SG20887G - Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives - Google Patents

Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives

Info

Publication number
SG20887G
SG20887G SG208/87A SG20887A SG20887G SG 20887 G SG20887 G SG 20887G SG 208/87 A SG208/87 A SG 208/87A SG 20887 A SG20887 A SG 20887A SG 20887 G SG20887 G SG 20887G
Authority
SG
Singapore
Prior art keywords
derivatives
trans
processes
medicaments containing
preparation intermediates
Prior art date
Application number
SG208/87A
Other languages
English (en)
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of SG20887G publication Critical patent/SG20887G/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SG208/87A 1979-07-09 1987-02-26 Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives SG20887G (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US5572879A 1979-07-09 1979-07-09
US06/142,903 US4281127A (en) 1979-07-09 1980-04-23 Trans-3-(4-oxo-4H-quinazolin-3-yl)-2-propenoic acid derivatives

Publications (1)

Publication Number Publication Date
SG20887G true SG20887G (en) 1988-09-16

Family

ID=26734565

Family Applications (1)

Application Number Title Priority Date Filing Date
SG208/87A SG20887G (en) 1979-07-09 1987-02-26 Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives

Country Status (21)

Country Link
US (1) US4281127A (pt)
EP (1) EP0023594B1 (pt)
AR (1) AR226854A1 (pt)
AU (1) AU521014B2 (pt)
CA (1) CA1134825A (pt)
DE (1) DE3067830D1 (pt)
DK (1) DK150483C (pt)
ES (2) ES8106302A1 (pt)
FI (1) FI74279C (pt)
GR (1) GR65952B (pt)
HK (1) HK52187A (pt)
HU (1) HU184797B (pt)
IE (1) IE49938B1 (pt)
IL (1) IL60514A (pt)
MC (1) MC1333A1 (pt)
NO (1) NO154426C (pt)
NZ (1) NZ194259A (pt)
PH (1) PH16413A (pt)
PT (1) PT71512B (pt)
SG (1) SG20887G (pt)
YU (1) YU42348B (pt)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4599336A (en) * 1983-08-08 1986-07-08 Hoffmann-La Roche Inc. Derivatives of (E)-3-(4-oxo-4H-quinazolin-3-yl)-2-propenamide
GB9404485D0 (en) 1994-03-09 1994-04-20 Cancer Res Campaign Tech Benzamide analogues
US6706721B1 (en) * 1998-04-29 2004-03-16 Osi Pharmaceuticals, Inc. N-(3-ethynylphenylamino)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine mesylate anhydrate and monohydrate
US7230000B1 (en) 1999-10-27 2007-06-12 Cytokinetics, Incorporated Methods and compositions utilizing quinazolinones
US6545004B1 (en) 1999-10-27 2003-04-08 Cytokinetics, Inc. Methods and compositions utilizing quinazolinones
US7087613B2 (en) * 1999-11-11 2006-08-08 Osi Pharmaceuticals, Inc. Treating abnormal cell growth with a stable polymorph of N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine hydrochloride
UA74803C2 (uk) 1999-11-11 2006-02-15 Осі Фармасьютікалз, Інк. Стійкий поліморф гідрохлориду n-(3-етинілфеніл)-6,7-біс(2-метоксіетокси)-4-хіназолінаміну, спосіб його одержання (варіанти) та фармацевтичне застосування
JP2005529076A (ja) * 2002-02-15 2005-09-29 サイトキネティクス・インコーポレーテッド キナゾリノンの合成
AU2003270015A1 (en) 2002-05-09 2003-12-02 Cytokinetics, Inc. Compounds, compositions, and methods
MXPA04011074A (es) * 2002-05-09 2005-06-08 Cytokinetics Inc Compuestos de pirimidinona, composiciones y metodos.
EP1513820A4 (en) * 2002-05-23 2006-09-13 Cytokinetics Inc COMPOUNDS, COMPOSITIONS AND METHODS
AU2003236527A1 (en) * 2002-06-14 2003-12-31 Cytokinetics, Inc. Compounds, compositions, and methods
US7211580B2 (en) * 2002-07-23 2007-05-01 Cytokinetics, Incorporated Compounds, compositions, and methods
JP2005536553A (ja) * 2002-08-21 2005-12-02 サイトキネティクス・インコーポレーテッド 化合物、組成物および方法
WO2004034972A2 (en) * 2002-09-30 2004-04-29 Cytokinetics, Inc. Compounds, compositions, and methods
US20050197327A1 (en) * 2003-11-03 2005-09-08 Gustave Bergnes Compounds, compositions, and methods
US20050148593A1 (en) * 2003-11-07 2005-07-07 Gustave Bergnes Compounds, compositions, and methods
US7439254B2 (en) * 2003-12-08 2008-10-21 Cytokinetics, Inc. Compounds, compositions, and methods
UY29198A1 (es) * 2004-11-09 2006-05-31 Cancer Rec Tech Ltd Derivados sustituidos de quinazolinona y derivados sustituidos de quinazolina-2, 4-diona, composiciones conteniéndolos, procedimientos de preparación y aplicaciones

