SE8207294L - 1,4-THIAZANCARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE AND COMPOSITIONS OF THESE DERIVATIVES - Google Patents

1,4-THIAZANCARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE AND COMPOSITIONS OF THESE DERIVATIVES

Info

Publication number
SE8207294L
SE8207294L SE8207294A SE8207294A SE8207294L SE 8207294 L SE8207294 L SE 8207294L SE 8207294 A SE8207294 A SE 8207294A SE 8207294 A SE8207294 A SE 8207294A SE 8207294 L SE8207294 L SE 8207294L
Authority
SE
Sweden
Prior art keywords
derivatives
hydrogen
alkyl
preparation
thiazancarboxylic
Prior art date
Application number
SE8207294A
Other languages
Swedish (sv)
Other versions
SE8207294D0 (en
Inventor
C Gillet
M Snyers
J Roba
G Lambelin
Original Assignee
Midit
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Midit filed Critical Midit
Publication of SE8207294L publication Critical patent/SE8207294L/en
Publication of SE8207294D0 publication Critical patent/SE8207294D0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
    • C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
    • C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/10—Spiro-condensed systems

Abstract

Derivatives of 1,4-thiazane-3-carboxylic acid represented by the formula I, wherein R1 and R2 are hydrogen, an alkyl radical or a phenyl nucleus substituted or not or form a cycloalkyl radical; R3 is a hydroxyl group, OR9 group, wherein R9 may have different significations; R4 is hydrogen, alkyl or CONH2, R3 and R4 forming a hydantoin cycle, R5 and R6 representing hydrogen, alkyl, phenyl substituted or not; R7 is hydrogen, alkyl, particularly dimethyl, phenyl substituted or not, and the salts of those compounds. <IMAGE> as well as the pharmaceutical compositions containing them and the intermediaries for their preparation, having the formulas II, III, IV: <IMAGE>.
SE8207294A 1981-04-29 1982-12-21 1,4-THIAZANCARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE AND COMPOSITIONS OF THESE DERIVATIVES SE8207294D0 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
LU83327A LU83327A1 (en) 1981-04-29 1981-04-29 PROCESS FOR THE PREPARATION OF 1,4-THIAZINE DERIVATIVES, THEIR USE AND COMPOSITIONS CONTAINING SUCH DERIVATIVES

Publications (2)

Publication Number Publication Date
SE8207294L true SE8207294L (en) 1982-12-21
SE8207294D0 SE8207294D0 (en) 1982-12-21

Family

ID=19729637

Family Applications (1)

Application Number Title Priority Date Filing Date
SE8207294A SE8207294D0 (en) 1981-04-29 1982-12-21 1,4-THIAZANCARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND USE AND COMPOSITIONS OF THESE DERIVATIVES

Country Status (16)

Country Link
JP (1) JPS58500713A (en)
KR (1) KR830010089A (en)
BE (1) BE893025A (en)
ES (1) ES8307233A1 (en)
FI (1) FI66366C (en)
FR (1) FR2509303A1 (en)
GB (1) GB2111056B (en)
GR (1) GR75996B (en)
IT (1) IT1190794B (en)
LU (1) LU83327A1 (en)
NL (1) NL8220153A (en)
NO (1) NO824398L (en)
PT (1) PT74813B (en)
SE (1) SE8207294D0 (en)
WO (1) WO1982003860A1 (en)
ZA (1) ZA822926B (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3436386A1 (en) * 1984-10-04 1986-04-10 Merck Patent Gmbh, 6100 Darmstadt (THIO) MORPHOLINE
FR2618434B1 (en) * 1987-07-21 1991-02-08 Oreal ESTERS OF THIAMORPHOLINONE CARBOXYLIC ACID AND DERIVATIVES THEREOF, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE COSMETIC AND DERMO-PHARMACEUTICAL FIELD
WO1990007111A2 (en) * 1988-12-14 1990-06-28 Hicks, Richard Method for predicting biological activity of antibiotics, and novel non beta-lactam antibacterial agents derived therefrom
CN104169281B (en) 2012-02-03 2016-12-14 赛诺菲 The pyrroles's diformamide condensed and they are as the purposes of medicine

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2187327B1 (en) * 1972-06-15 1975-06-20 Rech Pharm Scientifiques
US4179276A (en) * 1977-02-01 1979-12-18 E. I. Du Pont De Nemours And Company Novel imidazothiazine-1,3 (2H)-diones
JPS5540658A (en) * 1978-09-19 1980-03-22 Tanabe Seiyaku Co Ltd 1,4-thiazan-3-carboxylic ester derivative and its preparation

Also Published As

Publication number Publication date
BE893025A (en) 1982-10-29
FI824279A0 (en) 1982-12-14
WO1982003860A1 (en) 1982-11-11
FI66366B (en) 1984-06-29
NO824398L (en) 1982-12-28
KR830010089A (en) 1983-12-26
LU83327A1 (en) 1983-03-24
PT74813A (en) 1982-05-01
JPS58500713A (en) 1983-05-06
PT74813B (en) 1983-10-26
JPH0330592B2 (en) 1991-04-30
ES511759A0 (en) 1983-07-01
ZA822926B (en) 1983-03-30
FR2509303A1 (en) 1983-01-14
GB2111056B (en) 1985-03-06
GR75996B (en) 1984-08-03
GB2111056A (en) 1983-06-29
FI66366C (en) 1984-10-10
SE8207294D0 (en) 1982-12-21
ES8307233A1 (en) 1983-07-01
FI824279L (en) 1982-12-14
IT8220998A0 (en) 1982-04-29
NL8220153A (en) 1983-03-01
IT1190794B (en) 1988-02-24

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