SG11201403540RA - Deuterated thiazolidinone analogues as agonists for follicle stimulating hormone receptor - Google Patents
Deuterated thiazolidinone analogues as agonists for follicle stimulating hormone receptorInfo
- Publication number
- SG11201403540RA SG11201403540RA SG11201403540RA SG11201403540RA SG11201403540RA SG 11201403540R A SG11201403540R A SG 11201403540RA SG 11201403540R A SG11201403540R A SG 11201403540RA SG 11201403540R A SG11201403540R A SG 11201403540RA SG 11201403540R A SG11201403540R A SG 11201403540RA
- Authority
- SG
- Singapore
- Prior art keywords
- agonists
- stimulating hormone
- hormone receptor
- follicle stimulating
- analogues
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/14—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61B—DIAGNOSIS; SURGERY; IDENTIFICATION
- A61B17/00—Surgical instruments, devices or methods, e.g. tourniquets
- A61B17/42—Gynaecological or obstetrical instruments or methods
- A61B17/425—Gynaecological or obstetrical instruments or methods for reproduction or fertilisation
- A61B17/435—Gynaecological or obstetrical instruments or methods for reproduction or fertilisation for embryo or ova transplantation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B59/00—Introduction of isotopes of elements into organic compounds ; Labelled organic compounds per se
- C07B59/002—Heterocyclic compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/05—Isotopically modified compounds, e.g. labelled
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Reproductive Health (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Surgery (AREA)
- Pregnancy & Childbirth (AREA)
- Gynecology & Obstetrics (AREA)
- Epidemiology (AREA)
- Endocrinology (AREA)
- Medical Informatics (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Transplantation (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261596417P | 2012-02-08 | 2012-02-08 | |
| PCT/EP2013/000215 WO2013117299A1 (en) | 2012-02-08 | 2013-01-24 | Deuterated thiazolidinone analogues as agonists for follicle stimulating hormone receptor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201403540RA true SG11201403540RA (en) | 2014-07-30 |
Family
ID=47666083
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201403540RA SG11201403540RA (en) | 2012-02-08 | 2013-01-24 | Deuterated thiazolidinone analogues as agonists for follicle stimulating hormone receptor |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20150111933A1 (ko) |
| EP (1) | EP2812320B1 (ko) |
| JP (1) | JP6386382B2 (ko) |
| KR (1) | KR20140120903A (ko) |
| CN (1) | CN104114544A (ko) |
| AU (1) | AU2013218368B2 (ko) |
| BR (1) | BR112014019351A8 (ko) |
| CA (1) | CA2860489C (ko) |
| ES (1) | ES2672326T3 (ko) |
| HK (1) | HK1201837A1 (ko) |
| IL (1) | IL233983B (ko) |
| MX (1) | MX2014009416A (ko) |
| RU (1) | RU2014136334A (ko) |
| SG (1) | SG11201403540RA (ko) |
| WO (1) | WO2013117299A1 (ko) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015196335A1 (en) | 2014-06-23 | 2015-12-30 | Tocopherx, Inc. | Pyrazole compounds as modulators of fshr and uses thereof |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6221335B1 (en) * | 1994-03-25 | 2001-04-24 | Isotechnika, Inc. | Method of using deuterated calcium channel blockers |
| ATE329911T1 (de) | 1998-08-07 | 2006-07-15 | Applied Research Systems | Fsh mimetika zur behandlung von infertilität |
| US6440710B1 (en) * | 1998-12-10 | 2002-08-27 | The Scripps Research Institute | Antibody-catalyzed deuteration, tritiation, dedeuteration or detritiation of carbonyl compounds |
| US6426357B1 (en) | 1999-07-27 | 2002-07-30 | Affymax, Inc. | Antagonists of follicle stimulating hormone activity |
| ATE234299T1 (de) * | 1999-12-03 | 2003-03-15 | Pfizer Prod Inc | Sulfamoylheteroarylpyrazolverbindungen zur verwendung als analgetisches/entzündungshemmendes mittel |
| AU2001278006A1 (en) * | 2000-07-27 | 2002-02-13 | Smithkline Beecham Corporation | Agonists of follicle stimulating hormone activity |
