SK18312000A3 - Aza-heterocyklické zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie - Google Patents
Aza-heterocyklické zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie Download PDFInfo
- Publication number
- SK18312000A3 SK18312000A3 SK1831-2000A SK18312000A SK18312000A3 SK 18312000 A3 SK18312000 A3 SK 18312000A3 SK 18312000 A SK18312000 A SK 18312000A SK 18312000 A3 SK18312000 A3 SK 18312000A3
- Authority
- SK
- Slovakia
- Prior art keywords
- carboxylic acid
- straight
- branched
- alkyl
- alkenyl
- Prior art date
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PCT/US1998/025573 WO1999062881A1 (en) | 1998-06-03 | 1998-12-03 | Aza-heterocyclic compounds used to treat neurological disorders and hair loss |
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SK18312000A3 true SK18312000A3 (sk) | 2001-06-11 |
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SK1831-2000A SK18312000A3 (sk) | 1998-06-03 | 1998-12-03 | Aza-heterocyklické zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie |
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EP (1) | EP1084107B1 (de) |
JP (2) | JP4722288B2 (de) |
KR (1) | KR20010052487A (de) |
CN (1) | CN100351230C (de) |
AT (1) | ATE359267T1 (de) |
AU (1) | AU772472B2 (de) |
BG (1) | BG105015A (de) |
BR (1) | BR9815920A (de) |
CA (1) | CA2333963C (de) |
DE (1) | DE69837564T2 (de) |
EA (1) | EA008723B1 (de) |
HU (1) | HUP0102923A3 (de) |
IL (1) | IL140042A0 (de) |
NO (1) | NO320643B1 (de) |
NZ (1) | NZ508462A (de) |
PL (1) | PL194262B1 (de) |
SK (1) | SK18312000A3 (de) |
WO (1) | WO1999062881A1 (de) |
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US6331537B1 (en) * | 1998-06-03 | 2001-12-18 | Gpi Nil Holdings, Inc. | Carboxylic acids and carboxylic acid isosteres of N-heterocyclic compounds |
JP4708567B2 (ja) * | 1998-12-03 | 2011-06-22 | ジーピーアイ ニル ホールディングス インコーポレイテッド | N−複素環化合物のカルボン酸およびカルボン酸アイソスター |
AU3587300A (en) * | 1999-02-03 | 2000-08-25 | Schering Aktiengesellschaft | Ether derivatives |
US6284779B1 (en) * | 1999-02-03 | 2001-09-04 | Schering Aktiiengesellschaft | Heteroaromatic compounds |
JP2000302757A (ja) * | 1999-04-16 | 2000-10-31 | Shiseido Co Ltd | N−置換ピペリジン誘導体 |
CA2379149A1 (en) | 1999-07-09 | 2001-01-18 | Ortho-Mcneil Pharmaceutical, Inc. | Neurotrophic pyrrolidines and piperidines, and related compositions and methods |
AU6913700A (en) * | 1999-08-18 | 2001-03-13 | Schering Aktiengesellschaft | Piperidine and pyrrolidine derivatives displaying neuronal activity |
US7598278B2 (en) | 2002-04-11 | 2009-10-06 | L'oreal | Administration of pyridinedicarboxylic acid compounds for stimulating or inducing the growth of human keratinous fibers and/or arresting their loss |
EP2283006B1 (de) | 2008-04-24 | 2015-02-25 | F2G Limited | Pyrrole als antipilzmittel |
TWI534142B (zh) * | 2011-03-15 | 2016-05-21 | 大正製藥股份有限公司 | Azole derivatives |
US10167259B2 (en) * | 2013-06-14 | 2019-01-01 | The Board Of Regents Of The University Of Texas System | Allosteric inhibitors of proteasome and methods of use thereof |
ES2694637T3 (es) | 2014-11-21 | 2018-12-26 | F2G Limited | Agentes antifúngicos |
FR3030248B1 (fr) | 2014-12-22 | 2018-03-23 | L'oreal | Association derive d'acide pyridine-dicarboxylique/agent anti-oxydant particulier |
GB201609222D0 (en) | 2016-05-25 | 2016-07-06 | F2G Ltd | Pharmaceutical formulation |
US11819503B2 (en) | 2019-04-23 | 2023-11-21 | F2G Ltd | Method of treating coccidioides infection |
Family Cites Families (10)
Publication number | Priority date | Publication date | Assignee | Title |
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US5192773A (en) * | 1990-07-02 | 1993-03-09 | Vertex Pharmaceuticals, Inc. | Immunosuppressive compounds |
