|
US4182879A
(en)
*
|
1975-09-24 |
1980-01-08 |
Hoffmann-La Roche Inc. |
N-[3-methyl-4-(2-methyl-4-oxo-3,4-dihydro-quinazolin-3-yl)phenyl]succinamic acid
|
|
US4159330A
(en)
*
|
1976-11-02 |
1979-06-26 |
Carlo Erba S.P.A. |
2-Disubstituted phenyl-3,4-dihydro-4-oxo-quinazoline derivatives and process for their preparation
|
|
FI70036C
(fi)
*
|
1980-01-31 |
1986-09-12 |
Ciba Geigy Ag |
Kromogena kinazolinfoereningar
|
|
US4625027A
(en)
*
|
1982-10-25 |
1986-11-25 |
Ciba-Geigy Corporation |
Bisquinazolines useful in color former systems
|
|
US4668966A
(en)
*
|
1984-04-18 |
1987-05-26 |
Ciba-Geigy Corporation |
Aliphatic bridged chromogenic bisquinazolines substituted with phenylamine or phenyl-containing heterobicyclic radicals
|
|
US4639454A
(en)
*
|
1985-01-17 |
1987-01-27 |
E. I. Du Pont De Nemours And Company |
Phenylquinazolinecarboxylic acids and derivatives as cancer chemotherapeutic agents
|
|
IL89029A
(en)
*
|
1988-01-29 |
1993-01-31 |
Lilly Co Eli |
Fungicidal quinoline and cinnoline derivatives, compositions containing them, and fungicidal methods of using them
|
|
US7473691B2
(en)
*
|
2000-09-15 |
2009-01-06 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
|
ZA200301703B
(en)
*
|
2000-09-15 |
2004-03-02 |
Vertex Pharma |
Pyrazole compounds useful as protein kinase inhibitors.
|
|
CA2422380C
(en)
*
|
2000-09-15 |
2009-03-24 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
|
SI1318997T1
(sl)
*
|
2000-09-15 |
2006-12-31 |
Vertex Pharma |
Pirazolne spojine, uporabne kot inhibitorji protein-kinaze
|
|
US6660731B2
(en)
*
|
2000-09-15 |
2003-12-09 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compounds useful as protein kinase inhibitors
|
|
RU2340611C2
(ru)
*
|
2000-09-15 |
2008-12-10 |
Вертекс Фармасьютикалз Инкорпорейтед |
Производные пиразола, используемые в качестве ингибиторов протеинкиназы
|
|
HUP0400908A3
(en)
*
|
2000-12-21 |
2010-03-29 |
Vertex Pharma |
Pyrazole compounds useful as protein kinase inhibitors, their use and pharmaceutical compositions containing them
|
|
CA2475633C
(en)
*
|
2002-02-06 |
2013-04-02 |
Vertex Pharmaceuticals Incorporated |
Heteroaryl compounds useful as inhibitors of gsk-3
|
|
WO2003078427A1
(en)
*
|
2002-03-15 |
2003-09-25 |
Vertex Pharmaceuticals, Inc. |
Azolylaminoazines as inhibitors of protein kinases
|
|
MY141867A
(en)
|
2002-06-20 |
2010-07-16 |
Vertex Pharma |
Substituted pyrimidines useful as protein kinase inhibitors
|
|
PL374967A1
(en)
|
2002-08-02 |
2005-11-14 |
Vertex Pharmaceuticals Incorporated |
Pyrazole compositions useful as inhibitors of gsk-3
|
|
WO2004072029A2
(en)
*
|
2003-02-06 |
2004-08-26 |
Vertex Pharmaceuticals Incorporated |
Pyrazolopyridazines useful as inhibitors of protein kinases
|
|
CA2548172A1
(en)
*
|
2003-12-04 |
2005-06-23 |
Vertex Pharmaceuticals Incorporated |
Quinoxalines useful as inhibitors of protein kinases
|
|
JP2009504771A
(ja)
*
|
2005-08-18 |
2009-02-05 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
ピラジンキナーゼ阻害剤
|
|
BRPI0619708A2
(pt)
*
|
2005-11-03 |
2011-10-11 |
Vertex Pharma |
composto, composição, método para inibir a atividade da proteìna aurora quinase numa amostra biológica, método para tratar distúrbio proliferativo e método para tratar cáncer
|
|
CA2668429A1
(en)
*
|
2006-11-02 |
2008-05-15 |
Vertex Pharmaceuticals Incorporated |
Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
|
|
WO2008077086A1
(en)
*
|
2006-12-19 |
2008-06-26 |
Vertex Pharmaceuticals Incorporated |
Aminopyrimidines useful as inhibitors of protein kinases
|
|
WO2008112646A1
(en)
|
2007-03-09 |
2008-09-18 |
Vertex Pharmaceuticals Incorporated |
Aminopyridines useful as inhibitors of protein kinases
|
|
JP5520057B2
(ja)
*
|
2007-03-09 |
2014-06-11 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
蛋白キナーゼの阻害剤として有用なアミノピリミジン
|
|
ATE526328T1
(de)
*
|
2007-03-09 |
2011-10-15 |
Vertex Pharma |
Als inhibitoren von proteinkinasen geeignete aminopyrimidine
|
|
AU2008240313A1
(en)
|
2007-04-13 |
2008-10-23 |
Aj Park |
Aminopyrimidines useful as kinase inhibitors
|
|
JP5389785B2
(ja)
|
2007-05-02 |
2014-01-15 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
キナーゼ阻害剤として有用なチアゾールおよびピラゾール
|
|
MX2009011811A
(es)
*
|
2007-05-02 |
2010-01-14 |
Vertex Pharma |
Aminopirimidinas utiles como inhibidores de cinasa.
|
|
CA2694381A1
(en)
*
|
2007-05-02 |
2008-11-13 |
Vertex Pharmaceuticals Incorporated |
Aminopyrimidines useful as kinase inhibitors
|
|
MX2009012719A
(es)
*
|
2007-05-24 |
2010-02-04 |
Vertex Pharma |
Tiazoles y pirazoles utiles como inhibidores de cinasa.
|
|
AR067762A1
(es)
*
|
2007-07-31 |
2009-10-21 |
Vertex Pharma |
Proceso para preparar 5-fluoro-1h-pirazolo (3,4-b) piridin-3-amina y derivados de la misma
|
|
CN102215816A
(zh)
*
|
2008-09-03 |
2011-10-12 |
沃泰克斯药物股份有限公司 |
共晶和包含所述共晶的药物制剂
|