UA74767C2 - Method and composition for oral use of taxanes in patients - Google Patents
Method and composition for oral use of taxanes in patients Download PDFInfo
- Publication number
- UA74767C2 UA74767C2 UA99116450A UA99116450A UA74767C2 UA 74767 C2 UA74767 C2 UA 74767C2 UA 99116450 A UA99116450 A UA 99116450A UA 99116450 A UA99116450 A UA 99116450A UA 74767 C2 UA74767 C2 UA 74767C2
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- UA
- Ukraine
- Prior art keywords
- paclitaxel
- taxane
- administration
- agents
- cyclosporin
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Urology & Nephrology (AREA)
- Gastroenterology & Hepatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US86351397A | 1997-05-27 | 1997-05-27 | |
| PCT/US1998/007776 WO1998053811A1 (en) | 1997-05-27 | 1998-04-22 | Method and compositions for administering taxanes orally to human patients |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UA74767C2 true UA74767C2 (en) | 2006-02-15 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UA99116450A UA74767C2 (en) | 1997-05-27 | 1998-04-22 | Method and composition for oral use of taxanes in patients |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP0994706B1 (xx) |
| JP (1) | JP2002500667A (xx) |
| KR (1) | KR100615783B1 (xx) |
| CN (2) | CN1261275A (xx) |
| AR (1) | AR012731A1 (xx) |
| AT (1) | ATE308365T1 (xx) |
| AU (1) | AU7130098A (xx) |
| BR (1) | BR9809694A (xx) |
| CA (1) | CA2290446C (xx) |
| CZ (1) | CZ9904244A3 (xx) |
| DE (1) | DE69832173T2 (xx) |
| DK (1) | DK0994706T3 (xx) |
| ES (1) | ES2247690T3 (xx) |
| HK (1) | HK1026637A1 (xx) |
| HU (1) | HUP0003546A3 (xx) |
| IL (2) | IL132992A0 (xx) |
| NO (1) | NO995812L (xx) |
| PL (1) | PL337064A1 (xx) |
| RU (1) | RU2205005C2 (xx) |
| SK (1) | SK157599A3 (xx) |
| UA (1) | UA74767C2 (xx) |
| WO (1) | WO1998053811A1 (xx) |
| ZA (1) | ZA984268B (xx) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6964946B1 (en) * | 1995-10-26 | 2005-11-15 | Baker Norton Pharmaceuticals, Inc. | Oral pharmaceutical compositions containing taxanes and methods of treatment employing the same |
| AU3574097A (en) * | 1997-06-20 | 1999-01-04 | Baker Norton Pharmaceuticals, Inc. | Soluble prodrugs of paclitaxel |
| GB9718903D0 (en) | 1997-09-05 | 1997-11-12 | Glaxo Group Ltd | Method,compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| EP1749540B1 (en) | 1999-05-17 | 2010-10-13 | Cancer Research Ventures Limited | Compositions for improving bioavailability of orally administered drugs |
| HUP0203303A3 (en) * | 1999-10-27 | 2005-01-28 | Baker Norton Pharma | Compositions for administering taxanes orally to human patients |
| KR20020013174A (ko) * | 2000-08-11 | 2002-02-20 | 민경윤 | 경구 흡수율이 낮은 약물의 흡수율을 증가시키기 위한경구용 조성물 |
| EP1365759A2 (en) * | 2001-01-18 | 2003-12-03 | PHARMACIA & UPJOHN COMPANY | Chemotherapeutic microemulsion compositions of paclitaxel with improved oral bioavailability |
| US7115565B2 (en) | 2001-01-18 | 2006-10-03 | Pharmacia & Upjohn Company | Chemotherapeutic microemulsion compositions of paclitaxel with improved oral bioavailability |
| EP1623706A3 (en) * | 2001-02-28 | 2006-02-22 | Bristol-Myers Squibb Company | Metronomic dosing of taxanes for inhibiting tumor growth |
| UY27185A1 (es) * | 2001-02-28 | 2002-09-30 | Bristol Myers Squibb Co | Dosificación metronómica de taxanos |
| US7063977B2 (en) | 2001-08-21 | 2006-06-20 | Bristol-Myers Squibb Company | Enzymatic resolution of t-butyl taxane derivatives |
| GB0523659D0 (en) * | 2005-11-21 | 2005-12-28 | Novartis Ag | Organic compounds |
| NZ596868A (en) * | 2009-06-02 | 2014-04-30 | Nikan Pharmaceuticals Llc | Antagonism of human formyl peptide receptor for treatment of disease |
| EP4059497A1 (en) * | 2021-03-17 | 2022-09-21 | Dompé farmaceutici S.p.a. | C5ar1 inhibitors for treating hypersensitivity reactions to taxanes |
| EP4308114A1 (en) * | 2021-03-17 | 2024-01-24 | Dompe' Farmaceutici SpA | C5ar1 inhibitors for treating hypersensitivity reactions to taxanes |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5411947A (en) * | 1989-06-28 | 1995-05-02 | Vestar, Inc. | Method of converting a drug to an orally available form by covalently bonding a lipid to the drug |
| CA2098198A1 (en) * | 1990-12-18 | 1992-06-18 | Ann Christie King | Agents for potentiating the effects of antitumour agents and combating multiple drug resistance |
