UY35526A - Derivados de espiroindolina y composiciones farma céuticas de los mismos - Google Patents
Derivados de espiroindolina y composiciones farma céuticas de los mismosInfo
- Publication number
- UY35526A UY35526A UY0001035526A UY35526A UY35526A UY 35526 A UY35526 A UY 35526A UY 0001035526 A UY0001035526 A UY 0001035526A UY 35526 A UY35526 A UY 35526A UY 35526 A UY35526 A UY 35526A
- Authority
- UY
- Uruguay
- Prior art keywords
- spiroindoline
- derivatives
- compositions
- céuticas
- sisos
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/10—Spiro-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
- A61P5/04—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
Abstract
Derivados de espiroindolina, procesos para su preparación y composiciones farmacéuticas con los mismos, su uso para el tratamiento de enfermedades y su uso en la elaboración de medicamentos para el tratamiento de enfermedades, en especial enfermeda des relacionadas con las hormonas sexuales, tanto en hombres como en mujeres. La presente solicitud se relaciona en particular con derivados de espiroindolina como antagonistas del receptor de la hormona liberadora de gonadotropina (GnRH).
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP13162986 | 2013-04-09 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY35526A true UY35526A (es) | 2014-11-28 |
Family
ID=48047908
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY0001035526A UY35526A (es) | 2013-04-09 | 2014-04-09 | Derivados de espiroindolina y composiciones farma céuticas de los mismos |
Country Status (28)
Country | Link |
---|---|
US (1) | US20160052936A1 (es) |
EP (1) | EP2984092A1 (es) |
JP (1) | JP2016519104A (es) |
KR (1) | KR20150139917A (es) |
CN (1) | CN105308053A (es) |
AP (1) | AP2015008822A0 (es) |
AR (1) | AR095785A1 (es) |
AU (1) | AU2014253232A1 (es) |
BR (1) | BR112015025700A2 (es) |
CA (1) | CA2908869A1 (es) |
CL (1) | CL2015003013A1 (es) |
CR (1) | CR20150530A (es) |
CU (1) | CU20150141A7 (es) |
DO (1) | DOP2015000259A (es) |
EA (1) | EA201501000A1 (es) |
HK (1) | HK1216101A1 (es) |
IL (1) | IL241067A0 (es) |
MA (1) | MA38463B1 (es) |
MX (1) | MX2015014267A (es) |
NI (1) | NI201500149A (es) |
PE (1) | PE20160007A1 (es) |
PH (1) | PH12015502318A1 (es) |
SG (1) | SG11201506962TA (es) |
TN (1) | TN2015000453A1 (es) |
TW (1) | TW201518304A (es) |
UY (1) | UY35526A (es) |
WO (1) | WO2014166958A1 (es) |
ZA (1) | ZA201508209B (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU2018280742B2 (en) | 2017-06-05 | 2023-12-21 | Kissei Pharmaceutical Co., Ltd. | Gonadotropin-releasing hormone antagonist dosing regimens for the treatment of endometriosis |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0213715D0 (en) * | 2002-06-14 | 2002-07-24 | Syngenta Ltd | Chemical compounds |
SG11201403749VA (en) * | 2012-01-16 | 2014-07-30 | Bayer Ip Gmbh | Spiroindoline derivatives as gonadotropin- releasing hormone receptor antagonists |
-
2014
- 2014-04-07 AR ARP140101498A patent/AR095785A1/es unknown
- 2014-04-08 AP AP2015008822A patent/AP2015008822A0/xx unknown
- 2014-04-08 CA CA2908869A patent/CA2908869A1/en not_active Abandoned
- 2014-04-08 PE PE2015002137A patent/PE20160007A1/es not_active Application Discontinuation
- 2014-04-08 MA MA38463A patent/MA38463B1/fr unknown
- 2014-04-08 EA EA201501000A patent/EA201501000A1/ru unknown
- 2014-04-08 WO PCT/EP2014/057079 patent/WO2014166958A1/en active Application Filing
- 2014-04-08 BR BR112015025700A patent/BR112015025700A2/pt not_active IP Right Cessation
- 2014-04-08 EP EP14715930.5A patent/EP2984092A1/en not_active Withdrawn
- 2014-04-08 AU AU2014253232A patent/AU2014253232A1/en not_active Abandoned
- 2014-04-08 KR KR1020157031635A patent/KR20150139917A/ko not_active Application Discontinuation
- 2014-04-08 JP JP2016506935A patent/JP2016519104A/ja active Pending
- 2014-04-08 TN TN2015000453A patent/TN2015000453A1/en unknown
- 2014-04-08 SG SG11201506962TA patent/SG11201506962TA/en unknown
- 2014-04-08 MX MX2015014267A patent/MX2015014267A/es unknown
- 2014-04-08 CN CN201480032796.7A patent/CN105308053A/zh active Pending
- 2014-04-08 US US14/783,458 patent/US20160052936A1/en not_active Abandoned
- 2014-04-09 TW TW103113078A patent/TW201518304A/zh unknown
- 2014-04-09 UY UY0001035526A patent/UY35526A/es not_active Application Discontinuation
-
2015
- 2015-09-02 IL IL241067A patent/IL241067A0/en unknown
