SG181850A1 - Inhibitors of receptor tyrosine kinases (rtk) and methods of use thereof - Google Patents
Inhibitors of receptor tyrosine kinases (rtk) and methods of use thereof Download PDFInfo
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- SG181850A1 SG181850A1 SG2012045803A SG2012045803A SG181850A1 SG 181850 A1 SG181850 A1 SG 181850A1 SG 2012045803 A SG2012045803 A SG 2012045803A SG 2012045803 A SG2012045803 A SG 2012045803A SG 181850 A1 SG181850 A1 SG 181850A1
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/705—Receptors; Cell surface antigens; Cell surface determinants
- C07K14/71—Receptors; Cell surface antigens; Cell surface determinants for growth factors; for growth regulators
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K16/00—Immunoglobulins [IGs], e.g. monoclonal or polyclonal antibodies
-
- G—PHYSICS
- G01—MEASURING; TESTING
- G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
- G01N2500/00—Screening for compounds of potential therapeutic value
- G01N2500/04—Screening involving studying the effect of compounds C directly on molecule A (e.g. C are potential ligands for a receptor A, or potential substrates for an enzyme A)
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Organic Chemistry (AREA)
- Molecular Biology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biomedical Technology (AREA)
- Hematology (AREA)
- Genetics & Genomics (AREA)
- Cell Biology (AREA)
- Urology & Nephrology (AREA)
- Gastroenterology & Hepatology (AREA)
- General Chemical & Material Sciences (AREA)
- Zoology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biophysics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biotechnology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Food Science & Technology (AREA)
- Pathology (AREA)
- Physical Education & Sports Medicine (AREA)
- Microbiology (AREA)
- Epidemiology (AREA)
- Toxicology (AREA)
- Physics & Mathematics (AREA)
- Analytical Chemistry (AREA)
- General Physics & Mathematics (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33595010P | 2010-01-14 | 2010-01-14 | |
| PCT/US2011/021109 WO2011088196A2 (en) | 2010-01-14 | 2011-01-13 | Inhibitors of receptor tyrosine kinases (rtk) and methods of use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG181850A1 true SG181850A1 (en) | 2012-08-30 |
Family
ID=44304965
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG2012045803A SG181850A1 (en) | 2010-01-14 | 2011-01-13 | Inhibitors of receptor tyrosine kinases (rtk) and methods of use thereof |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US20120328599A1 (enExample) |
| EP (1) | EP2523679A4 (enExample) |
| JP (1) | JP2013517282A (enExample) |
| KR (1) | KR20120130758A (enExample) |
| CN (1) | CN102762221A (enExample) |
| AU (1) | AU2011205297A1 (enExample) |
| BR (1) | BR112012016992A2 (enExample) |
| CA (1) | CA2786276A1 (enExample) |
| IL (1) | IL220206A0 (enExample) |
| IN (1) | IN2012DN05017A (enExample) |
| MX (1) | MX2012008222A (enExample) |
| RU (1) | RU2012134637A (enExample) |
| SG (1) | SG181850A1 (enExample) |
| WO (1) | WO2011088196A2 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103694351A (zh) | 2007-06-05 | 2014-04-02 | 耶鲁大学 | 受体酪氨酸激酶抑制剂及其使用方法 |
| EP3763740A1 (en) | 2011-01-26 | 2021-01-13 | Celldex Therapeutics, Inc. | Anti-kit antibodies and uses thereof |
| CN104812775B (zh) | 2012-07-25 | 2019-05-03 | 塞尔德克斯医疗公司 | 抗kit抗体及其用途 |