| CZ283038B6 (cs) * | 1991-01-11 | 1997-12-17 | Laboratoires Glaxo Sa | Akridinové deriváty, způsob výroby a farmaceutické prostředky s jejich obsahem |
| US5567592A (en) * | 1994-02-02 | 1996-10-22 | Regents Of The University Of California | Screening method for the identification of bioenhancers through the inhibition of P-glycoprotein transport in the gut of a mammal |
| ES2126919T3 (es) * | 1994-07-26 | 1999-04-01 | Indena Spa | Taxanos semisinteticos con actividad antitumoral. |
| TW354293B (en) * | 1995-06-06 | 1999-03-11 | Bristol Myers Squibb Co | Prodrugs of paclitaxel derivatives |
| JPH11507356A (ja) * | 1995-06-07 | 1999-06-29 | アブマックス，インコーポレイティド | 経口薬理化合物の生物有用性を高めるためのエッセンシャルオイルの利用 |
| US6245805B1 (en) * | 1995-10-26 | 2001-06-12 | Baker Norton Pharmaceuticals, Inc. | Method, compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| CA2221444A1 (en) * | 1996-01-31 | 1997-08-07 | Steven B. Hansel | A method of making pharmaceutically active taxanes orally bioavailable |
| US6025359A (en) * | 1996-06-17 | 2000-02-15 | Eli Lilly And Company | Drug resistance and multidrug resistance modulators |
| GB9718903D0 (en) * | 1997-09-05 | 1997-11-12 | Glaxo Group Ltd | Method,compositions and kits for increasing the oral bioavailability of pharmaceutical agents |
| AU756752B2 (en) * | 1998-04-01 | 2003-01-23 | Skyepharma Canada Inc. | Anticancer compositions |
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1998
- 1998-04-22 JP JP50066399A patent/JP2002500667A/ja active Pending
- 1998-04-22 IL IL13299298A patent/IL132992A0/xx active IP Right Grant
- 1998-04-22 AU AU71300/98A patent/AU7130098A/en not_active Abandoned
- 1998-04-22 ES ES98918361T patent/ES2247690T3/es not_active Expired - Lifetime
- 1998-04-22 PL PL98337064A patent/PL337064A1/xx unknown
- 1998-04-22 WO PCT/US1998/007776 patent/WO1998053811A1/en active IP Right Grant
- 1998-04-22 EP EP98918361A patent/EP0994706B1/en not_active Expired - Lifetime
- 1998-04-22 SK SK1575-99A patent/SK157599A3/sk unknown
- 1998-04-22 RU RU99128033/14A patent/RU2205005C2/ru not_active IP Right Cessation
- 1998-04-22 UA UA99116450A patent/UA74767C2/uk unknown
- 1998-04-22 KR KR1019997011000A patent/KR100615783B1/ko not_active IP Right Cessation
- 1998-04-22 DE DE69832173T patent/DE69832173T2/de not_active Expired - Fee Related
- 1998-04-22 BR BR9809694-0A patent/BR9809694A/pt not_active IP Right Cessation
- 1998-04-22 HU HU0003546A patent/HUP0003546A3/hu unknown
- 1998-04-22 AT AT98918361T patent/ATE308365T1/de not_active IP Right Cessation
- 1998-04-22 CZ CZ19994244A patent/CZ9904244A3/cs unknown
- 1998-04-22 CN CN98806440A patent/CN1261275A/zh active Pending
- 1998-04-22 CA CA002290446A patent/CA2290446C/en not_active Expired - Fee Related
- 1998-04-22 DK DK98918361T patent/DK0994706T3/da active
- 1998-04-22 CN CNA2004100304785A patent/CN1550231A/zh active Pending
- 1998-05-20 ZA ZA984268A patent/ZA984268B/xx unknown
- 1998-05-21 AR ARP980102356A patent/AR012731A1/es unknown
-
1999
- 1999-11-17 IL IL132992A patent/IL132992A/en not_active IP Right Cessation
- 1999-11-26 NO NO995812A patent/NO995812L/no not_active Application Discontinuation
-
2000
- 2000-09-20 HK HK00105943A patent/HK1026637A1/xx not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CN1550231A (zh) | 2004-12-01 |
| KR100615783B1 (ko) | 2006-08-25 |
| NO995812D0 (no) | 1999-11-26 |
| IL132992A (en) | 2006-08-20 |
| WO1998053811A1 (en) | 1998-12-03 |
| ATE308365T1 (de) | 2005-11-15 |
| RU2205005C2 (ru) | 2003-05-27 |
| ES2247690T3 (es) | 2006-03-01 |
| BR9809694A (pt) | 2000-10-03 |
| DE69832173T2 (de) | 2006-08-03 |
| ZA984268B (en) | 1999-06-23 |
| EP0994706A4 (en) | 2001-05-16 |
| CZ9904244A3 (cs) | 2001-10-17 |
| JP2002500667A (ja) | 2002-01-08 |
| IL132992A0 (en) | 2001-03-19 |
| EP0994706A1 (en) | 2000-04-26 |
| AR012731A1 (es) | 2000-11-08 |
| KR20010013025A (ko) | 2001-02-26 |
| PL337064A1 (en) | 2000-07-31 |
| HUP0003546A3 (en) | 2002-12-28 |
| AU7130098A (en) | 1998-12-30 |
| CA2290446C (en) | 2008-01-29 |
| NO995812L (no) | 2000-01-25 |
| HUP0003546A2 (hu) | 2002-11-28 |
| SK157599A3 (en) | 2002-10-08 |
| EP0994706B1 (en) | 2005-11-02 |
| CA2290446A1 (en) | 1998-12-03 |
| DK0994706T3 (da) | 2006-03-06 |
| HK1026637A1 (en) | 2000-12-22 |
| CN1261275A (zh) | 2000-07-26 |
| DE69832173D1 (de) | 2005-12-08 |
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