TNSN97033A1 - NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS. - Google Patents

NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS.

Info

Publication number
TNSN97033A1
TNSN97033A1 TNTNSN97033A TNSN97033A TNSN97033A1 TN SN97033 A1 TNSN97033 A1 TN SN97033A1 TN TNSN97033 A TNTNSN97033 A TN TNSN97033A TN SN97033 A TNSN97033 A TN SN97033A TN SN97033 A1 TNSN97033 A1 TN SN97033A1
Authority
TN
Tunisia
Prior art keywords
oxazolidinones
preparing
medicaments
novel heteroaryl
heteroaryl
Prior art date
Application number
TNTNSN97033A
Other languages
French (fr)
Inventor
Bernd Riedl Dr
Dieter Habich Dr
Andreas Stolle Dr
Martin Ruppelt Dr
Stephan Bartel Dr
Walter Guarnieri Dr
Rainer Endermann Dr
Hein Peter Kroll Dr
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of TNSN97033A1 publication Critical patent/TNSN97033A1/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

L'INVENTION CONCERNE DE NOUVELLES HETEROARYL-OXAZOLIDINONES DE FORMULE GENERALE ( I) DANS LAQUELLE LES SUBSTITUANTS SONT TELS QUE DEFINIS DANS LA DESCRIPTION, DES PROCEDES POUR LES PREPARER, ET LEUR UTILISATION EN TANT QUE MEDICAMENTS, EN PARTICULIER EN TANT QUE MEDICAMENTS ANTIBACTERIENS.THE INVENTION RELATES TO NEW HETEROARYL-OXAZOLIDINONES OF GENERAL FORMULA (I) IN WHICH THE SUBSTITUTES ARE AS DEFINED IN THE DESCRIPTION, METHODS FOR PREPARING THEM, AND THEIR USE AS DRUGS, PARTICULARLY AS ANTIBACTERIALS.

TNTNSN97033A 1996-02-06 1997-02-04 NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS. TNSN97033A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19604224 1996-02-06
DE19649095A DE19649095A1 (en) 1996-02-06 1996-11-27 New 5-(acyl-aminomethyl)-3-hetero-aryl-oxazolidinone compounds

Publications (1)

Publication Number Publication Date
TNSN97033A1 true TNSN97033A1 (en) 2005-03-15

Family

ID=7784634

Family Applications (1)

Application Number Title Priority Date Filing Date
TNTNSN97033A TNSN97033A1 (en) 1996-02-06 1997-02-04 NOVEL HETEROARYL-OXAZOLIDINONES, PROCESS FOR PREPARING THEM, AND THEIR USE AS MEDICAMENTS.

Country Status (10)

Country Link
KR (1) KR970061891A (en)
AR (1) AR005704A1 (en)
CO (1) CO4761067A1 (en)
DE (1) DE19649095A1 (en)
PE (1) PE36098A1 (en)
SV (1) SV1997000010A (en)
TN (1) TNSN97033A1 (en)
TW (1) TW362974B (en)
YU (1) YU4497A (en)
ZA (1) ZA97928B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds
DE19802239A1 (en) * 1998-01-22 1999-07-29 Bayer Ag New oxazolidinone derivatives useful as antimicrobial agents against Gram-positive and some Gram-negative bacteria, mycobacteria, etc.
JP2002501059A (en) 1998-01-23 2002-01-15 ファルマシア・アンド・アップジョン・カンパニー Oxazolidinone combinatorial libraries, compositions and preparation methods
US7002020B1 (en) 1998-01-23 2006-02-21 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
US6562844B2 (en) 1998-01-23 2003-05-13 Pharmacia & Upjohn Company Oxazolidinone combinatorial libraries, compositions and methods of preparation
AU2006231919A1 (en) 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents
WO2006106426A1 (en) * 2005-04-06 2006-10-12 Pharmacia & Upjohn Company Llc An oxindole oxazolidinone as antibacterial agent
WO2008021337A1 (en) 2006-08-15 2008-02-21 Wyeth Oxazinan-2-one derivatives useful as pr modulators
TW200815428A (en) 2006-08-15 2008-04-01 Wyeth Corp Oxazolidone derivatives as PR modulators

Also Published As

Publication number Publication date
KR970061891A (en) 1997-09-12
AR005704A1 (en) 1999-07-14
CO4761067A1 (en) 1999-04-27
ZA97928B (en) 1997-08-05
PE36098A1 (en) 1998-08-29
SV1997000010A (en) 1997-10-23
TW362974B (en) 1999-07-01
YU4497A (en) 1999-09-27
DE19649095A1 (en) 1997-08-07

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