UY32624A - Procedimiento y composición para mejorar la absorción de agentes terapéuticos - Google Patents

Procedimiento y composición para mejorar la absorción de agentes terapéuticos

Info

Publication number
UY32624A
UY32624A UY0001032624A UY32624A UY32624A UY 32624 A UY32624 A UY 32624A UY 0001032624 A UY0001032624 A UY 0001032624A UY 32624 A UY32624 A UY 32624A UY 32624 A UY32624 A UY 32624A
Authority
UY
Uruguay
Prior art keywords
absorption
procedure
composition
improve
therapeutic agents
Prior art date
Application number
UY0001032624A
Other languages
English (en)
Inventor
Eric R First
Ashish B Patel
Schmitz Guido
Stephanie Petaway-Hickson
Tong Julin
Original Assignee
Bayer Healthcare Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43062708&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY32624(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Llc filed Critical Bayer Healthcare Llc
Publication of UY32624A publication Critical patent/UY32624A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/143Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Inorganic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un comprimido con un perfil de disolución mejorado para un ingrediente medicinalmente activo tal como aspirina y procedimientos para fabricar el comprimido. El comprimido comprende una mezcla de cristales de un ingrediente medicinalmente activo y un coadyuvante de disolución tal como carbonato de sodio o calcio que recubre los cristales al molerlos conjuntamente. La mezcla se prensa después para moldear comprimidos que tienen un perfil de disolución mejorado para el ingrediente medicinalmente activo.
UY0001032624A 2009-05-11 2010-05-11 Procedimiento y composición para mejorar la absorción de agentes terapéuticos UY32624A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12/387,977 US11135188B2 (en) 2009-05-11 2009-05-11 Method and composition to improve absorption of therapeutic agents

Publications (1)

Publication Number Publication Date
UY32624A true UY32624A (es) 2010-12-31

Family

ID=43062708

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032624A UY32624A (es) 2009-05-11 2010-05-11 Procedimiento y composición para mejorar la absorción de agentes terapéuticos

Country Status (15)

Country Link
US (1) US11135188B2 (es)
EP (1) EP2429502B1 (es)
AR (1) AR076864A1 (es)
BR (1) BRPI1013509A2 (es)
CA (1) CA2761678A1 (es)
CL (1) CL2011002807A1 (es)
CO (1) CO6460753A2 (es)
EA (1) EA201171399A1 (es)
HU (1) HUE043173T2 (es)
MX (1) MX2011011928A (es)
PL (1) PL2429502T3 (es)
PT (1) PT2429502T (es)
SI (1) SI2429502T1 (es)
UY (1) UY32624A (es)
WO (1) WO2010132095A1 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US11135188B2 (en) 2009-05-11 2021-10-05 Bayer Healthcare Llc Method and composition to improve absorption of therapeutic agents
US20150366823A1 (en) * 2013-02-06 2015-12-24 Hermes Arzneimittel Gmbh Pharmaceutical compositions incorporating low-dose drugs
WO2015023675A2 (en) 2013-08-12 2015-02-19 Pharmaceutical Manufacturing Research Services, Inc. Extruded immediate release abuse deterrent pill
US10172797B2 (en) 2013-12-17 2019-01-08 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
US9492444B2 (en) 2013-12-17 2016-11-15 Pharmaceutical Manufacturing Research Services, Inc. Extruded extended release abuse deterrent pill
ES2942619T3 (es) 2014-06-11 2023-06-05 SpecGx LLC Composiciones secadas por aspersión con diferentes perfiles de disolución y procedimientos para su preparación
CA2955229C (en) 2014-07-17 2020-03-10 Pharmaceutical Manufacturing Research Services, Inc. Immediate release abuse deterrent liquid fill dosage form
JP2017531026A (ja) 2014-10-20 2017-10-19 ファーマシューティカル マニュファクチュアリング リサーチ サービシズ,インコーポレーテッド 徐放性乱用抑止性液体充填剤形
US11197830B2 (en) * 2019-02-27 2021-12-14 Aft Pharmaceuticals Limited Pharmaceutical composition containing acetaminophen and ibuprofen
WO2022103620A1 (en) * 2020-11-13 2022-05-19 Bayer Healthcare Llc Oral bilayer tablets comprising acetylsalicylic acid and pseudoephedrine, methods of preparing and using thereof

