TW200612964A - Methods for preparing p2x7 inhibitors - Google Patents

Methods for preparing p2x7 inhibitors

Info

Publication number
TW200612964A
TW200612964A TW094121706A TW94121706A TW200612964A TW 200612964 A TW200612964 A TW 200612964A TW 094121706 A TW094121706 A TW 094121706A TW 94121706 A TW94121706 A TW 94121706A TW 200612964 A TW200612964 A TW 200612964A
Authority
TW
Taiwan
Prior art keywords
methods
preparing
inhibitors
present
compounds
Prior art date
Application number
TW094121706A
Other languages
English (en)
Inventor
Zhengong B Li
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34972172&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW200612964(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TW200612964A publication Critical patent/TW200612964A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D253/00—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00
    • C07D253/02—Heterocyclic compounds containing six-membered rings having three nitrogen atoms as the only ring hetero atoms, not provided for by group C07D251/00 not condensed with other rings
    • C07D253/06—1,2,4-Triazines
    • C07D253/065—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members
    • C07D253/07—1,2,4-Triazines having three double bonds between ring members or between ring members and non-ring members with hetero atoms, or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D253/075—Two hetero atoms, in positions 3 and 5
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
TW094121706A 2004-06-29 2005-06-28 Methods for preparing p2x7 inhibitors TW200612964A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US58385104P 2004-06-29 2004-06-29

Publications (1)

Publication Number Publication Date
TW200612964A true TW200612964A (en) 2006-05-01

Family

ID=34972172

Family Applications (1)

Application Number Title Priority Date Filing Date
TW094121706A TW200612964A (en) 2004-06-29 2005-06-28 Methods for preparing p2x7 inhibitors

Country Status (15)

Country Link
US (1) US7235657B2 (zh)
EP (1) EP1776352A1 (zh)
JP (1) JP2008504360A (zh)
CN (1) CN1980902A (zh)
AR (1) AR049653A1 (zh)
AU (1) AU2005258911A1 (zh)
BR (1) BRPI0512781A (zh)
CA (1) CA2571124A1 (zh)
IL (1) IL179461A0 (zh)
MX (1) MXPA06014022A (zh)
NO (1) NO20065327L (zh)
RU (1) RU2006146675A (zh)
TW (1) TW200612964A (zh)
WO (1) WO2006003500A1 (zh)
ZA (1) ZA200609579B (zh)

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ES2396565T3 (es) 2003-05-12 2013-02-22 Pah Usa 15 Llc Inhibidores benzamida del receptor P2X7
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SG157299A1 (en) * 2008-05-09 2009-12-29 Agency Science Tech & Res Diagnosis and treatment of kawasaki disease
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EP2322149A1 (en) 2009-11-03 2011-05-18 Universidad del Pais Vasco Methods and compositions for the treatment of ischemia
BR112012028850A2 (pt) 2010-05-14 2015-09-15 Affectis Pharmaceuticals Ag métodos para a preparação de antagonistas de p2x7r
WO2012110190A1 (en) 2011-02-17 2012-08-23 Affectis Pharmaceuticals Ag Novel p2x7r antagonists and their use
WO2012163456A1 (en) 2011-05-27 2012-12-06 Affectis Pharmaceuticals Ag Novel p2x7r antagonists and their use
WO2012163792A1 (en) 2011-05-27 2012-12-06 Affectis Pharmaceuticals Ag Novel p2x7r antagonists and their use
US9988373B2 (en) 2013-12-26 2018-06-05 Shionogi & Co., Ltd. Nitrogen-containing six-membered cyclic derivatives and pharmaceutical composition comprising the same
WO2016171249A1 (ja) * 2015-04-24 2016-10-27 塩野義製薬株式会社 ６員複素環誘導体およびそれらを含有する医薬組成物
WO2017209265A1 (ja) * 2016-06-03 2017-12-07 塩野義製薬株式会社 二環性複素環誘導体およびそれらを含有する医薬組成物
CA3039458A1 (en) 2016-10-17 2018-04-26 Shionogi & Co., Ltd. Bicyclic nitrogen-containing heterocyclic derivatives and pharmaceutical composition comprising the same
JP6692113B2 (ja) * 2016-10-21 2020-05-13 塩野義製薬株式会社 ６員複素環誘導体を含有する医薬組成物

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Also Published As

Publication number Publication date
NO20065327L (no) 2006-12-18
WO2006003500A8 (en) 2006-04-13
CN1980902A (zh) 2007-06-13
IL179461A0 (en) 2007-05-15
EP1776352A1 (en) 2007-04-25
BRPI0512781A (pt) 2008-04-08
JP2008504360A (ja) 2008-02-14
CA2571124A1 (en) 2006-01-12
ZA200609579B (en) 2008-08-27
WO2006003500A1 (en) 2006-01-12
AU2005258911A1 (en) 2006-01-12
US7235657B2 (en) 2007-06-26
MXPA06014022A (es) 2007-02-08
RU2006146675A (ru) 2008-07-10
US20050288256A1 (en) 2005-12-29
AR049653A1 (es) 2006-08-23

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