TW362974B - Novel heteroaryl-oxazolidinones - Google Patents

Novel heteroaryl-oxazolidinones

Info

Publication number
TW362974B
TW362974B TW086101260A TW86101260A TW362974B TW 362974 B TW362974 B TW 362974B TW 086101260 A TW086101260 A TW 086101260A TW 86101260 A TW86101260 A TW 86101260A TW 362974 B TW362974 B TW 362974B
Authority
TW
Taiwan
Prior art keywords
carbon atoms
substituents
oxazolidinones
side chain
group
Prior art date
Application number
TW086101260A
Other languages
Chinese (zh)
Inventor
Bernd Riedl
Dieter Habich
Andreas Stolle
Martin Tuppelt
Stephan Bartel
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Application granted granted Critical
Publication of TW362974B publication Critical patent/TW362974B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

A kind of novel heteroaryl-oxazolidinones of the general formula and cubic isomer thereof and mixture of cubic isomer thereof and the salt, in which the R1 represents the group of D-R2 or -CO-R3 or -CONR4R5, in which D represents the group of carbon dioxide or sulfide oxide; R2 represents the trifluoride or the alkyl of normal chain or side chain; and R4 and R5 are same or different which is hydrogen and contains at most 3 carbon atoms and A is thienyl group, pyridine or quinoline; these substituents can be selectively chosen by at most two same or different substituents; those said substituents are chosen from chlorine, bromine, pyridazine, normal chain or side chain alkyl or alkoxyl which are composed at most five carbon atoms, pyrimidine and pyridazine which can be substituted by normal chain or side chain alkyl or alkoxyl with at most five carbon atoms.
TW086101260A 1996-02-06 1997-02-04 Novel heteroaryl-oxazolidinones TW362974B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19604224 1996-02-06
DE19649095A DE19649095A1 (en) 1996-02-06 1996-11-27 New 5-(acyl-aminomethyl)-3-hetero-aryl-oxazolidinone compounds

Publications (1)

Publication Number Publication Date
TW362974B true TW362974B (en) 1999-07-01

Family

ID=7784634

Family Applications (1)

Application Number Title Priority Date Filing Date
TW086101260A TW362974B (en) 1996-02-06 1997-02-04 Novel heteroaryl-oxazolidinones

Country Status (10)

Country Link
KR (1) KR970061891A (en)
AR (1) AR005704A1 (en)
CO (1) CO4761067A1 (en)
DE (1) DE19649095A1 (en)
PE (1) PE36098A1 (en)
SV (1) SV1997000010A (en)
TN (1) TNSN97033A1 (en)
TW (1) TW362974B (en)
YU (1) YU4497A (en)
ZA (1) ZA97928B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
DE19802239A1 (en) * 1998-01-22 1999-07-29 Bayer Ag New oxazolidinone derivatives useful as antimicrobial agents against Gram-positive and some Gram-negative bacteria, mycobacteria, etc.
WO1999037630A1 (en) 1998-01-23 1999-07-29 Versicor, Inc. Oxazolidinone combinatorial libraries, compositions and methods of preparation
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
WO2006106426A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc An oxindole oxazolidinone as antibacterial agent
AU2006231919A1 (en) 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents
WO2008021337A1 (en) 2006-08-15 2008-02-21 Wyeth Oxazinan-2-one derivatives useful as pr modulators
TW200815428A (en) 2006-08-15 2008-04-01 Wyeth Corp Oxazolidone derivatives as PR modulators

Also Published As

Publication number Publication date
ZA97928B (en) 1997-08-05
SV1997000010A (en) 1997-10-23
KR970061891A (en) 1997-09-12
AR005704A1 (en) 1999-07-14
PE36098A1 (en) 1998-08-29
CO4761067A1 (en) 1999-04-27
DE19649095A1 (en) 1997-08-07
YU4497A (en) 1999-09-27
TNSN97033A1 (en) 2005-03-15

Similar Documents

Publication Publication Date Title
ATE218859T1 (en) LIGANDS OF NEUROPEPTIDE Y
TW349843B (en) Substituted 1-arylpyrazoles
NZ332605A (en) Tricyclic benzazepine vasopressin antagonists
GB9300763D0 (en) Chemical compound
EP1000999A4 (en) Compounds for organic el devices and organic el devices
EP0640586A4 (en) Stilbene derivative and stilbene analog derivative, and use thereof.
TW362974B (en) Novel heteroaryl-oxazolidinones
WO1999009965A3 (en) Anti-inflammatory agent
MY117092A (en) Chemotherapeutic pyrrolocarbazole derivatives
PL356541A1 (en) 2-(1h-indol-3-yl)-2-oxo-acetamides with antitumor activity
GR81961B (en)
SI1086096T1 (en) Benzamides with tetrahydrofuranyloxy substitutents as phosphodiesterase 4 inhibitors
HUP9904198A2 (en) Novel fungicide composition containing a 2-imidazoline-5-one
ES8705425A1 (en) Isoindolinyl-alkyl-piperazines
ES2108618A1 (en) Triphendioxazine compounds
TW324009B (en) Pyrazole condensation ring derivative, its production process and its use as androgen inhibitor
TW351718B (en) Acylated aminoalkanimidazoles and -triazoles
ES453881A1 (en) 1,3-dithiolo(4,5-b)pyrazin-2-ylidene-propanedinitrile 4-oxide
MX9805858A (en) Pyridine derivatives as fungicides.
NZ333854A (en) Intermediates for the preparation of 2-imidazoline-5-ones
GR3031162T3 (en) Thiazolotriazole and thiazolodiazole derivatives with fungicidal activity.
ES8300757A1 (en) Isoxazolyl indolamines.
AU567867B2 (en) 5(e)-13,14,18,18,19,19-hexahydro-6a-carbaprostaglandin 12 derivatives
EP0940388A4 (en) Oxime derivatives, hydrazone derivatives, and use thereof
IE780540L (en) Pyrano triazines