TW200502220A - Novel process for the preparation of 2-aminomethylpyridine derivatives - Google Patents
Novel process for the preparation of 2-aminomethylpyridine derivativesInfo
- Publication number
- TW200502220A TW200502220A TW093110136A TW93110136A TW200502220A TW 200502220 A TW200502220 A TW 200502220A TW 093110136 A TW093110136 A TW 093110136A TW 93110136 A TW93110136 A TW 93110136A TW 200502220 A TW200502220 A TW 200502220A
- Authority
- TW
- Taiwan
- Prior art keywords
- derivatives
- formula
- preparation
- novel process
- aminomethylpyridine
- Prior art date
Links
- WOXFMYVTSLAQMO-UHFFFAOYSA-N 2-Pyridinemethanamine Chemical class NCC1=CC=CC=N1 WOXFMYVTSLAQMO-UHFFFAOYSA-N 0.000 title 1
- KBRRIEFTVXTTCR-UHFFFAOYSA-N 2-(nitromethyl)pyridine Chemical class [O-][N+](=O)CC1=CC=CC=N1 KBRRIEFTVXTTCR-UHFFFAOYSA-N 0.000 abstract 2
- -1 2-substituted pyridine Chemical class 0.000 abstract 1
- RGDQRXPEZUNWHX-UHFFFAOYSA-N 3-methylpyridin-2-amine Chemical class CC1=CC=CN=C1N RGDQRXPEZUNWHX-UHFFFAOYSA-N 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 239000003054 catalyst Substances 0.000 abstract 1
- 125000004971 nitroalkyl group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/36—Radicals substituted by singly-bound nitrogen atoms
- C07D213/38—Radicals substituted by singly-bound nitrogen atoms having only hydrogen or hydrocarbon radicals attached to the substituent nitrogen atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
- C07D213/26—Radicals substituted by halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0309631.0A GB0309631D0 (en) | 2003-04-28 | 2003-04-28 | Novel process for the preparation of 2-aminomethylpyridine derivatives |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW200502220A true TW200502220A (en) | 2005-01-16 |
| TWI359139B TWI359139B (en) | 2012-03-01 |
Family
ID=9957269
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW093110136A TWI359139B (en) | 2003-04-28 | 2004-04-12 | Novel process for the preparation of 2-aminomethyl |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US7608720B2 (zh) |
| EP (1) | EP1620404B1 (zh) |
| JP (1) | JP4718446B2 (zh) |
| KR (2) | KR101213005B1 (zh) |
| CN (1) | CN100413847C (zh) |
| AT (1) | ATE356116T1 (zh) |
| BR (1) | BRPI0409517A (zh) |
| DE (1) | DE602004005175T2 (zh) |
| DK (1) | DK1620404T3 (zh) |
| ES (1) | ES2279383T3 (zh) |
| GB (1) | GB0309631D0 (zh) |
| IL (1) | IL170657A (zh) |
| PL (1) | PL1620404T3 (zh) |
| TW (1) | TWI359139B (zh) |
| WO (1) | WO2004096772A1 (zh) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI650318B (zh) * | 2017-10-30 | 2019-02-11 | 財團法人工業技術研究院 | 以結晶法純化２，５－呋喃二甲酸的粗產物之方法與聚酯之形成方法 |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN107266333A (zh) | 2012-07-12 | 2017-10-20 | 日产化学工业株式会社 | 肟取代酰胺化合物和有害生物防除剂 |
| CN106220555B (zh) * | 2016-07-29 | 2019-06-21 | 天津市均凯化工科技有限公司 | 一种制备2-氨甲基-3-氯-5-三氟甲基吡啶的方法 |
| US11236070B2 (en) | 2019-05-16 | 2022-02-01 | Novartis Ag | Chemical process |
| CN115819330A (zh) * | 2022-12-28 | 2023-03-21 | 天津均凯农业科技有限公司 | 一种连续化制备2-氨基甲基-3-氯-5-三氟甲基吡啶的方法 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3615293A1 (de) * | 1986-05-06 | 1987-11-12 | Bayer Ag | Verwendung von heteroarylethylaminen zur leistungsfoerderung bei tieren, heteroarylethylamine und verfahren zu ihrer herstellung |