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB191225486A (en) 1912-11-06 1913-04-24 Herbert Sefton-Jones Manufacture and Production of Improved Pharmaceutical Preparations.
US2293359A (en) 1941-01-08 1942-08-18 Quisling Sverre Acetyl salicylic acid preparation
FI89004C (fi) 1988-02-16 1993-08-10 Pertti J Neuvonen Anvaendning av tillsatsmedel foer oekning av absorptionshastigheten av laekemedel i orala laekemedelspreparat
RU2099058C1 (ru) 1992-06-15 1997-12-20 Институт химии твердого тела и переработки минерального сырья СО РАН Способ получения твердой быстрорастворимой дисперсной системы, содержащей ацетилсалициловую кислоту
US5665388A (en) 1995-11-13 1997-09-09 Health Corporation Method for preparation of an alkaline and aspirin combination compound
BR9812018A (pt) 1997-08-27 2000-09-26 Hexal Ag Composições farmacêuticas de meloxicam com solubilidade e biodisponibilidade melhoradas
US8231899B2 (en) * 1998-09-10 2012-07-31 Nycomed Danmark Aps Quick release pharmaceutical compositions of drug substances
US20030180352A1 (en) * 1999-11-23 2003-09-25 Patel Mahesh V. Solid carriers for improved delivery of active ingredients in pharmaceutical compositions
RU2170582C1 (ru) 2000-02-17 2001-07-20 Институт химии твердого тела и механохимии СО РАН Способ получения быстрорастворимой таблетированной формы ацетилсалициловой кислоты
US20080255104A1 (en) 2004-05-04 2008-10-16 Equitech Corporation Nsaid Compositions
US8216610B2 (en) 2004-05-28 2012-07-10 Imaginot Pty Ltd. Oral paracetamol formulations
PL1916994T3 (pl) * 2004-06-29 2014-05-30 Takeda Pharma As Wytwarzanie kompozycji farmaceutycznej o szybkim uwalnianiu leków nierozpuszczalnych w wodzie i kompozycje farmaceutyczne otrzymywane sposobem według wynalazku
NZ709754A (en) * 2004-10-21 2017-02-24 Adare Pharmaceuticals Inc Taste-masked pharmaceutical compositions with gastrosoluble pore-formers
JP2009517346A (ja) 2005-11-28 2009-04-30 イメイジノット ピーティーワイ エルティーディー 治療用化合物の経口送達系
US11135188B2 (en) 2009-05-11 2021-10-05 Bayer Healthcare Llc Method and composition to improve absorption of therapeutic agents

Also Published As

Publication number Publication date
EP2429502A1 (en) 2012-03-21
EA201171399A1 (ru) 2012-05-30
AR076864A1 (es) 2011-07-13
PL2429502T3 (pl) 2019-07-31
BRPI1013509A2 (pt) 2016-04-05
EP2429502B1 (en) 2018-12-26
HUE043173T2 (hu) 2019-08-28
EP2429502A4 (en) 2012-10-24
PT2429502T (pt) 2019-03-29
US20100286100A1 (en) 2010-11-11
CA2761678A1 (en) 2010-11-18
CO6460753A2 (es) 2012-06-15
CL2011002807A1 (es) 2012-06-15
SI2429502T1 (sl) 2019-05-31
WO2010132095A1 (en) 2010-11-18
MX2011011928A (es) 2011-12-06
WO2010132095A8 (en) 2011-07-07
US11135188B2 (en) 2021-10-05

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20181129