US3883526A - 3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride - Google Patents

3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride Download PDF

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Publication number
US3883526A
US3883526A US367500A US36750073A US3883526A US 3883526 A US3883526 A US 3883526A US 367500 A US367500 A US 367500A US 36750073 A US36750073 A US 36750073A US 3883526 A US3883526 A US 3883526A
Authority
US
United States
Prior art keywords
benzylpyrido
triazine
dihydro
hydrochloride
washed
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
US367500A
Other languages
English (en)
Inventor
George C Wright
Allan V Bayless
Joseph E Gray
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Warner Chilcott Pharmaceuticals Inc
Original Assignee
Morton Norwich Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Morton Norwich Products Inc filed Critical Morton Norwich Products Inc
Priority to US367500A priority Critical patent/US3883526A/en
Priority to ZA00741277A priority patent/ZA741277B/xx
Priority to IL44304A priority patent/IL44304A/en
Priority to GB943574A priority patent/GB1391900A/en
Priority to NL7403598A priority patent/NL7403598A/xx
Priority to SE7405655A priority patent/SE7405655L/xx
Priority to AU68846/74A priority patent/AU473797B2/en
Priority to JP49056787A priority patent/JPS5019772A/ja
Priority to FR7419426A priority patent/FR2232322B1/fr
Priority to BE145155A priority patent/BE816006A/xx
Priority to DE19742427382 priority patent/DE2427382A1/de
Priority to CH774274A priority patent/CH591479A5/xx
Priority to DK302274A priority patent/DK302274A/da
Application granted granted Critical
Publication of US3883526A publication Critical patent/US3883526A/en
Assigned to NORWICH EATON PHARMACEUTICALS, INC., A CORP. OF OH reassignment NORWICH EATON PHARMACEUTICALS, INC., A CORP. OF OH ASSIGNMENT OF ASSIGNORS INTEREST. Assignors: MORTON-NORWICH PRODUCTS, INC., A CORP. OF DE
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/76—Nitrogen atoms to which a second hetero atom is attached
    • C07D213/77—Hydrazine radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Definitions

  • the compounds of this invention are potent antifungal agents. They are capable in small concentration of inhibiting the growth of pathogenic fungi such as Candida albicans and Microsporum Cam's, Such capabilities are represented in the table herebelow which reflects results secured in the commonly used in vitro antifungal test employing Sabourauds dextrose agar as the medium supportive of fungal growth and measuring the amount of inhibition of such growth in millimeters over a period of eight days:

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
US367500A 1973-06-06 1973-06-06 3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride Expired - Lifetime US3883526A (en)

Priority Applications (13)

Application Number Priority Date Filing Date Title
US367500A US3883526A (en) 1973-06-06 1973-06-06 3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride
ZA00741277A ZA741277B (en) 1973-06-06 1974-02-26 3-benzylpyrido (3,4-e)-as-triazine and 1,2-dihydro-3-benzylpyrido (3,4-e)-as -triazine hydrochloride
IL44304A IL44304A (en) 1973-06-06 1974-02-27 History 3 - Benzyl - pyrido] e - 4 [- sa, 3 - triazine and their preparation
GB943574A GB1391900A (en) 1973-06-06 1974-03-01 3-benzylpyrido-3,4-e-astriazine and 1,2-dihydro-3-benzylpyrido- 3,4-e-as-triazine hydrochloride
NL7403598A NL7403598A (enrdf_load_stackoverflow) 1973-06-06 1974-03-18
SE7405655A SE7405655L (enrdf_load_stackoverflow) 1973-06-06 1974-04-26
AU68846/74A AU473797B2 (en) 1973-06-06 1974-05-13 3-benzylpyrido [3,4-e]-as-triazine and 1,2-dihydro-3-benzylpyrido [3,4-e]-as-triazine hydrochloride
JP49056787A JPS5019772A (enrdf_load_stackoverflow) 1973-06-06 1974-05-22
FR7419426A FR2232322B1 (enrdf_load_stackoverflow) 1973-06-06 1974-06-05
BE145155A BE816006A (fr) 1973-06-06 1974-06-06 3-benzylpyrido-/3,4-e/-as-triazine et chlorhydrate de 1,2-dihydro-3-benzylpyrido
DE19742427382 DE2427382A1 (de) 1973-06-06 1974-06-06 3-benzylpyrido- eckige klammer auf 3,4-e eckige klammer zu -as-triazine und verfahren zu deren herstellung
CH774274A CH591479A5 (enrdf_load_stackoverflow) 1973-06-06 1974-06-06
DK302274A DK302274A (enrdf_load_stackoverflow) 1973-06-06 1974-06-06

