TW202317586A - 治療性化合物及方法 - Google Patents

治療性化合物及方法 Download PDF

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Publication number
TW202317586A
TW202317586A TW111126584A TW111126584A TW202317586A TW 202317586 A TW202317586 A TW 202317586A TW 111126584 A TW111126584 A TW 111126584A TW 111126584 A TW111126584 A TW 111126584A TW 202317586 A TW202317586 A TW 202317586A
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Taiwan
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group
compound
groups
pharmaceutically acceptable
prodrug
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TW111126584A
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Chinese (zh)
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莎曼莎 艾利森 格林
潔西卡 瑪麗 格蘭德
史蒂芬 湯瑪斯 史戴本
內裡 阿瑪拉
維施瓦 Ｍ 狄克斯特
艾莉西亞 維勒木
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美商建南德克公司
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Publication of TW202317586A publication Critical patent/TW202317586A/zh

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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02—Inorganic compounds
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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    • C07F9/02—Phosphorus compounds
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    • C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings

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  • Diabetes (AREA)
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TW111126584A 2021-07-15 2022-07-15 治療性化合物及方法 TW202317586A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US202163222288P 2021-07-15 2021-07-15
US63/222,288 2021-07-15

Publications (1)

Publication Number Publication Date
TW202317586A true TW202317586A (zh) 2023-05-01

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TW111126584A TW202317586A (zh) 2021-07-15 2022-07-15 治療性化合物及方法

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US (2) US12006331B2 (https=)
EP (1) EP4370130A4 (https=)
JP (1) JP2024527604A (https=)
KR (1) KR20240036571A (https=)
CN (1) CN117642170A (https=)
AR (1) AR126470A1 (https=)
AU (1) AU2022309856A1 (https=)
CA (1) CA3226225A1 (https=)
CL (1) CL2024000114A1 (https=)
CO (1) CO2024001017A2 (https=)
CR (1) CR20240016A (https=)
IL (1) IL309878A (https=)
MX (1) MX2024000610A (https=)
PE (1) PE20240776A1 (https=)
TW (1) TW202317586A (https=)
WO (1) WO2023287793A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN117642170A (zh) 2021-07-15 2024-03-01 基因泰克公司 治疗性化合物及方法
WO2025082533A1 (zh) * 2023-10-21 2025-04-24 上海轶诺药业有限公司 一种稠环化合物及其制备和应用

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2003508401A (ja) * 1999-08-27 2003-03-04 アボット・ラボラトリーズ Ｃｏｘ−２阻害薬として有用なスルホニルフェニルピラゾール化合物
JP2003510280A (ja) * 1999-09-27 2003-03-18 アメリカン・サイアナミド・カンパニー バソプレッシンアゴニスト処方および製法
AR039475A1 (es) * 2002-05-01 2005-02-23 Wyeth Corp 6-alquiliden-penems triciclicos como inhibidores de beta-lactamasa
US20070232582A1 (en) 2004-04-28 2007-10-04 Wyeth Holdings Corporation 4-substituted or unsubtituted-7-hydro-1,4-thiazepine-7-[bicyclic or tricyclic heteroaryl] substituted-3,6-dicarboxylic acid derivatives as beta-lactamase inhibitors
CA3103432A1 (en) * 2018-06-27 2020-01-02 Children's Medical Center Corporation Compounds for inhibition of inflammation
EP3833345B1 (en) 2018-08-07 2024-07-17 Kemijski Institut Small molecule-inhibitors of 6-phosphofructo-1-kinase for reducing lactate generation by cancer cells
CN117642170A (zh) 2021-07-15 2024-03-01 基因泰克公司 治疗性化合物及方法

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Publication number Publication date
KR20240036571A (ko) 2024-03-20
CO2024001017A2 (es) 2024-03-07
EP4370130A4 (en) 2025-06-11
WO2023287793A1 (en) 2023-01-19
JP2024527604A (ja) 2024-07-25
US12459957B2 (en) 2025-11-04
AU2022309856A1 (en) 2024-01-18
US12006331B2 (en) 2024-06-11
US20250109142A1 (en) 2025-04-03
US20230119740A1 (en) 2023-04-20
CL2024000114A1 (es) 2024-08-02
CN117642170A (zh) 2024-03-01
MX2024000610A (es) 2024-02-02
AR126470A1 (es) 2023-10-11
PE20240776A1 (es) 2024-04-17
IL309878A (en) 2024-03-01
EP4370130A1 (en) 2024-05-22
CA3226225A1 (en) 2023-01-19
CR20240016A (es) 2024-02-13

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