| ZA885069B (en) * | 1987-07-24 | 1989-03-29 | Fujisawa Pharmaceutical Co | Sustained-release percutaneous preparations |
| FR2649978B1 (fr) * | 1989-07-20 | 1991-10-25 | Rhone Poulenc Chimie | Procede d'hydrogenation de derives halogeno nitroaromatiques en presence d'iodures |
| AU2002213948B2 (en) * | 2000-08-25 | 2006-08-17 | Bayer Cropscience S.A. | Process for the preparation of 2-aminoethylpyridines |
| DE10101647A1 (de) | 2001-01-16 | 2002-07-18 | Degussa | Verfahren zur Herstellung von substituierten Aminen durch Hydrierung von substituierten organischen Nitroverbindungen |
-
2003
- 2003-04-28 GB GBGB0309631.0A patent/GB0309631D0/en not_active Ceased
-
2004
- 2004-04-12 TW TW093110136A patent/TWI359139B/zh not_active IP Right Cessation
- 2004-04-26 AT AT04739624T patent/ATE356116T1/de not_active IP Right Cessation
- 2004-04-26 JP JP2006505421A patent/JP4718446B2/ja not_active Expired - Lifetime
- 2004-04-26 ES ES04739624T patent/ES2279383T3/es not_active Expired - Lifetime
- 2004-04-26 WO PCT/EP2004/006075 patent/WO2004096772A1/en active IP Right Grant
- 2004-04-26 EP EP04739624A patent/EP1620404B1/en not_active Expired - Lifetime
- 2004-04-26 DE DE602004005175T patent/DE602004005175T2/de not_active Expired - Lifetime
- 2004-04-26 US US10/554,880 patent/US7608720B2/en not_active Expired - Fee Related
- 2004-04-26 KR KR1020117027963A patent/KR101213005B1/ko active IP Right Grant
- 2004-04-26 CN CNB2004800110082A patent/CN100413847C/zh not_active Expired - Lifetime
- 2004-04-26 KR KR1020057020214A patent/KR101130601B1/ko active IP Right Grant
- 2004-04-26 DK DK04739624T patent/DK1620404T3/da active
- 2004-04-26 BR BRPI0409517-0A patent/BRPI0409517A/pt active Search and Examination
- 2004-04-26 PL PL04739624T patent/PL1620404T3/pl unknown
-
2005
- 2005-09-04 IL IL170657A patent/IL170657A/en active IP Right Grant
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI650318B (zh) * | 2017-10-30 | 2019-02-11 | 財團法人工業技術研究院 | 以結晶法純化２，５－呋喃二甲酸的粗產物之方法與聚酯之形成方法 |
| US10344010B2 (en) | 2017-10-30 | 2019-07-09 | Industrial Technology Research Institute | Method for purifying crude of 2,5-furandicarboxylic acid by crystallization |
Also Published As
| Publication number | Publication date |
|---|---|
| US20060235229A1 (en) | 2006-10-19 |
| EP1620404A1 (en) | 2006-02-01 |
| EP1620404B1 (en) | 2007-03-07 |
| US7608720B2 (en) | 2009-10-27 |
| BRPI0409517A (pt) | 2006-04-18 |
| IL170657A (en) | 2011-02-28 |
| WO2004096772A1 (en) | 2004-11-11 |
| KR20060005396A (ko) | 2006-01-17 |
| CN100413847C (zh) | 2008-08-27 |
| DE602004005175T2 (de) | 2007-12-20 |
| GB0309631D0 (en) | 2003-06-04 |
| TWI359139B (en) | 2012-03-01 |
| JP4718446B2 (ja) | 2011-07-06 |
| KR20110133063A (ko) | 2011-12-09 |
| DE602004005175D1 (de) | 2007-04-19 |
| KR101130601B1 (ko) | 2012-04-02 |
| DK1620404T3 (da) | 2007-04-02 |
| CN1777588A (zh) | 2006-05-24 |
| PL1620404T3 (pl) | 2007-07-31 |
| ES2279383T3 (es) | 2007-08-16 |
| JP2006524665A (ja) | 2006-11-02 |
| KR101213005B1 (ko) | 2012-12-18 |
| ATE356116T1 (de) | 2007-03-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4A | Expiration of patent term of an invention patent |