr) * 1996-11-04 1998-05-14 Basf Aktiengesellschaft 3-benzylpyrazoles substitues et leur utilisation comme herbicides et pour abaisser la teneur en sucre du sang
WO1998027090A2 (fr) * 1996-12-16 1998-06-25 Basf Aktiengesellschaft Pyrazol-3-ylbenzazoles substitues
FR2773155A1 (fr) * 1997-12-29 1999-07-02 Rhone Poulenc Agrochimie Nouveaux composes fongicides
FR2773153A1 (fr) * 1997-12-29 1999-07-02 Rhone Poulenc Agrochimie Nouveaux composes fongicides
WO1999055702A1 (fr) * 1998-04-29 1999-11-04 Basf Aktiengesellschaft (4-brompyrazol-3-yl)benzazoles substitues
US6096689A (en) * 1995-07-06 2000-08-01 Basf Aktiengesellschaft 5-pyrazolylbenzoic acid derivatives as herbicides
US6100218A (en) * 1996-02-16 2000-08-08 Basf Aktiengesellschaft Substituted 2-phenylpyridines
US6103667A (en) * 1995-06-15 2000-08-15 Novartis Corporation Phenylpyrazole herbicides
US6197973B1 (en) 1996-08-01 2001-03-06 Basf Aktiengesellschaft Substituted 3-phenylpyrazoles
WO2001016138A1 (fr) * 1999-08-27 2001-03-08 Abbott Laboratories Composes sulfonylphenylpyrazoles utiles en tant qu'inhibiteurs de cox-2
WO2001087863A1 (fr) * 2000-05-15 2001-11-22 Basf Aktiengesellschaft 3-arylisothiazoles et leur utilisation en tant qu'herbicides
US6613718B2 (en) 2001-10-01 2003-09-02 Ishihara Sangyo Kaisha, Ltd. Aryl ether derivatives and processes for their preparation and herbicidal and desiccant compositions containing them
WO2006125370A1 (fr) 2005-05-26 2006-11-30 Sinochem Corporation Composes ether aromatiques, leur preparation et leur utilisation
USRE39708E1 (en) 1998-08-07 2007-06-26 Chiron Corporation Estrogen receptor modulators
WO2011042389A2 (fr) 2009-10-09 2011-04-14 Bayer Cropscience Ag Phenylpyri(mi)dinylazoles
US20150105252A1 (en) * 2013-10-15 2015-04-16 E I Du Pont De Nemours And Company Substituted pyrazoles as herbicides

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0372460A (ja) * 1988-06-01 1991-03-27 Nippon Nohyaku Co Ltd ３一置換フェニルピラゾール誘導体又はその塩類及び除草剤
WO1992006962A1 (fr) * 1990-10-18 1992-04-30 Monsanto Company Composes herbicides d'haloalkylpyrazoles aryle substitue

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0372460A (ja) * 1988-06-01 1991-03-27 Nippon Nohyaku Co Ltd ３一置換フェニルピラゾール誘導体又はその塩類及び除草剤
WO1992006962A1 (fr) * 1990-10-18 1992-04-30 Monsanto Company Composes herbicides d'haloalkylpyrazoles aryle substitue

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
CHEMICAL ABSTRACTS, vol. 115, no. 5, 5 August 1991, Columbus, Ohio, US; abstract no. 49684h, J. MIURA ET AL.: "Preparation of 3-phenylpyrazole derivatives as herbicides." page 849; column 1; *

