TWI345465B - Proteasome inhibitors and methods of using the same - Google Patents
Proteasome inhibitors and methods of using the same Download PDFInfo
- Publication number
- TWI345465B TWI345465B TW93124291A TW93124291A TWI345465B TW I345465 B TWI345465 B TW I345465B TW 93124291 A TW93124291 A TW 93124291A TW 93124291 A TW93124291 A TW 93124291A TW I345465 B TWI345465 B TW I345465B
- Authority
- TW
- Taiwan
- Prior art keywords
- amino
- methylbutyl
- hexahydro
- carbonyl
- imino
- Prior art date
Links
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49576403P | 2003-08-14 | 2003-08-14 |
Publications (2)
Publication Number | Publication Date |
---|---|
TW200529810A TW200529810A (en) | 2005-09-16 |
TWI345465B true TWI345465B (en) | 2011-07-21 |
Family
ID=37426112
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW93124291A TWI345465B (en) | 2003-08-14 | 2004-08-13 | Proteasome inhibitors and methods of using the same |
Country Status (7)
Country | Link |
---|---|
CN (1) | CN1867572B (es) |
AR (2) | AR045381A1 (es) |
MY (1) | MY162518A (es) |
PE (1) | PE20050360A1 (es) |
TW (1) | TWI345465B (es) |
UA (1) | UA88771C2 (es) |
ZA (1) | ZA200601293B (es) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI598352B (zh) * | 2008-09-29 | 2017-09-11 | 千禧製藥公司 | 1-胺基-2-環丁基乙酸衍生物 |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2178888B1 (en) * | 2007-08-06 | 2012-07-04 | Millennium Pharmaceuticals, Inc. | Proteasome inhibitors |
CN105837608B (zh) * | 2007-08-06 | 2018-06-08 | 米伦纽姆医药公司 | 蛋白酶体抑制剂及其组合物和用途 |
CN102961387B (zh) * | 2007-08-06 | 2016-04-27 | 米伦纽姆医药公司 | 蛋白酶体抑制剂 |
EA201500431A1 (ru) * | 2008-06-17 | 2015-11-30 | Милленниум Фармасьютикалз, Инк. | Соединения боронатного эфира и его фармацевтические составы |
CN101638414B (zh) * | 2008-07-30 | 2014-01-08 | 江苏先声药物研究有限公司 | 肽硼酸及其酯类化合物、制备方法及其用途 |
CN101747354B (zh) * | 2008-12-04 | 2014-08-13 | 江苏先声药物研究有限公司 | 一类β氨基酸组成的二肽硼酸及其酯类化合物、制备方法及其用途 |
CA2785300A1 (en) * | 2009-12-22 | 2011-07-21 | Cephalon, Inc. | Proteasome inhibitors and processes for their preparation, purification and use |
RU2012146101A (ru) * | 2010-03-31 | 2014-05-10 | Милленниум Фармасьютикалз, Инк. | Производные 1-амино-2-циклопропилэтилбороновой кислоты |
SG11201702628XA (en) * | 2014-10-01 | 2017-04-27 | Merck Patent Gmbh | Boronic acid derivatives |
CN106588965A (zh) * | 2015-10-15 | 2017-04-26 | 北京大学 | 脲拟肽硼酸化合物及其药物组合物、制备方法和用途 |
WO2017198194A1 (zh) * | 2016-05-19 | 2017-11-23 | 成都奥璟生物科技有限公司 | 一种硼酸和硼酸酯类化合物及其应用 |
JP7071400B6 (ja) * | 2017-01-18 | 2022-06-07 | プリンシピア バイオファーマ インコーポレイテッド | 免疫プロテアソーム阻害剤 |
TW201831191A (zh) * | 2017-01-23 | 2018-09-01 | 大陸商成都奥璟生物科技有限公司 | 一種新的硼酸衍生物及其藥物組合物 |
CN114437119A (zh) * | 2020-10-30 | 2022-05-06 | 苏州开拓药业股份有限公司 | 一种c-Myc蛋白抑制剂及其制备方法和用途 |
-
2004
- 2004-08-13 MY MYPI20043299A patent/MY162518A/en unknown
- 2004-08-13 UA UAA200602694A patent/UA88771C2/ru unknown
- 2004-08-13 TW TW93124291A patent/TWI345465B/zh active
- 2004-08-13 PE PE2004000784A patent/PE20050360A1/es active IP Right Grant
- 2004-08-13 CN CN2004800301520A patent/CN1867572B/zh active Active
- 2004-08-17 AR ARP040102935 patent/AR045381A1/es not_active Application Discontinuation
-
2006
- 2006-02-13 ZA ZA200601293A patent/ZA200601293B/xx unknown
-
2014
- 2014-03-11 AR ARP140100859A patent/AR095249A2/es not_active Application Discontinuation
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI598352B (zh) * | 2008-09-29 | 2017-09-11 | 千禧製藥公司 | 1-胺基-2-環丁基乙酸衍生物 |
Also Published As
Publication number | Publication date |
---|---|
AR095249A2 (es) | 2015-09-30 |
TW200529810A (en) | 2005-09-16 |
PE20050360A1 (es) | 2005-06-10 |
ZA200601293B (en) | 2009-09-30 |
UA88771C2 (ru) | 2009-11-25 |
CN1867572A (zh) | 2006-11-22 |
MY162518A (en) | 2017-06-15 |
CN1867572B (zh) | 2012-03-28 |
AR045381A1 (es) | 2005-10-26 |
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