UA50762C2 - Похідні арилгліцинаміду та фармацевтична композиція - Google Patents

Похідні арилгліцинаміду та фармацевтична композиція

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Publication number
UA50762C2
UA50762C2 UA98105275A UA98105275A UA50762C2 UA 50762 C2 UA50762 C2 UA 50762C2 UA 98105275 A UA98105275 A UA 98105275A UA 98105275 A UA98105275 A UA 98105275A UA 50762 C2 UA50762 C2 UA 50762C2
Authority
UA
Ukraine
Prior art keywords
pharmaceutical composition
glycinamide derivatives
aryl glycinamide
aryl
derivatives
Prior art date
Application number
UA98105275A
Other languages
English (en)
Russian (ru)
Inventor
Франц Ессер
Герд Шнорренберг
Курт Шромм
Хорст Доллінгер
Біргіт Юнг
Биргит Юнг
Георг Шпек
Original Assignee
Бьорінгер Інгельхайм Фарма Кг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Бьорінгер Інгельхайм Фарма Кг filed Critical Бьорінгер Інгельхайм Фарма Кг
Publication of UA50762C2 publication Critical patent/UA50762C2/uk

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    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/14—Aza-phenalenes, e.g. 1,8-naphthalimide
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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Pulmonology (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Cardiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Винахід стосується нових похідних арилгліцинаміду загальної формули (I) та їх фармацевтично прийнятних солей, в яких R1 і R2 разом з атомом азоту, до якого вони приєднані, утворюють цикли однієї із формул (а), (b), (с) або (d), а R3, R4, R5, Аr, R6, R7, R8, R9, R10, R11, r, s і t мають значення, наведені в описі. Винахід стосується також фармацевтичної композиції, що містить ці сполуки. Сполуки є цінними нейрокінін(тахікінін)-антагоністами.
UA98105275A 1996-03-06 1997-03-03 Похідні арилгліцинаміду та фармацевтична композиція UA50762C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19608665A DE19608665A1 (de) 1996-03-06 1996-03-06 Neue Arylglycinamidderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
PCT/EP1997/001038 WO1997032865A1 (de) 1996-03-06 1997-03-03 Neue arylglycinamidderivate, verfahren zu ihrer herstellung und diese verbindungen enthaltende pharmazeutische zusammensetzungen

Publications (1)

Publication Number Publication Date
UA50762C2 true UA50762C2 (uk) 2002-11-15

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UA98105275A UA50762C2 (uk) 1996-03-06 1997-03-03 Похідні арилгліцинаміду та фармацевтична композиція

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US (2) US6498162B1 (uk)
EP (1) EP0885204B1 (uk)
JP (1) JP3465795B2 (uk)
KR (1) KR19990087636A (uk)
CN (1) CN1072664C (uk)
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AT (1) ATE219069T1 (uk)
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DE (2) DE19608665A1 (uk)
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HR (1) HRP970130A2 (uk)
HU (1) HUP9901823A3 (uk)
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NZ (1) NZ332201A (uk)
PL (1) PL328779A1 (uk)
PT (1) PT885204E (uk)
SK (1) SK283052B6 (uk)
TR (1) TR199801734T2 (uk)
TW (1) TW375614B (uk)
UA (1) UA50762C2 (uk)
WO (1) WO1997032865A1 (uk)
YU (1) YU8197A (uk)
ZA (1) ZA971850B (uk)

Families Citing this family (26)

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DE19824470A1 (de) * 1998-05-30 1999-12-02 Boehringer Ingelheim Pharma Neue Neurokininantagonisten, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
GB9923748D0 (en) 1999-10-07 1999-12-08 Glaxo Group Ltd Chemical compounds
USRE39921E1 (en) 1999-10-07 2007-11-13 Smithkline Beecham Corporation Chemical compounds
US6664253B2 (en) 2000-10-17 2003-12-16 Boehringer Ingelheim Pharma Kg Neurokinin antagonists
GB0025354D0 (en) 2000-10-17 2000-11-29 Glaxo Group Ltd Chemical compounds
DE10051320A1 (de) * 2000-10-17 2002-04-25 Boehringer Ingelheim Pharma Neue Neurokininantagonisten, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen
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AU718584B2 (en) 2000-04-13
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