SE9802574D0 - Novel compounds - Google Patents

Novel compounds

Info

Publication number
SE9802574D0
SE9802574D0 SE9802574A SE9802574A SE9802574D0 SE 9802574 D0 SE9802574 D0 SE 9802574D0 SE 9802574 A SE9802574 A SE 9802574A SE 9802574 A SE9802574 A SE 9802574A SE 9802574 D0 SE9802574 D0 SE 9802574D0
Authority
SE
Sweden
Prior art keywords
novel compounds
medicaments
processes
formula
preparation
Prior art date
Application number
SE9802574A
Other languages
English (en)
Swedish (sv)
Inventor
Simon Guile
Brian Springthorpe
Original Assignee
Astra Pharma Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astra Pharma Prod filed Critical Astra Pharma Prod
Priority to SE9802574A priority Critical patent/SE9802574D0/xx
Publication of SE9802574D0 publication Critical patent/SE9802574D0/xx
Priority to AT99941925T priority patent/ATE251162T1/de
Priority to DE69911785T priority patent/DE69911785T2/de
Priority to EP99941925A priority patent/EP1097153B1/en
Priority to JP2000560127A priority patent/JP2003519080A/ja
Priority to PCT/SE1999/001277 priority patent/WO2000004021A1/en
Priority to AU55398/99A priority patent/AU5539899A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SE9802574A 1998-07-17 1998-07-17 Novel compounds SE9802574D0 (sv)

Priority Applications (7)

Application Number Priority Date Filing Date Title
SE9802574A SE9802574D0 (sv) 1998-07-17 1998-07-17 Novel compounds
AT99941925T ATE251162T1 (de) 1998-07-17 1999-07-15 Triazolo(4,5-d)pyrimidin-verbindungen
DE69911785T DE69911785T2 (de) 1998-07-17 1999-07-15 Triazolo[4,5-d]pyrimidin-verbindungen
EP99941925A EP1097153B1 (en) 1998-07-17 1999-07-15 Novel triazolo[4,5-d]pyrimidine compounds
JP2000560127A JP2003519080A (ja) 1998-07-17 1999-07-15 新規のトリアゾロ[4,5−d]ピリミジン化合物
PCT/SE1999/001277 WO2000004021A1 (en) 1998-07-17 1999-07-15 NOVEL TRIAZOLO[4,5-d]PYRIMIDINE COMPOUNDS
AU55398/99A AU5539899A (en) 1998-07-17 1999-07-15 Novel triazolo(4,5-(d))pyrimidine compounds

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9802574A SE9802574D0 (sv) 1998-07-17 1998-07-17 Novel compounds

Publications (1)

Publication Number Publication Date
SE9802574D0 true SE9802574D0 (sv) 1998-07-17

Family

ID=20412117

Family Applications (1)

Application Number Title Priority Date Filing Date
SE9802574A SE9802574D0 (sv) 1998-07-17 1998-07-17 Novel compounds

Country Status (7)

Country Link
EP (1) EP1097153B1 (https=)
JP (1) JP2003519080A (https=)
AT (1) ATE251162T1 (https=)
AU (1) AU5539899A (https=)
DE (1) DE69911785T2 (https=)
SE (1) SE9802574D0 (https=)
WO (1) WO2000004021A1 (https=)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE9904129D0 (sv) 1999-11-15 1999-11-15 Astra Pharma Prod Novel compounds
US7504497B2 (en) 2003-10-21 2009-03-17 Inspire Pharmaceuticals, Inc. Orally bioavailable compounds and methods for inhibiting platelet aggregation
AU2004284098B2 (en) 2003-10-21 2009-07-16 Inspire Pharmaceuticals, Inc. Tetrahydro-furo [3,4-d] dioxole compounds and compositions and method for inhibiting platelet aggregation
US7335648B2 (en) 2003-10-21 2008-02-26 Inspire Pharmaceuticals, Inc. Non-nucleotide composition and method for inhibiting platelet aggregation
GB2422782A (en) 2003-10-21 2006-08-09 Inspire Pharmaceuticals Inc Non-nucleotide compositions and method for treating pain
US7749981B2 (en) 2003-10-21 2010-07-06 Inspire Pharmaceuticals, Inc. Drug-eluting stents coated with non-nucleotide P2Y12 receptor antagonist compound
US7932376B2 (en) 2005-05-05 2011-04-26 Inspire Pharmaceuticals, Inc. Pyrimidine-based non-nucleotide composition and method for inhibiting platelet aggregation
JP2010508350A (ja) 2006-10-31 2010-03-18 ヤンセン ファーマシューティカ エヌ.ベー. Adpp2y12レセプターアンタゴニストとしてのトリアゾロピリミジン誘導体
WO2015162630A1 (en) * 2014-04-25 2015-10-29 Anlon Chemical Research Organization Novel processes for preparing triazolo [4,5-d]- pyrimidines, including ticagrelor, vianew intermediates and new route of synthesis.
AR107928A1 (es) 2016-03-22 2018-06-28 Merck Sharp & Dohme Moduladores alostéricos de receptores de acetilcolina nicotínicos
CN111116592A (zh) * 2019-11-27 2020-05-08 杭州沧海帆医药科技有限公司 嘧啶并三氮唑类化合物及其医药用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TR199800019T1 (xx) * 1995-07-11 1998-05-21 Astra Pharmaceuticals Limited Trombosit topaklanmas�n� �nleyici yeni maddeler.
EP0929218A4 (en) * 1996-10-30 2001-05-16 Univ North Carolina P2Y RECEPTOR ANTAGONISTS
EP0946561B1 (en) * 1996-12-20 2002-02-13 AstraZeneca AB Triazolo(4,5-d)pyrimidinyl derivatives and their use as medicaments
SE9702772D0 (sv) * 1997-07-22 1997-07-22 Astra Pharma Prod Novel compounds

Also Published As

Publication number Publication date
EP1097153B1 (en) 2003-10-01
JP2003519080A (ja) 2003-06-17
AU5539899A (en) 2000-02-07
DE69911785T2 (de) 2004-07-29
ATE251162T1 (de) 2003-10-15
DE69911785D1 (de) 2003-11-06
EP1097153A1 (en) 2001-05-09
WO2000004021A1 (en) 2000-01-27

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