SK285295B6 - Farmaceutický prípravok s riadeným uvoľňovaním účinnej látky skladajúci sa z jadra obsahujúceho účinnú látku a soľ organickej kyseliny a z vonkajšieho obalu - Google Patents

Farmaceutický prípravok s riadeným uvoľňovaním účinnej látky skladajúci sa z jadra obsahujúceho účinnú látku a soľ organickej kyseliny a z vonkajšieho obalu Download PDF

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Publication number
SK285295B6
SK285295B6 SK426-2001A SK4262001A SK285295B6 SK 285295 B6 SK285295 B6 SK 285295B6 SK 4262001 A SK4262001 A SK 4262001A SK 285295 B6 SK285295 B6 SK 285295B6
Authority
SK
Slovakia
Prior art keywords
meth
acid
acrylate
weight
methacrylic acid
Prior art date
Application number
SK426-2001A
Other languages
English (en)
Slovak (sk)
Other versions
SK4262001A3 (en
Inventor
Hans-Ulrich Petereit
Thomas Beckert
Eva Lynenskjold
Original Assignee
R�Hm Gmbh & Co. Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by R�Hm Gmbh & Co. Kg filed Critical R�Hm Gmbh & Co. Kg
Publication of SK4262001A3 publication Critical patent/SK4262001A3/sk
Publication of SK285295B6 publication Critical patent/SK285295B6/sk

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
    • A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
SK426-2001A 1998-10-02 1999-09-28 Farmaceutický prípravok s riadeným uvoľňovaním účinnej látky skladajúci sa z jadra obsahujúceho účinnú látku a soľ organickej kyseliny a z vonkajšieho obalu SK285295B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19845358A DE19845358A1 (de) 1998-10-02 1998-10-02 Überzogene Arzneiformen mit kontrollierter Wirkstoffabgabe
PCT/EP1999/007179 WO2000019984A2 (de) 1998-10-02 1999-09-28 Überzogene arzneiformen mit kontrollierter wirkstoffabgabe

Publications (2)

Publication Number Publication Date
SK4262001A3 SK4262001A3 (en) 2002-10-08
SK285295B6 true SK285295B6 (sk) 2006-10-05

Family

ID=7883150

Family Applications (1)

Application Number Title Priority Date Filing Date
SK426-2001A SK285295B6 (sk) 1998-10-02 1999-09-28 Farmaceutický prípravok s riadeným uvoľňovaním účinnej látky skladajúci sa z jadra obsahujúceho účinnú látku a soľ organickej kyseliny a z vonkajšieho obalu

Country Status (16)

Country Link
US (1) US6878387B1 (zh)
EP (1) EP1117387B1 (zh)
JP (1) JP4615124B2 (zh)
KR (1) KR100657779B1 (zh)
CN (1) CN1182840C (zh)
AT (1) ATE286724T1 (zh)
AU (1) AU6197499A (zh)
BR (1) BR9913104B1 (zh)
CA (1) CA2346062C (zh)
DE (2) DE19845358A1 (zh)
ES (1) ES2234303T3 (zh)
HK (1) HK1058152A1 (zh)
MX (1) MXPA01003392A (zh)
PL (1) PL193899B1 (zh)
SK (1) SK285295B6 (zh)
WO (1) WO2000019984A2 (zh)

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WO2005009364A2 (en) 2003-07-21 2005-02-03 Advancis Pharmaceutical Corporation Antibiotic product, use and formulation thereof
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WO2005016278A2 (en) 2003-08-12 2005-02-24 Advancis Pharmaceuticals Corporation Antibiotic product, use and formulation thereof
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DE10353196A1 (de) * 2003-11-13 2005-06-16 Röhm GmbH & Co. KG Mehrschichtige Arzneiform mit einer die Abgabe einer modulatorischen Substanz beeinflussenden Matrix
DE10353186A1 (de) * 2003-11-13 2005-06-16 Röhm GmbH & Co. KG Mehrschichtige Arzneiform, enthaltend eine in Bezug auf die Wirkstoffabgabe modulatorisch wirkende Substanz
TWI388280B (zh) 2004-01-23 2013-03-11 Univ Pennsylvania 面上兩性之聚芳基和聚芳炔基聚合物與寡聚物及其用途
JP2008505124A (ja) 2004-07-02 2008-02-21 アドバンシス ファーマスーティカル コーポレイション パルス送達用錠剤
JP5027659B2 (ja) * 2004-07-23 2012-09-19 ザ トラスティーズ オブ ザ ユニバーシティ オブ ペンシルバニア 抗菌コポリマーおよびその使用
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KR20080002789A (ko) * 2005-03-29 2008-01-04 에보니크 룀 게엠베하 조절 물질의 전달에 영향을 미치는 매트릭스를 가지는펠렛을 포함하는 다중 미립자 제약 형태
US8357394B2 (en) 2005-12-08 2013-01-22 Shionogi Inc. Compositions and methods for improved efficacy of penicillin-type antibiotics
US8778924B2 (en) 2006-12-04 2014-07-15 Shionogi Inc. Modified release amoxicillin products
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ATE553754T1 (de) 2006-08-18 2012-05-15 Evonik Roehm Gmbh Pharmazeutische zusammensetzung mit kontrollierter wirkstoffabgabe für wirkstoffe mit guter löslichkeit in wasser
HUE043474T2 (hu) * 2008-01-10 2019-08-28 Evonik Roehm Gmbh Bevont gyógyszerészeti vagy gyógyhatású étrend-kiegészítõ készítmény javított pulzáló hatóanyag-felszabadulással
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Also Published As

Publication number Publication date
HK1058152A1 (en) 2004-05-07
JP4615124B2 (ja) 2011-01-19
SK4262001A3 (en) 2002-10-08
KR20010075502A (ko) 2001-08-09
ES2234303T3 (es) 2005-06-16
CA2346062C (en) 2008-09-16
CN1182840C (zh) 2005-01-05
AU6197499A (en) 2000-04-26
BR9913104B1 (pt) 2010-11-30
MXPA01003392A (es) 2003-07-21
WO2000019984A2 (de) 2000-04-13
CA2346062A1 (en) 2000-04-13
US6878387B1 (en) 2005-04-12
EP1117387A2 (de) 2001-07-25
JP2002526401A (ja) 2002-08-20
BR9913104A (pt) 2001-05-08
EP1117387B1 (de) 2005-01-12
ATE286724T1 (de) 2005-01-15
WO2000019984A3 (de) 2000-07-20
CN1446083A (zh) 2003-10-01
DE59911452D1 (de) 2005-02-17
DE19845358A1 (de) 2000-04-06
PL347780A1 (en) 2002-04-22
KR100657779B1 (ko) 2006-12-21
PL193899B1 (pl) 2007-03-30

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Legal Events

Date Code Title Description
PC4A Assignment and transfer of rights

Owner name: ROEHM GMBH, DARMSTADT, DE

Free format text: FORMER OWNER: ROEHM GMBH & CO. KG, DARMSTADT, DE

Effective date: 20100407

TC4A Change of owner's name

Owner name: EVONIK ROEHM GMBH, DARMSTADT, DE

Effective date: 20100407

MM4A Patent lapsed due to non-payment of maintenance fees

Effective date: 20180928