- 2015-10-06 PH PH12015502318A patent/PH12015502318A1/en unknown
- 2015-10-08 CU CUP2015000141A patent/CU20150141A7/es unknown
- 2015-10-09 NI NI201500149A patent/NI201500149A/es unknown
- 2015-10-09 CL CL2015003013A patent/CL2015003013A1/es unknown
- 2015-10-09 DO DO2015000259A patent/DOP2015000259A/es unknown
- 2015-10-09 CR CR20150530A patent/CR20150530A/es unknown
- 2015-11-06 ZA ZA2015/08209A patent/ZA201508209B/en unknown
-
2016
- 2016-04-11 HK HK16104067.2A patent/HK1216101A1/zh unknown
Also Published As
Publication number | Publication date |
---|---|
BR112015025700A2 (pt) | 2017-07-18 |
DOP2015000259A (es) | 2015-11-15 |
EA201501000A1 (ru) | 2016-04-29 |
MX2015014267A (es) | 2016-03-01 |
HK1216101A1 (zh) | 2016-10-14 |
KR20150139917A (ko) | 2015-12-14 |
ZA201508209B (en) | 2018-05-30 |
TN2015000453A1 (en) | 2017-04-06 |
NI201500149A (es) | 2015-11-30 |
PH12015502318A1 (en) | 2016-02-15 |
TW201518304A (zh) | 2015-05-16 |
CR20150530A (es) | 2016-01-29 |
WO2014166958A1 (en) | 2014-10-16 |
US20160052936A1 (en) | 2016-02-25 |
MA38463A1 (fr) | 2018-05-31 |
CL2015003013A1 (es) | 2016-04-08 |
CU20150141A7 (es) | 2016-03-31 |
CN105308053A (zh) | 2016-02-03 |
IL241067A0 (en) | 2015-11-30 |
PE20160007A1 (es) | 2016-02-14 |
JP2016519104A (ja) | 2016-06-30 |
AP2015008822A0 (en) | 2015-10-31 |
EP2984092A1 (en) | 2016-02-17 |
AR095785A1 (es) | 2015-11-11 |
CA2908869A1 (en) | 2014-10-16 |
MA38463B1 (fr) | 2018-11-30 |
SG11201506962TA (en) | 2015-10-29 |
AU2014253232A1 (en) | 2015-11-05 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ECSP19010079A (es) | 3-metil pirazinas 2,5-disustituidas y 3-metil pirazinas 2,5,6-trisustituidas como inhibidores alostéricos de shp2 | |
CL2015003395A1 (es) | Derivados pirazolopirrolidina y su uso en el tratamiento de la enfermedad | |
CL2016000153A1 (es) | Derivados de pirrolamida sustituidos con glioxamida y su uso como medicamentos para el tratamiento de la hepatitis b | |
DOP2016000150A (es) | Nuevas indazolcarboxamidas, procedimientos para su preparación, preparaciones farmacéuticas que las contienen, así como su uso para la preparación de medicamentos | |
CL2015002335A1 (es) | Derivados de 2-aminopirimidina para el tratamiento de infecciones víricas. | |
NI201600144A (es) | Derivados de quinoxalina utiles como moduladores del fgfr cinasa | |
DOP2015000246A (es) | Derivados de oxopiridina sustituida y usos de los mismos en el tratamiento de trastornos cardiovasculares | |
CL2016000807A1 (es) | Amino heteroarilo benzamidas como inhibidores de quinasa. | |
CL2014003444A1 (es) | Compuestos derivados tienopirimidina; proceso de preparacion; composicion farmaceutica que los comprende; combinacion farmaceutica; uso en el tratamiento de canceres y enfermedades autoinmunes. | |
GT201500138A (es) | Novedososo derivados de bencimidazol como antagonistas de ep4 | |
EA201691988A1 (ru) | Производные бороновой кислоты и их терапевтическое применение | |
UY35590A (es) | Nuevos compuestos para el tratamiento del cáncer | |
EA201591004A1 (ru) | Производные бороновой кислоты и их терапевтическое применение | |
EA201591003A1 (ru) | Производные бороновой кислоты и их терапевтическое применение | |
GT201400153A (es) | Derivados de espiroindolina como antagonistas del receptor de la hormona liberadora de gonadotropina | |
UY36779A (es) | Nuevos derivados de exendina-4 como agonistas peptídicos duales específicos de los receptores de glp-1 / glucagón | |
DOP2014000255A (es) | Uracilos sustituidos bicíclicamente y uso de los mismos | |
CL2016000063A1 (es) | Nuevos derivados de indolizina, su procedimiento de preparación y las composiciones farmacéuticas que los contienen. | |
BR112015030387A8 (pt) | compostos de pirazol moduladores de fshr, seu processo de fabricação, composição farmacêutica que os compreende, bem como uso dos mesmos | |
CL2016002091A1 (es) | Compuesto de triazina y su uso para fines medicinales | |
ECSP16012582A (es) | Compuestos heterocíclicos y métodos de uso | |
CL2015002202A1 (es) | Benzamidas sustituidas con actividad hacia receptores ep4. | |
UY35906A (es) | Novedosos derivados de bencimidazol como ligandos de ep4 | |
SV2018005760A (es) | Derivados de aminotiazol utiles como agentes antiviricos | |
UY37947A (es) | Amidas de imidazopiridina sustituidas y su uso |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20211206 |