TW200504088A - Avermectin B1 monosaccharide derivatives - Google Patents
Avermectin B1 monosaccharide derivativesInfo
- Publication number
- TW200504088A TW200504088A TW093117009A TW93117009A TW200504088A TW 200504088 A TW200504088 A TW 200504088A TW 093117009 A TW093117009 A TW 093117009A TW 93117009 A TW93117009 A TW 93117009A TW 200504088 A TW200504088 A TW 200504088A
- Authority
- TW
- Taiwan
- Prior art keywords
- avermectin
- c12alkenyl
- c12alkyl
- tautomers
- isomers
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0313937.5A GB0313937D0 (en) | 2003-06-16 | 2003-06-16 | Avermectin B1 monosaccharide derivatives having an aminosulfonyloxy substituentin the 4'-position |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200504088A true TW200504088A (en) | 2005-02-01 |
Family
ID=27636648
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW093117009A TW200504088A (en) | 2003-06-16 | 2004-06-14 | Avermectin B1 monosaccharide derivatives |
Country Status (15)
Country | Link |
---|---|
US (1) | US7521429B2 (zh) |
EP (1) | EP1638984B1 (zh) |
JP (1) | JP4750698B2 (zh) |
AR (1) | AR045693A1 (zh) |
AT (1) | ATE370157T1 (zh) |
CY (1) | CY1106940T1 (zh) |
DE (1) | DE602004008281T2 (zh) |
DK (1) | DK1638984T3 (zh) |
ES (1) | ES2293276T3 (zh) |
GB (1) | GB0313937D0 (zh) |
PL (1) | PL1638984T3 (zh) |
PT (1) | PT1638984E (zh) |
SI (1) | SI1638984T1 (zh) |
TW (1) | TW200504088A (zh) |
WO (1) | WO2004111070A1 (zh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200538461A (en) * | 2004-04-07 | 2005-12-01 | Syngenta Participations Ag | Avermectin and avermectin monosaccharide substituted in the 4"-and 4'-position respectively |
AU2011252987B2 (en) | 2010-05-12 | 2013-05-02 | Boehringer Ingelheim Animal Health USA Inc. | Injectable parasiticidal formulations of levamisole and macrocyclic lactones |
NZ612185A (en) | 2010-12-07 | 2015-10-30 | Merial Inc | Topical combination formulations of macrocyclic lactones with synthetic pyrethroids |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4622313A (en) | 1985-08-01 | 1986-11-11 | Merck & Co., Inc. | O-sulfate derivatives of avermectins and milbemycins having improved water solubility |
US4833168A (en) * | 1986-10-03 | 1989-05-23 | Merck & Co., Inc. | Avermectin reformatsky adducts |
US4906619A (en) * | 1988-07-22 | 1990-03-06 | Merck & Co., Inc. | Alkyl avermectin derivatives |
NZ231773A (en) * | 1988-12-23 | 1992-09-25 | Merck & Co Inc | Avermectin derivatives, preparation and parasiticidal pharmaceutical compositions thereof |
US5208222A (en) | 1991-03-28 | 1993-05-04 | Merck & Co., Inc. | 4"-and 4'-alkylthio avermectin derivatives |
GB9205007D0 (en) * | 1992-03-07 | 1992-04-22 | Pfizer Ltd | Antiparasitic agents |
AR037938A1 (es) | 2001-12-21 | 2004-12-22 | Syngenta Participations Ag | Derivados de avermectina b1 que tienen un substituyente de aminosulfoniloxilo en la posicion 4'' |
-
2003
- 2003-06-16 GB GBGB0313937.5A patent/GB0313937D0/en not_active Ceased
-
2004
- 2004-06-14 AR ARP040102059A patent/AR045693A1/es unknown
- 2004-06-14 TW TW093117009A patent/TW200504088A/zh unknown
- 2004-06-15 DE DE602004008281T patent/DE602004008281T2/de not_active Expired - Lifetime
- 2004-06-15 EP EP04739912A patent/EP1638984B1/en not_active Expired - Lifetime
- 2004-06-15 PL PL04739912T patent/PL1638984T3/pl unknown
- 2004-06-15 JP JP2006515942A patent/JP4750698B2/ja not_active Expired - Fee Related
- 2004-06-15 ES ES04739912T patent/ES2293276T3/es not_active Expired - Lifetime
- 2004-06-15 DK DK04739912T patent/DK1638984T3/da active
- 2004-06-15 US US10/560,390 patent/US7521429B2/en not_active Expired - Lifetime
- 2004-06-15 SI SI200430477T patent/SI1638984T1/sl unknown
- 2004-06-15 PT PT04739912T patent/PT1638984E/pt unknown
- 2004-06-15 WO PCT/EP2004/006442 patent/WO2004111070A1/en active IP Right Grant
- 2004-06-15 AT AT04739912T patent/ATE370157T1/de active
-
2007
- 2007-10-19 CY CY20071101344T patent/CY1106940T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
ES2293276T3 (es) | 2008-03-16 |
GB0313937D0 (en) | 2003-07-23 |
US20060229263A1 (en) | 2006-10-12 |
ATE370157T1 (de) | 2007-09-15 |
CY1106940T1 (el) | 2012-09-26 |
DE602004008281D1 (en) | 2007-09-27 |
PT1638984E (pt) | 2007-11-09 |
EP1638984A1 (en) | 2006-03-29 |
DE602004008281T2 (de) | 2008-05-15 |
US7521429B2 (en) | 2009-04-21 |
JP4750698B2 (ja) | 2011-08-17 |
JP2006527724A (ja) | 2006-12-07 |
SI1638984T1 (sl) | 2007-12-31 |
PL1638984T3 (pl) | 2008-02-29 |
WO2004111070A1 (en) | 2004-12-23 |
AR045693A1 (es) | 2005-11-09 |
EP1638984B1 (en) | 2007-08-15 |
DK1638984T3 (da) | 2007-12-03 |
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