TW202509017A - 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途 - Google Patents

胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途 Download PDF

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TW202509017A
TW202509017A TW113124586A TW113124586A TW202509017A TW 202509017 A TW202509017 A TW 202509017A TW 113124586 A TW113124586 A TW 113124586A TW 113124586 A TW113124586 A TW 113124586A TW 202509017 A TW202509017 A TW 202509017A
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Taiwan
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amino
phenyl
nicotinamide
azabicyclo
hexane
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TW113124586A
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Chinese (zh)
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路卡 亞力斯塔
麥可 派翠客 狄隆
瑞妮 拉特曼
迪米崔歐斯 利卓斯
尼可勞斯 喬漢尼斯 史蒂夫
湯瑪士 優兒瑞其
佩姬 烏索曼
史文 威勒
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瑞士商諾華公司
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
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TW113124586A 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途 TW202509017A (zh)

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TW113124586A TW202509017A (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW106123900A TWI712598B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW111103316A TWI806385B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW112118991A TWI851226B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW110101592A TWI755255B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途

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TW111103316A TWI806385B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW112118991A TWI851226B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途
TW110101592A TWI755255B (zh) 2016-07-20 2017-07-18 胺基吡啶衍生物及其作為選擇性alk-2抑制劑之用途

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