TW201206891A - Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response - Google Patents
Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response Download PDFInfo
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Classifications
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- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36075510P | 2010-07-01 | 2010-07-01 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201206891A true TW201206891A (en) | 2012-02-16 |
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Family Applications (1)
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| TW100123408A TW201206891A (en) | 2010-07-01 | 2011-07-01 | Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response |
Country Status (18)
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| US (3) | US8492424B2 (OSRAM) |
| EP (1) | EP2588459B1 (OSRAM) |
| JP (1) | JP5922116B2 (OSRAM) |
| KR (1) | KR20130141434A (OSRAM) |
| CN (1) | CN103038219B (OSRAM) |
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| BR (1) | BR112013000065A2 (OSRAM) |
| CA (1) | CA2804194C (OSRAM) |
| CL (1) | CL2013000002A1 (OSRAM) |
| CO (1) | CO6680625A2 (OSRAM) |
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| PH (1) | PH12013500121A1 (OSRAM) |
| RU (1) | RU2013102967A (OSRAM) |
| SG (1) | SG186886A1 (OSRAM) |
| TW (1) | TW201206891A (OSRAM) |
| WO (1) | WO2012003414A1 (OSRAM) |
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| US10206813B2 (en) | 2009-05-18 | 2019-02-19 | Dose Medical Corporation | Implants with controlled drug delivery features and methods of using same |
| US12478503B2 (en) | 2009-05-18 | 2025-11-25 | Glaukos Corporation | Implants with controlled drug delivery features and methods of using same |
| US8859606B2 (en) * | 2010-07-01 | 2014-10-14 | Allergan, Inc. | Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response |
| US9006450B2 (en) | 2010-07-01 | 2015-04-14 | Boehringer Ingelheim International Gmbh | Compounds, pharmaceutical compositions and uses thereof |
| US8969589B2 (en) * | 2011-12-21 | 2015-03-03 | Allergan, Inc. | Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response |
| CA2862263C (en) * | 2011-12-27 | 2016-09-06 | Allergan, Inc. | Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response |
| EP2966064A1 (en) * | 2011-12-27 | 2016-01-13 | Allergan, Inc. | Pyrazole-3-carboxylic acid compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response |
| WO2014028762A1 (en) | 2012-08-15 | 2014-02-20 | University Of Virginia Patent Foundation | Compositions and methods for treating peripheral arterial disease |
| JP6403688B2 (ja) * | 2013-01-21 | 2018-10-10 | アラーガン、インコーポレイテッドＡｌｌｅｒｇａｎ，Ｉｎｃｏｒｐｏｒａｔｅｄ | 全身性抗炎症反応を提供する複数のプロスタグランジン受容体で作用する化合物 |
| EP3063133A1 (en) | 2013-10-31 | 2016-09-07 | Allergan, Inc. | 3-{1-[5-chloro-2-(2-ethylbutoxy)benzyl]-5-methyl-1h-pyrazol-3-yl}propanoic acid in crystalline form and methods for use thereof |
| CN106146400A (zh) * | 2015-03-20 | 2016-11-23 | 四川大学 | 苄基-1h-吡唑、苄基-1h-吡咯衍生物及其制备方法和用途 |
| US10462745B2 (en) | 2016-01-15 | 2019-10-29 | Google Llc | Systems and methods for extending battery life by monitoring device activity |
| CN107723304A (zh) * | 2016-08-10 | 2018-02-23 | 中国科学院上海生命科学研究院 | Prkar2a在炎症消退中的应用 |
| CA3121202A1 (en) | 2018-11-30 | 2020-06-04 | Nuvation Bio Inc. | Pyrrole and pyrazole compounds and methods of use thereof |
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| US4166452A (en) | 1976-05-03 | 1979-09-04 | Generales Constantine D J Jr | Apparatus for testing human responses to stimuli |
| US4256108A (en) | 1977-04-07 | 1981-03-17 | Alza Corporation | Microporous-semipermeable laminated osmotic system |
| US4265874A (en) | 1980-04-25 | 1981-05-05 | Alza Corporation | Method of delivering drug with aid of effervescent activity generated in environment of use |
| US4826868A (en) * | 1986-05-29 | 1989-05-02 | Ortho Pharmaceutical Corporation | 1,5-Diaryl-3-substituted pyrazoles pharmaceutical compositions and use |
| US6511999B2 (en) | 2000-09-14 | 2003-01-28 | Allergan, Inc. | Interheteroaryl 7-oxabicyclic [2.2.1]heptane oxazoles as prostaglandin F2α antagonists |
| US7273883B2 (en) | 2000-09-14 | 2007-09-25 | Allergan, Inc. | Prostaglandin EP4 antagonist |
| US7217725B2 (en) | 2000-09-14 | 2007-05-15 | Allergan, Inc. | Prostaglandin D2 antagonist |
| CA2526013A1 (en) * | 2003-05-20 | 2004-12-02 | Merck Frosst Canada Ltd. | Fluoro-methanesulfonyl-substituted cycloalkanoindoles and their use as prostaglandin d2 antagonists |
| US20070060596A1 (en) | 2003-10-24 | 2007-03-15 | Giblin Gerard M P | Heterocyclyl compounds |
| GB0508472D0 (en) | 2005-04-26 | 2005-06-01 | Glaxo Group Ltd | Compounds |
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| AU2011272716A1 (en) | 2013-02-07 |
| EP2588459B1 (en) | 2017-03-01 |
| BR112013000065A2 (pt) | 2019-09-24 |
| US20140121258A1 (en) | 2014-05-01 |
| US8492424B2 (en) | 2013-07-23 |
| US20130253028A1 (en) | 2013-09-26 |
| ES2625355T3 (es) | 2017-07-19 |
| EP2588459A1 (en) | 2013-05-08 |
| KR20130141434A (ko) | 2013-12-26 |
| AR082073A1 (es) | 2012-11-07 |
| PH12013500121A1 (en) | 2013-03-11 |
| US20120165382A1 (en) | 2012-06-28 |
| AU2011272716B2 (en) | 2016-05-19 |
| MX2013000170A (es) | 2013-05-28 |
| CA2804194A1 (en) | 2012-01-05 |
| JP2013535424A (ja) | 2013-09-12 |
| CN103038219A (zh) | 2013-04-10 |
| SG186886A1 (en) | 2013-02-28 |
| CA2804194C (en) | 2019-03-05 |
| CL2013000002A1 (es) | 2013-05-31 |
| CN103038219B (zh) | 2016-08-24 |
| WO2012003414A1 (en) | 2012-01-05 |
| CO6680625A2 (es) | 2013-05-31 |
| JP5922116B2 (ja) | 2016-05-24 |
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