UY37032A - Compuestos de heteroarilbenzimidazol - Google Patents

Compuestos de heteroarilbenzimidazol

Info

Publication number
UY37032A
UY37032A UY0001037032A UY37032A UY37032A UY 37032 A UY37032 A UY 37032A UY 0001037032 A UY0001037032 A UY 0001037032A UY 37032 A UY37032 A UY 37032A UY 37032 A UY37032 A UY 37032A
Authority
UY
Uruguay
Prior art keywords
compounds
heteroarilbenzimidazol
preparing
pharmaceutical compositions
heteroarylbenzimidazole
Prior art date
Application number
UY0001037032A
Other languages
English (en)
Inventor
Horst Irlbacher Dr
Wilhelm Bone Dr
Volker Schulze Dr
Tobias Heinrich Dr
Julien Lefranc Dr
Anne Mengel Dra
Florian Prinz Dr
Antje Wengner Dra
Clara Christ Dra
Roman Hillig Dr
Joszef Bálint Dr
Hans Briem Dr
Ulf Bömer Dr
Detlef Stöckigt Dr
Philip Lienau Dr
Knut Eis Dr
Marcus Koppitz Dr
Benjamin Bader Dr
Jens Schröder Dr
Original Assignee
Bayer Pharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma AG filed Critical Bayer Pharma AG
Publication of UY37032A publication Critical patent/UY37032A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/08Bridged systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La presente invención abarca compuestos heteroarilbenzimidazol de fórmula general (I): en donde R1, R2, R3, R4 y R5 son como se definen en la presente, métodos para preparar dichos compuestos, compuestos intermediarios útiles para preparar dichos compuestos, composiciones farmacéuticas y combinaciones que comprenden dichos compuestos y el uso de dichos compuestos para fabricar composiciones farmacéuticas para el tratamiento o la profilaxis de enfermedades, en particular de trastornos hiperproliferativos y/o inflamatorios, como agente único o en combinación con otros ingredientes activos.
UY0001037032A 2015-12-18 2016-12-16 Compuestos de heteroarilbenzimidazol UY37032A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP15201230 2015-12-18
EP16160885 2016-03-17
EP16193418 2016-10-12

Publications (1)

Publication Number Publication Date
UY37032A true UY37032A (es) 2017-07-31

Family

ID=57882041

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001037032A UY37032A (es) 2015-12-18 2016-12-16 Compuestos de heteroarilbenzimidazol

Country Status (2)

Country Link
TW (1) TW201726657A (es)
UY (1) UY37032A (es)

Also Published As

Publication number Publication date
TW201726657A (zh) 2017-08-01

Similar Documents

Publication Publication Date Title
ECSP19030002A (es) 1,2,4-triazolonas 2,4,5-trisustituidas
CO2018010966A2 (es) Nuevos derivados de pirazolopirimidina
NI201900085A (es) 2-heteroaril-3-oxo-2,3-dihidropiridazin-4-carboxamidas
CO2020001244A2 (es) Derivados de quinolina para tratar infecciones con helmintos
DOP2019000117A (es) Nuevos derivados de quinolina
CO2017011851A2 (es) Compuestos novedosos
ECSP17007538A (es) 2-(morfolin-4-il)-1,7-naftiridinas
UY37460A (es) 1,2,4-triazolonas con anelación en 4 y 5
ECSP20008441A (es) Dihidrooxadiazinonas
DOP2016000253A (es) Nuevos compuestos
UY37971A (es) Derivados de indol macrocíclicos sustituidos
PH12017501133A1 (en) Pyrazolopyridinamines
UY37705A (es) Nuevos derivados de pirazol bicíclicos
UY37972A (es) Derivados de indol macrocíclicos sustituidos con cloro
UY37973A (es) Derivados de indol macrocíclicos
UY35848A (es) Tienopirimidinas
DOP2016000268A (es) Compuestos de azol amido–sustituidos como inhibidores de tnks1 y/o tnks2
DOP2020000100A (es) Novedosos derivados de pirazolo-pirrolo-pirimidina como inhibidores de p2x3
UY37444A (es) Derivados sustituidos de 6-(1h-pirazol-1-il)pirimidin-4-amina y su uso
UY36983A (es) Pirazolopiridinaminas sustituidas
UY37032A (es) Compuestos de heteroarilbenzimidazol
UY34630A (es) Imidazopiridazinas sustituidas con amino

Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20221212