SI2501680T1 - Postopek za pripravo marbofloksacina in njegovih intermediatov - Google Patents

Postopek za pripravo marbofloksacina in njegovih intermediatov

Info

Publication number
SI2501680T1
SI2501680T1 SI201031175A SI201031175A SI2501680T1 SI 2501680 T1 SI2501680 T1 SI 2501680T1 SI 201031175 A SI201031175 A SI 201031175A SI 201031175 A SI201031175 A SI 201031175A SI 2501680 T1 SI2501680 T1 SI 2501680T1
Authority
SI
Slovenia
Prior art keywords
marbofloxacin
preparation
Prior art date
Application number
SI201031175A
Other languages
English (en)
Inventor
Rok Zupet
Jernej Iskra
Milos Ruzic
Anica Pecavar
Ivanka Kolenc
Joze Pucelj
Igor Plaper
Original Assignee
Krka, Tovarna Zdravil, D.D., Novo Mesto
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Krka, Tovarna Zdravil, D.D., Novo Mesto filed Critical Krka, Tovarna Zdravil, D.D., Novo Mesto
Publication of SI2501680T1 publication Critical patent/SI2501680T1/sl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/58Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
SI201031175A 2009-11-19 2010-11-19 Postopek za pripravo marbofloksacina in njegovih intermediatov SI2501680T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
SI200900366 2009-11-19
EP10156733A EP2332916A3 (en) 2009-11-19 2010-03-17 A process for a preparation of marbofloxacin and intermediate thereof
PCT/EP2010/067828 WO2011061292A1 (en) 2009-11-19 2010-11-19 A process for a preparation of marbofloxacin and intermediate thereof
EP10777039.8A EP2501680B1 (en) 2009-11-19 2010-11-19 A process for a preparation of marbofloxacin and intermediate thereof

Publications (1)

Publication Number Publication Date
SI2501680T1 true SI2501680T1 (sl) 2016-08-31

Family

ID=43480997

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201031175A SI2501680T1 (sl) 2009-11-19 2010-11-19 Postopek za pripravo marbofloksacina in njegovih intermediatov

Country Status (5)

Country Link
EP (2) EP2332916A3 (sl)
CN (1) CN102712598A (sl)
EA (1) EA021239B1 (sl)
SI (1) SI2501680T1 (sl)
WO (1) WO2011061292A1 (sl)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN105130892B (zh) * 2015-08-19 2016-08-17 海门慧聚药业有限公司 马波沙星关键中间体的制备
CN105198905A (zh) * 2015-10-14 2015-12-30 海门慧聚药业有限公司 一种纯化制备超纯马波沙星的方法
CN107056811A (zh) * 2017-04-20 2017-08-18 山东方明邦嘉制药有限公司 一种马波沙星的精制方法
CN107383058B (zh) * 2017-08-28 2019-07-26 海门慧聚药业有限公司 马波沙星的制备
CN107522718B (zh) * 2017-09-14 2019-11-08 浙江国邦药业有限公司 一种马波沙星的合成方法
US20230346736A1 (en) * 2020-06-23 2023-11-02 Laila Nutraceuticals Water soluble 3-o-acetyl-11-keto-b-boswellic acid and metal ion compositions, process for their preparation and uses thereof
CN114249749B (zh) * 2022-01-08 2024-03-22 天象生物药业邢台有限责任公司 一种马波沙星甲酸盐的转化方法

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3409922A1 (de) 1984-03-17 1985-09-26 Bayer Ag, 5090 Leverkusen 1,7-diamino-1,4-dihydro-4-oxo-3-(aza)chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie ihre verwendung bei der bekaempfung bakterieller erkrankungen
US4604401A (en) 1984-07-20 1986-08-05 Warner-Lambert Company Antibacterial agents III
EP0259804B1 (de) 1986-09-12 1993-11-18 F. Hoffmann-La Roche Ag Pyrido [3,2,1-ij]-1,3,4-benzoxadiazinderivate, Verfahren zu deren Herstellung, entsprechende pharmazeutische Präparate und im Verfahren verwendbare Zwischenprodukte
ES2125895T3 (es) 1991-03-22 1999-03-16 Phillips Petroleum Co Alfa-olefinas superiores ramificadas, injertadas, reforzadas con vidrio.
NZ261106A (en) * 1993-01-23 1997-06-24 Pfizer Preparation of 6-fluoro-1,4-dihydro-8-hydroxy-1-(n-methylamino)-7-(4-methylpiperaz in-1-yl)-4-oxoquinoline-3-carboxylic acid salts; use in preparing the corresponding pyrido [3,2,1-ij]-1,3,4-benzoxadiazine
IT1313683B1 (it) 1999-11-25 2002-09-09 Fabbrica Italiana Sintetici Spa Procedimento per la preparazione di marbofloxacina.
US20020122824A1 (en) 2001-01-24 2002-09-05 Francisco Cabrera Solid phase dispersion of quinolone-or naphthyridonecarboxylic acids
FR2896416B1 (fr) 2006-01-24 2010-08-13 Vetoquinol Composition anti-infectieuse comprenant un compose de type pyrido (3,2,1-ij)-benzoxadiazine
DE102006010642A1 (de) 2006-03-08 2007-09-27 Bayer Healthcare Aktiengesellschaft Arzneimittelformulierungen, enthaltend Fluorchinolone
DE102006010643A1 (de) 2006-03-08 2007-09-13 Bayer Healthcare Aktiengesellschaft Arzneimittel enthaltend Fluorchinolone
WO2008030469A2 (en) 2006-09-07 2008-03-13 Merial Limited Soft chewable, tablet, and long-acting injectable veterinary antibiotic formulations

Also Published As

Publication number Publication date
EP2501680B1 (en) 2016-02-10
WO2011061292A1 (en) 2011-05-26
EA201290361A1 (ru) 2012-11-30
EA021239B1 (ru) 2015-05-29
EP2501680A1 (en) 2012-09-26
EP2332916A2 (en) 2011-06-15
CN102712598A (zh) 2012-10-03
EP2332916A3 (en) 2011-08-03

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