UA95780C2 - Xanthine derivatives as selective hm74a agonists - Google Patents

Xanthine derivatives as selective hm74a agonists

Info

Publication number
UA95780C2
UA95780C2 UAA200801702A UAA200801702A UA95780C2 UA 95780 C2 UA95780 C2 UA 95780C2 UA A200801702 A UAA200801702 A UA A200801702A UA A200801702 A UAA200801702 A UA A200801702A UA 95780 C2 UA95780 C2 UA 95780C2
Authority
UA
Ukraine
Prior art keywords
xanthine derivatives
compounds
hm74a agonists
selective
derivatives
Prior art date
Application number
UAA200801702A
Other languages
English (en)
Russian (ru)
Inventor
Ричард Джонатан Дениэл Хетли
Эндрю МкМертри Мейсон
Иван Лео Пинто
Original Assignee
Глаксосмитклайн Ллс
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глаксосмитклайн Ллс filed Critical Глаксосмитклайн Ллс
Publication of UA95780C2 publication Critical patent/UA95780C2/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Даний винахід стосується сполук формули (І), які є похідними ксантину, способів одержання зазначених похідних, фармацевтичних композицій, що містять ці сполуки, і застосування сполук у терапії, наприклад, у лікуванні захворювань, при яких передактивація рецептора НМ74А могла б мати ефект у відношенні захворювання або при яких активація рецептора буде ефективною.(І)
UAA200801702A 2005-08-10 2006-08-08 Xanthine derivatives as selective hm74a agonists UA95780C2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB0516464A GB0516464D0 (en) 2005-08-10 2005-08-10 Novel compounds

Publications (1)

Publication Number Publication Date
UA95780C2 true UA95780C2 (en) 2011-09-12

Family

ID=34984414

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200801702A UA95780C2 (en) 2005-08-10 2006-08-08 Xanthine derivatives as selective hm74a agonists

Country Status (4)

Country Link
CN (2) CN101282976A (uk)
GB (1) GB0516464D0 (uk)
UA (1) UA95780C2 (uk)
ZA (1) ZA200800778B (uk)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS53777B1 (en) * 2008-12-08 2015-06-30 Glaxosmithkline Llc 8-CHLORO-3-PENTYL-3,7-DIHYDRO-1H-PURIN-2,6-DION 2-AMINO-2- (HYDROXYMETHYL) -1,3-PROPANDIOL ANHYDRID FOR DISEASE TREATMENT
SG187549A1 (en) * 2010-08-16 2013-03-28 Boehringer Ingelheim Int Oxadiazole inhibitors of leukotriene production
CN102276610B (zh) * 2011-05-04 2013-01-09 北京工业大学 N7-鸟嘌呤烷化物的制备方法
CN114874209A (zh) * 2017-03-07 2022-08-09 豪夫迈·罗氏有限公司 噁二唑瞬时受体电位通道抑制剂
JP2022549807A (ja) * 2019-09-25 2022-11-29 ゴールドフィンチ バイオ，インク． キサンチンｃｂ１阻害物質

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1404675B1 (en) * 2001-07-03 2008-03-12 Novo Nordisk A/S Dpp-iv-inhibiting purine derivatives for the treatment of diabetes
GB0319124D0 (en) * 2003-08-14 2003-09-17 Smithkline Beecham Corp Chemical compounds

Also Published As

Publication number Publication date
CN101282976A (zh) 2008-10-08
GB0516464D0 (en) 2005-09-14
CN101282977B (zh) 2011-07-27
ZA200800778B (en) 2008-11-26
CN101282977A (zh) 2008-10-08

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