| TW200413273A (en) * | 2002-11-15 | 2004-08-01 | Wako Pure Chem Ind Ltd | Heavy hydrogenation method of heterocyclic rings |
| AU2006299424A1 (en) * | 2005-10-06 | 2007-04-12 | Auspex Pharmaceuticals, Inc. | Deuterated inhibitors of gastric H+, K+-ATPase with enhanced therapeutic properties |
| US7750168B2 (en) * | 2006-02-10 | 2010-07-06 | Sigma-Aldrich Co. | Stabilized deuteroborane-tetrahydrofuran complex |
| EP2209774A1 (en) * | 2007-10-02 | 2010-07-28 | Concert Pharmaceuticals Inc. | Pyrimidinedione derivatives |
| WO2010028015A2 (en) * | 2008-09-03 | 2010-03-11 | Auspex Pharmaceuticals, Inc | 2-oxo-1,2-dihydro-quinoline modulators of immune function |
| TWI461426B (zh) * | 2009-05-27 | 2014-11-21 | Merck Sharp & Dohme | （二氫）咪唑並異〔５，１－ａ〕喹啉類 |
-
2013
- 2013-01-24 AU AU2013218368A patent/AU2013218368B2/en not_active Ceased
- 2013-01-24 ES ES13702741.3T patent/ES2672326T3/es active Active
- 2013-01-24 RU RU2014136334A patent/RU2014136334A/ru unknown
- 2013-01-24 SG SG11201403540RA patent/SG11201403540RA/en unknown
- 2013-01-24 MX MX2014009416A patent/MX2014009416A/es unknown
- 2013-01-24 BR BR112014019351A patent/BR112014019351A8/pt not_active IP Right Cessation
- 2013-01-24 JP JP2014555967A patent/JP6386382B2/ja not_active Expired - Fee Related
- 2013-01-24 WO PCT/EP2013/000215 patent/WO2013117299A1/en active Application Filing
- 2013-01-24 CA CA2860489A patent/CA2860489C/en not_active Expired - Fee Related
- 2013-01-24 EP EP13702741.3A patent/EP2812320B1/en not_active Not-in-force
- 2013-01-24 KR KR20147021930A patent/KR20140120903A/ko not_active Application Discontinuation
- 2013-01-24 US US14/372,102 patent/US20150111933A1/en not_active Abandoned
- 2013-01-24 CN CN201380008413.8A patent/CN104114544A/zh active Pending
-
2014
- 2014-08-06 IL IL233983A patent/IL233983B/en active IP Right Grant
-
2015
- 2015-03-10 HK HK15102455.7A patent/HK1201837A1/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR112014019351A2 (ko) | 2017-06-20 |
| IL233983A0 (en) | 2014-09-30 |
| KR20140120903A (ko) | 2014-10-14 |
| JP2015511943A (ja) | 2015-04-23 |
| AU2013218368A1 (en) | 2014-07-17 |
| EP2812320A1 (en) | 2014-12-17 |
| AU2013218368B2 (en) | 2017-09-07 |
| US20150111933A1 (en) | 2015-04-23 |
| ES2672326T3 (es) | 2018-06-13 |
| CN104114544A (zh) | 2014-10-22 |
| MX2014009416A (es) | 2014-11-10 |
| JP6386382B2 (ja) | 2018-09-05 |
| EP2812320B1 (en) | 2018-03-07 |
| RU2014136334A (ru) | 2016-04-10 |
| HK1201837A1 (en) | 2015-09-11 |
| CA2860489A1 (en) | 2013-08-15 |
| WO2013117299A1 (en) | 2013-08-15 |
| CA2860489C (en) | 2019-11-12 |
| BR112014019351A8 (pt) | 2017-07-11 |
| IL233983B (en) | 2019-12-31 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL233759A0 (en) | Emulsion containing hormones | |
| PL2806886T3 (pl) | Stabilizowane kompozycje białkowe oparte na semifluorowanych alkanach | |
| IL258357A (en) | A semi-solid aqueous pharmaceutical preparation containing tapentadol | |
| HK1201826A1 (en) | Benzamide derivatives as modulators of the follicle stimulating hormone | |
| AP2014007738A0 (en) | Spiroindoline derivatives as gonadotropin-releasing hormone receptor antagonists | |
| GB201203181D0 (en) | Blade tip timing uncertainty | |
| IL244986A0 (en) | Formulation for gonadotropins | |
| HK1207985A1 (en) | Somatostatin receptor agonist formulations | |
| HRP20190141T1 (hr) | Oblik doziranja antagonista receptora progesterona | |
| HK1198424A1 (en) | Thyroid stimulating hormone compositions | |
| HK1201837A1 (en) | Deuterated thiazolidinone analogues as agonists for follicle stimulating hormone receptor | |
| IL243730B (en) | Vasopressin-2 receptor agonist peptides | |
| HK1216101A1 (zh) | 用作促性腺激素釋放激素受體拮抗劑的螺二氫吲哚衍生物 | |
| HUE050861T2 (hu) | Rianodinreceptor-antagonista dantrolent tartalmazó gyógyászati készítmény sebgyógyulás elõsegítésére | |
| IL233770A0 (en) | Xanthocillin analogs with formalin groups for use as neuroprotective agents | |
| HK1250664A1 (zh) | 含有他噴他多的半固體水性藥物組合物 | |
| GB201105108D0 (en) | Wing tip pod |