US5798355A (en) * | 1995-06-07 | 1998-08-25 | Gpi Nil Holdings, Inc. | Inhibitors of rotamase enzyme activity |
JP4470226B2 (ja) * | 1994-08-18 | 2010-06-02 | アリアド・ファーマシューティカルズ・インコーポレイテッド | 新規な多量体化剤 |
US5859031A (en) * | 1995-06-07 | 1999-01-12 | Gpi Nil Holdings, Inc. | Small molecule inhibitors of rotamase enzyme activity |
US5614547A (en) * | 1995-06-07 | 1997-03-25 | Guilford Pharmaceuticals Inc. | Small molecule inhibitors of rotamase enzyme |
AU731826B2 (en) * | 1996-02-28 | 2001-04-05 | Ariad Pharmaceuticals, Inc. | Synthetic Multimerizing Agents |
US5786378A (en) * | 1996-09-25 | 1998-07-28 | Gpi Nil Holdings, Inc. | Heterocyclic thioesters |
US5846979A (en) * | 1997-02-28 | 1998-12-08 | Gpi Nil Holdings, Inc. | N-oxides of heterocyclic esters, amides, thioesters, and ketones |
US5945441A (en) * | 1997-06-04 | 1999-08-31 | Gpi Nil Holdings, Inc. | Pyrrolidine carboxylate hair revitalizing agents |
AU742040C (en) * | 1997-09-24 | 2003-10-02 | Amgen, Inc. | Method for preventing and treating hearing loss using sensorineurotrophic compounds |
-
1998
- 1998-12-03 CA CA002333963A patent/CA2333963C/en not_active Expired - Fee Related
- 1998-12-03 AT AT98961866T patent/ATE359267T1/de not_active IP Right Cessation
- 1998-12-03 IL IL14004298A patent/IL140042A0/xx unknown
- 1998-12-03 AU AU17081/99A patent/AU772472B2/en not_active Ceased
- 1998-12-03 KR KR1020007013614A patent/KR20010052487A/ko active Search and Examination
- 1998-12-03 NZ NZ508462A patent/NZ508462A/xx unknown
- 1998-12-03 HU HU0102923A patent/HUP0102923A3/hu unknown
- 1998-12-03 DE DE69837564T patent/DE69837564T2/de not_active Expired - Fee Related
- 1998-12-03 EP EP98961866A patent/EP1084107B1/de not_active Expired - Lifetime
- 1998-12-03 WO PCT/US1998/025573 patent/WO1999062881A1/en active IP Right Grant
- 1998-12-03 JP JP2000552093A patent/JP4722288B2/ja not_active Expired - Fee Related
- 1998-12-03 SK SK1831-2000A patent/SK18312000A3/sk unknown
- 1998-12-03 CN CNB988140993A patent/CN100351230C/zh not_active Expired - Fee Related
- 1998-12-03 BR BR9815920-8A patent/BR9815920A/pt not_active Application Discontinuation
- 1998-12-03 EA EA200001145A patent/EA008723B1/ru not_active IP Right Cessation
- 1998-12-03 PL PL98344580A patent/PL194262B1/pl unknown
-
2000
- 2000-11-21 NO NO20005903A patent/NO320643B1/no unknown
- 2000-12-01 BG BG105015A patent/BG105015A/xx unknown
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2010
- 2010-08-13 JP JP2010181409A patent/JP2011006439A/ja active Pending
Also Published As
Publication number | Publication date |
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WO1999062881A1 (en) | 1999-12-09 |
AU772472B2 (en) | 2004-04-29 |
CA2333963C (en) | 2010-02-02 |
HUP0102923A2 (hu) | 2001-12-28 |
BR9815920A (pt) | 2001-02-20 |
PL194262B1 (pl) | 2007-05-31 |
NO20005903D0 (no) | 2000-11-21 |
JP2002516905A (ja) | 2002-06-11 |
AU1708199A (en) | 1999-12-20 |
NO320643B1 (no) | 2006-01-09 |
WO1999062881A8 (en) | 2000-07-27 |
EP1084107B1 (de) | 2007-04-11 |
PL344580A1 (en) | 2001-11-05 |
JP2011006439A (ja) | 2011-01-13 |
NZ508462A (en) | 2004-02-27 |
EA008723B1 (ru) | 2007-06-29 |
CN100351230C (zh) | 2007-11-28 |
DE69837564T2 (de) | 2007-12-27 |
HUP0102923A3 (en) | 2002-01-28 |
NO20005903L (no) | 2001-02-02 |
EA200001145A1 (ru) | 2001-10-22 |
KR20010052487A (ko) | 2001-06-25 |
IL140042A0 (en) | 2002-02-10 |
ATE359267T1 (de) | 2007-05-15 |
CN1336915A (zh) | 2002-02-20 |
BG105015A (en) | 2001-08-31 |
CA2333963A1 (en) | 1999-12-09 |
DE69837564D1 (de) | 2007-05-24 |
EP1084107A1 (de) | 2001-03-21 |
JP4722288B2 (ja) | 2011-07-13 |
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