Cited By (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6103667A (en) * 1995-06-15 2000-08-15 Novartis Corporation Phenylpyrazole herbicides
WO1997000246A1 (fr) * 1995-06-15 1997-01-03 Novartis Ag Nouveaux herbicides
US6096689A (en) * 1995-07-06 2000-08-01 Basf Aktiengesellschaft 5-pyrazolylbenzoic acid derivatives as herbicides
WO1997012884A1 (fr) * 1995-10-04 1997-04-10 Fmc Corporation Derives de la 6-heterocyclyl-indazole, comme herbicides
WO1997015559A1 (fr) * 1995-10-26 1997-05-01 Basf Aktiengesellschaft 4,5-di(trifluoromethyl)pyrazoles substitues et leur utilisation comme herbicides et pour la dessiccation/defoliation de plantes
US5962694A (en) * 1995-11-15 1999-10-05 Basf Aktiengesellschaft Substituted 1-methyl-3-phenylpyrazoles and the use thereof as herbicides and for the desiccation or defoliation of plants
WO1997018195A1 (fr) * 1995-11-15 1997-05-22 Basf Aktiengesellschaft 1-methyl-3-phenylpyrazoles substitues et leur utilisation comme herbicides et pour la dessiccation/defoliation de plantes
US6100218A (en) * 1996-02-16 2000-08-08 Basf Aktiengesellschaft Substituted 2-phenylpyridines
WO1997040018A1 (fr) * 1996-04-18 1997-10-30 Bayer Aktiengesellschaft 3-cyanoarylpyrazoles et leur utilisation comme herbicides
WO1997046535A1 (fr) * 1996-06-03 1997-12-11 Bayer Aktiengesellschaft 3-cyanoaryl-pyrazoles et leur utilisation comme herbicides
US6197973B1 (en) 1996-08-01 2001-03-06 Basf Aktiengesellschaft Substituted 3-phenylpyrazoles
WO1998020000A3 (fr) * 1996-11-04 1998-10-29 Basf Ag 3-benzylpyrazoles substitues et leur utilisation comme herbicides et pour abaisser la teneur en sucre du sang
WO1998020000A2 (fr) * 1996-11-04 1998-05-14 Basf Aktiengesellschaft 3-benzylpyrazoles substitues et leur utilisation comme herbicides et pour abaisser la teneur en sucre du sang
US6451734B1 (en) 1996-11-04 2002-09-17 Basf Aktiengesellschaft Substituted 3-benzylpyrazoles and their use as herbicides
EA002350B1 (ru) * 1996-12-16 2002-04-25 Басф Акциенгезельшафт Замещенные пиразол-3-илбензазолы
WO1998027090A3 (fr) * 1996-12-16 1998-09-17 Basf Ag Pyrazol-3-ylbenzazoles substitues
WO1998027090A2 (fr) * 1996-12-16 1998-06-25 Basf Aktiengesellschaft Pyrazol-3-ylbenzazoles substitues
US6232470B1 (en) 1996-12-16 2001-05-15 Basf Aktiengesellschaft Substituted pyrazol-3-ylbenzazoles, their use as herbicides or desiccants/defoliants, and their preparation
FR2773153A1 (fr) * 1997-12-29 1999-07-02 Rhone Poulenc Agrochimie Nouveaux composes fongicides
WO1999033813A1 (fr) * 1997-12-29 1999-07-08 Aventis Cropscience S.A.; Derives 3-hydroxy-pyrazole fongicides
FR2773155A1 (fr) * 1997-12-29 1999-07-02 Rhone Poulenc Agrochimie Nouveaux composes fongicides
US6482774B1 (en) 1998-04-29 2002-11-19 Basf Aktiengesellschaft Substituted (4-brompyrazole-3-yl) benzazoles
WO1999055702A1 (fr) * 1998-04-29 1999-11-04 Basf Aktiengesellschaft (4-brompyrazol-3-yl)benzazoles substitues
AU758553B2 (en) * 1998-04-29 2003-03-27 Basf Aktiengesellschaft Substituted (4-brompyrazole-3-yl)benzazoles
USRE39708E1 (en) 1998-08-07 2007-06-26 Chiron Corporation Estrogen receptor modulators
WO2001016138A1 (fr) * 1999-08-27 2001-03-08 Abbott Laboratories Composes sulfonylphenylpyrazoles utiles en tant qu'inhibiteurs de cox-2
WO2001087863A1 (fr) * 2000-05-15 2001-11-22 Basf Aktiengesellschaft 3-arylisothiazoles et leur utilisation en tant qu'herbicides
US6613718B2 (en) 2001-10-01 2003-09-02 Ishihara Sangyo Kaisha, Ltd. Aryl ether derivatives and processes for their preparation and herbicidal and desiccant compositions containing them
US6927193B2 (en) 2001-10-01 2005-08-09 Ishihara Sangyo Kaisha, Ltd. Aryl ether derivatives and processes for their preparation and herbicidal and desiccant compositions containing them
WO2006125370A1 (fr) 2005-05-26 2006-11-30 Sinochem Corporation Composes ether aromatiques, leur preparation et leur utilisation
WO2011042389A2 (fr) 2009-10-09 2011-04-14 Bayer Cropscience Ag Phenylpyri(mi)dinylazoles
EP2784071A1 (fr) 2009-10-09 2014-10-01 Bayer CropScience AG 3-phenyl-4-pyri(mi)dinyl-1h-pyrazoles et leur utilisation comme fongicides
EP2784070A1 (fr) 2009-10-09 2014-10-01 Bayer CropScience AG 3-phenyl-4-pyri(mi)dinyl-1h-pyrazoles et leur utilisation comme fongicides
EP2784073A1 (fr) 2009-10-09 2014-10-01 Bayer CropScience AG 3-phenyl-4-pyri(mi)dinyl-1h-pyrazoles et leur utilisation comme fongicides
EP2784072A1 (fr) 2009-10-09 2014-10-01 Bayer CropScience AG 3-phenyl-4-pyri(mi)dinyl-1h-pyrazoles et leur utilisation comme fongicides
US20150105252A1 (en) * 2013-10-15 2015-04-16 E I Du Pont De Nemours And Company Substituted pyrazoles as herbicides

Also Published As

Publication number Publication date
GB9422667D0 (en) 1995-01-04
ZA959001B (en) 1996-05-28
IL115712A0 (en) 1996-01-19
AU3659995A (en) 1996-06-06

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