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US367500A US3883526A (en) 1973-06-06 1973-06-06 3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride

Publications (1)

Publication Number Publication Date
US3883526A true US3883526A (en) 1975-05-13

Family

ID=23447426

Family Applications (1)

Application Number Title Priority Date Filing Date
US367500A Expired - Lifetime US3883526A (en) 1973-06-06 1973-06-06 3-Benzylpyrido {8 3,4-e{9 -as-triazine and 1,2-dihydro-3-benzylpyrido{8 3,4-e{9 -as-triazine hydrochloride

Country Status (13)

Country Link
US (1) US3883526A (enrdf_load_stackoverflow)
JP (1) JPS5019772A (enrdf_load_stackoverflow)
AU (1) AU473797B2 (enrdf_load_stackoverflow)
BE (1) BE816006A (enrdf_load_stackoverflow)
CH (1) CH591479A5 (enrdf_load_stackoverflow)
DE (1) DE2427382A1 (enrdf_load_stackoverflow)
DK (1) DK302274A (enrdf_load_stackoverflow)
FR (1) FR2232322B1 (enrdf_load_stackoverflow)
GB (1) GB1391900A (enrdf_load_stackoverflow)
IL (1) IL44304A (enrdf_load_stackoverflow)
NL (1) NL7403598A (enrdf_load_stackoverflow)
SE (1) SE7405655L (enrdf_load_stackoverflow)
ZA (1) ZA741277B (enrdf_load_stackoverflow)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5225797A (en) * 1975-08-01 1977-02-25 Egyt Gyogyszervegyeszeti Gyar Production of novel derivative pyridd*3*44e** asstriazine
EP0027693A1 (en) * 1979-10-18 1981-04-29 Interox Chemicals Limited Magnesium salts of peroxycarboxylic acids, processes for their preparation and their use as bleaching agents in washing compositions, and processes

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6336085A (ja) * 1986-07-30 1988-02-16 Taiko Kikai Kogyo Kk スクリユウ型真空ポンプ

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3597427A (en) * 1969-01-13 1971-08-03 American Cyanamid Co 1,2-dihydropyrido(3,4-e)-as-triazines

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3597427A (en) * 1969-01-13 1971-08-03 American Cyanamid Co 1,2-dihydropyrido(3,4-e)-as-triazines

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5225797A (en) * 1975-08-01 1977-02-25 Egyt Gyogyszervegyeszeti Gyar Production of novel derivative pyridd*3*44e** asstriazine
EP0027693A1 (en) * 1979-10-18 1981-04-29 Interox Chemicals Limited Magnesium salts of peroxycarboxylic acids, processes for their preparation and their use as bleaching agents in washing compositions, and processes

Also Published As

Publication number Publication date
AU473797B2 (en) 1976-07-01
FR2232322B1 (enrdf_load_stackoverflow) 1977-09-09
FR2232322A1 (enrdf_load_stackoverflow) 1975-01-03
AU6884674A (en) 1975-11-13
BE816006A (fr) 1974-12-06
DE2427382A1 (de) 1975-01-02
IL44304A0 (en) 1974-05-16
SE7405655L (enrdf_load_stackoverflow) 1974-12-09
CH591479A5 (enrdf_load_stackoverflow) 1977-09-15
GB1391900A (en) 1975-04-23
IL44304A (en) 1977-05-31
NL7403598A (enrdf_load_stackoverflow) 1974-12-10
ZA741277B (en) 1975-10-29
JPS5019772A (enrdf_load_stackoverflow) 1975-03-01
DK302274A (enrdf_load_stackoverflow) 1975-02-03

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Date Code Title Description
AS Assignment

Owner name: NORWICH EATON PHARMACEUTICALS, INC., 17 EATON AVE.

Free format text: ASSIGNMENT OF ASSIGNORS INTEREST.;ASSIGNOR:MORTON-NORWICH PRODUCTS, INC., A CORP. OF DE;REEL/FRAME:004085/0126

Effective date: 19820609