| US20150344855A1 (en) | 2013-01-16 | 2015-12-03 | INSERM (Institut National de la Santé et de la Recherche Médicale | A Soluble Fibroblast Growth Factor Receptor 3 (FGR3) Polypeptide For Use In The Prevention Or Treatment Of Skeletal Growth Retardation Disorders |
| US10300116B2 (en) | 2013-06-10 | 2019-05-28 | Ansun Biopharma, Inc. | Treatment for BK polyomavirus infection |
| PL3708583T3 (pl) | 2013-08-01 | 2022-06-06 | Five Prime Therapeutics, Inc. | Afukozylowane przeciwciała anty-fgfr2iiib |
| SG11201602069WA (en) | 2013-10-18 | 2016-04-28 | Eisai R&D Man Co Ltd | Pyrimidine fgfr4 inhibitors |
| WO2015179737A2 (en) | 2014-05-23 | 2015-11-26 | Kolltan Pharmaceuticals, Inc. | Treatment of eosinophil or mast cell related disorders |
| SG10201810057UA (en) | 2015-04-14 | 2018-12-28 | Eisai R&D Man Co Ltd | Crystalline fgfr4 inhibitor compound and uses thereof |
| JP7349787B2 (ja) | 2015-11-23 | 2023-09-25 | ファイヴ プライム セラピューティクス インク | 癌治療におけるｆｇｆｒ２阻害剤単独または免疫刺激剤との組み合わせ |
| US11357769B2 (en) | 2016-05-10 | 2022-06-14 | Eisai R&D Management Co., Ltd. | Drug combinations for reducing cell viability and/or cell proliferation |
| CN110129300B (zh) * | 2016-06-02 | 2021-08-03 | 天津科技大学 | 一种磷脂酶d |
| SI3481859T1 (sl) | 2016-07-07 | 2022-07-29 | Inserm (Institut National De La Sante Et De La Recherche Medicale) | Topni polipeptidi receptorja 3 fibroblastnega rastnega faktorja (SFGFR3) in njihove uporabe |
| JP7299842B2 (ja) | 2017-05-16 | 2023-06-28 | ファイヴ プライム セラピューティクス インク | がん治療における化学療法剤と組み合わせた抗ｆｇｆｒ２抗体 |
| JP2023538098A (ja) | 2020-08-21 | 2023-09-06 | ジェンザイム・コーポレーション | Ｆｇｆｒ３抗体および使用の方法 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8426396B2 (en) * | 2008-01-08 | 2013-04-23 | Shriners Hospitals For Children | Treatment for achondroplasia |
-
2011
- 2011-01-13 IN IN5017DEN2012 patent/IN2012DN05017A/en unknown
- 2011-01-13 MX MX2012008222A patent/MX2012008222A/es not_active Application Discontinuation
- 2011-01-13 AU AU2011205297A patent/AU2011205297A1/en not_active Abandoned
- 2011-01-13 JP JP2012549070A patent/JP2013517282A/ja not_active Withdrawn
- 2011-01-13 WO PCT/US2011/021109 patent/WO2011088196A2/en not_active Ceased
- 2011-01-13 BR BR112012016992A patent/BR112012016992A2/pt not_active IP Right Cessation
- 2011-01-13 RU RU2012134637/10A patent/RU2012134637A/ru not_active Application Discontinuation
- 2011-01-13 CN CN2011800061813A patent/CN102762221A/zh active Pending
- 2011-01-13 EP EP11733365.8A patent/EP2523679A4/en not_active Withdrawn
- 2011-01-13 CA CA2786276A patent/CA2786276A1/en not_active Abandoned
- 2011-01-13 KR KR1020127021221A patent/KR20120130758A/ko not_active Withdrawn
- 2011-01-13 US US13/519,837 patent/US20120328599A1/en not_active Abandoned
- 2011-01-13 SG SG2012045803A patent/SG181850A1/en unknown
-
2012
- 2012-06-06 IL IL220206A patent/IL220206A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011088196A3 (en) | 2011-11-17 |
| BR112012016992A2 (pt) | 2019-09-24 |
| EP2523679A2 (en) | 2012-11-21 |
| CA2786276A1 (en) | 2011-07-21 |
| IN2012DN05017A (enExample) | 2015-10-02 |
| EP2523679A4 (en) | 2013-07-24 |
| CN102762221A (zh) | 2012-10-31 |
| WO2011088196A2 (en) | 2011-07-21 |
| IL220206A0 (en) | 2012-07-31 |
| JP2013517282A (ja) | 2013-05-16 |
| RU2012134637A (ru) | 2014-02-20 |
| KR20120130758A (ko) | 2012-12-03 |
| AU2011205297A1 (en) | 2012-06-28 |
| US20120328599A1 (en) | 2012-12-27 |
| MX2012008222A (es) | 2012-08-17 |
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