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2786055A (en) * 1955-02-10 1957-03-19 Mallinckrodt Chemical Works Carboxyalkyl-iodoquinazolones
US3517005A (en) * 1967-10-26 1970-06-23 Pfizer & Co C Certain 2- and 4-substituted quinazolines
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones

Also Published As

Publication number Publication date
IL60514A (en) 1985-03-31
YU42348B (en) 1988-08-31
PT71512A (en) 1980-08-01
IE49938B1 (en) 1986-01-08
MC1333A1 (fr) 1981-04-21
FI74279C (fi) 1988-01-11
EP0023594B1 (de) 1984-05-16
FI74279B (fi) 1987-09-30
HK52187A (en) 1987-07-17
AR226854A1 (es) 1982-08-31
NO802056L (no) 1981-01-12
ES493203A0 (es) 1981-05-16
DK294780A (da) 1981-01-10
CA1134825A (en) 1982-11-02
IL60514A0 (en) 1980-09-16
GR65952B (pt) 1981-01-09
ES499035A0 (es) 1982-09-16
IE801412L (en) 1981-01-09
DK150483C (da) 1987-11-09
NZ194259A (en) 1984-09-28
ES8106302A1 (es) 1981-05-16
NO154426C (no) 1986-09-17
AU521014B2 (en) 1982-03-11
DE3067830D1 (en) 1984-06-20
PT71512B (en) 1981-12-11
US4281127A (en) 1981-07-28
NO154426B (no) 1986-06-09
HU184797B (en) 1984-10-29
AU6024480A (en) 1981-03-12
ES8207155A1 (es) 1982-09-16
EP0023594A1 (de) 1981-02-11
FI802195A (fi) 1981-01-10
YU176680A (en) 1984-12-31
PH16413A (en) 1983-09-29
DK150483B (da) 1987-03-09

Similar Documents

Publication Publication Date Title
DE3067868D1 (en) Imidazodiazepine derivatives, process and intermediates for their preparation, medicaments containing them and their therapeutic application
DE2960222D1 (en) Phenoxyalkylcarboxylic-acid derivatives, process for their preparation and medicaments containing them
DE2860330D1 (en) 3,4,5-trihydroxypiperidine derivatives, process for their preparation and medicaments and fodder containing them
DE3062971D1 (en) Derivatives of tetraline, their preparation and medicaments containing these compounds
SG20887G (en) Trans-quinazoline derivatives processes for their preparation intermediates and medicaments containing these derivatives
GB2054566B (en) 1-aryl-4-arylsulphonyl-3-aminopropoxy-1h-pyrazoles medicaments containing them and processes for their preparation
GB2046259B (en) Amino-alcohol derivatives and pharmaceutical compositions containing them
DE3071581D1 (en) Substituted tetraazatricyclic compounds, process for their preparation, their use and medicines containing them
GB2064527B (en) Moranoline derivatives and process for preparation thereof
NZ193078A (en) Derivatives of 9-aminoalkyl-flyorene medicinal preparations
DE2961983D1 (en) Pyrrolidine-2-methanol derivatives, process for their preparation and medicaments containing them
GB2063874B (en) Triazole derivatives processes for the preparation thereof and pharmaceutical compositions containing them
IL61371A (en) Medicaments containing phenyloxoalkanoic acids,some new such acids and processes for their preparation
PT73061B (en) Process for the preparation of new derivatives of taurina and its pharmaceutical use
ZA80922B (en) Pyrazole derivatives pharmaceutical formulations containing these derivatives and processes for their preparation
IL52611A0 (en) 2-benzylpyrrolidines process for their preparation and medicaments containing them
IL60376A0 (en) 3-methyleneazetidine derivatives and pharmaceutical compositions containing them
IL60892A (en) Triophosphonate derivatives and their use as insecticides and nematocides
GB2055093B (en) Substituted phenylacetylguanidine derivatives and processes for their preparation
DE2964198D1 (en) Indanamine derivatives, process for their preparation and medicaments containing them
GB2106504B (en) 9-bromo-indoloquinolisine derivatives and processes for their preparation
NZ193557A (en) 4-phenylchroman derivatives intermediates and pharmaceutical compositions
EP0034831A3 (en) Substituted phenoxy-aminopropanol derivatives, intermediates and process for their preparation, medicament containing them, and their use
DE3062972D1 (en) Pyridazopyridazine derivatives, processes for their preparation and pharmaceutical compositions containing these pyridazopyridazine derivatives
EP0025109A3 (en) 1-benzoxepin-5(2h)-one derivatives and their salts, processes and intermediates for their preparation and medicaments containing them