ES8307233A1 - Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same - Google Patents
Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing sameInfo
- Publication number
- ES8307233A1 ES8307233A1 ES82511759A ES511759A ES8307233A1 ES 8307233 A1 ES8307233 A1 ES 8307233A1 ES 82511759 A ES82511759 A ES 82511759A ES 511759 A ES511759 A ES 511759A ES 8307233 A1 ES8307233 A1 ES 8307233A1
- Authority
- ES
- Spain
- Prior art keywords
- hydrogen
- alkyl
- thiazane
- derivatives
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/12—1,4-Thiazines; Hydrogenated 1,4-thiazines not condensed with other rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
- C07D279/10—1,4-Thiazines; Hydrogenated 1,4-thiazines
- C07D279/14—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems
- C07D279/16—1,4-Thiazines; Hydrogenated 1,4-thiazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/10—Spiro-condensed systems
Abstract
Derivatives of 1,4-thiazane-3-carboxylic acid represented by the formula I, wherein R1 and R2 are hydrogen, an alkyl radical or a phenyl nucleus substituted or not or form a cycloalkyl radical R3 is a hydroxyl group, OR9 group, wherein R9 may have different significations R4 is hydrogen, alkyl or CONH2, R3 and R4 forming a hydantoin cycle, R5 and R6 representing hydrogen, alkyl, phenyl substituted or not R7 is hydrogen, alkyl, particularly dimethyl, phenyl substituted or not, and the salts of those compounds. < IMAGE > as well as the pharmaceutical compositions containing them and the intermediaries for their preparation, having the formulas II, III, IV: < IMAGE >.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU83327A LU83327A1 (en) | 1981-04-29 | 1981-04-29 | PROCESS FOR THE PREPARATION OF 1,4-THIAZINE DERIVATIVES, THEIR USE AND COMPOSITIONS CONTAINING SUCH DERIVATIVES |
Publications (2)
Publication Number | Publication Date |
---|---|
ES511759A0 ES511759A0 (en) | 1983-07-01 |
ES8307233A1 true ES8307233A1 (en) | 1983-07-01 |
Family
ID=19729637
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES82511759A Expired ES8307233A1 (en) | 1981-04-29 | 1982-04-28 | Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same |
Country Status (16)
Country | Link |
---|---|
JP (1) | JPS58500713A (en) |
KR (1) | KR830010089A (en) |
BE (1) | BE893025A (en) |
ES (1) | ES8307233A1 (en) |
FI (1) | FI66366C (en) |
FR (1) | FR2509303A1 (en) |
GB (1) | GB2111056B (en) |
GR (1) | GR75996B (en) |
IT (1) | IT1190794B (en) |
LU (1) | LU83327A1 (en) |
NL (1) | NL8220153A (en) |
NO (1) | NO824398L (en) |
PT (1) | PT74813B (en) |
SE (1) | SE8207294D0 (en) |
WO (1) | WO1982003860A1 (en) |
ZA (1) | ZA822926B (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3436386A1 (en) * | 1984-10-04 | 1986-04-10 | Merck Patent Gmbh, 6100 Darmstadt | (THIO) MORPHOLINE |
FR2618434B1 (en) * | 1987-07-21 | 1991-02-08 | Oreal | ESTERS OF THIAMORPHOLINONE CARBOXYLIC ACID AND DERIVATIVES THEREOF, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE COSMETIC AND DERMO-PHARMACEUTICAL FIELD |
WO1990007111A2 (en) * | 1988-12-14 | 1990-06-28 | Hicks, Richard | Method for predicting biological activity of antibiotics, and novel non beta-lactam antibacterial agents derived therefrom |
CN104169281B (en) | 2012-02-03 | 2016-12-14 | 赛诺菲 | The pyrroles's diformamide condensed and they are as the purposes of medicine |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2187327B1 (en) * | 1972-06-15 | 1975-06-20 | Rech Pharm Scientifiques | |
US4179276A (en) * | 1977-02-01 | 1979-12-18 | E. I. Du Pont De Nemours And Company | Novel imidazothiazine-1,3 (2H)-diones |
JPS5540658A (en) * | 1978-09-19 | 1980-03-22 | Tanabe Seiyaku Co Ltd | 1,4-thiazan-3-carboxylic ester derivative and its preparation |
-
1981
- 1981-04-29 LU LU83327A patent/LU83327A1/en unknown
-
1982
- 1982-04-21 JP JP57501451A patent/JPS58500713A/en active Granted
- 1982-04-21 WO PCT/BE1982/000009 patent/WO1982003860A1/en active IP Right Grant
- 1982-04-21 GB GB08235353A patent/GB2111056B/en not_active Expired
- 1982-04-21 NL NL8220153A patent/NL8220153A/en unknown
- 1982-04-28 ES ES82511759A patent/ES8307233A1/en not_active Expired
- 1982-04-28 PT PT74813A patent/PT74813B/en unknown
- 1982-04-29 GR GR68018A patent/GR75996B/el unknown
- 1982-04-29 ZA ZA822926A patent/ZA822926B/en unknown
- 1982-04-29 BE BE0/207967A patent/BE893025A/en not_active IP Right Cessation
- 1982-04-29 IT IT20998/82A patent/IT1190794B/en active
- 1982-04-29 KR KR1019820001874A patent/KR830010089A/en unknown
- 1982-04-29 FR FR8207461A patent/FR2509303A1/en not_active Withdrawn
- 1982-12-14 FI FI771226A patent/FI66366C/en not_active IP Right Cessation
- 1982-12-21 SE SE8207294A patent/SE8207294D0/en not_active Application Discontinuation
- 1982-12-28 NO NO824398A patent/NO824398L/en unknown
Also Published As
Publication number | Publication date |
---|---|
BE893025A (en) | 1982-10-29 |
FI824279A0 (en) | 1982-12-14 |
WO1982003860A1 (en) | 1982-11-11 |
FI66366B (en) | 1984-06-29 |
NO824398L (en) | 1982-12-28 |
KR830010089A (en) | 1983-12-26 |
SE8207294L (en) | 1982-12-21 |
LU83327A1 (en) | 1983-03-24 |
PT74813A (en) | 1982-05-01 |
JPS58500713A (en) | 1983-05-06 |
PT74813B (en) | 1983-10-26 |
JPH0330592B2 (en) | 1991-04-30 |
ES511759A0 (en) | 1983-07-01 |
ZA822926B (en) | 1983-03-30 |
FR2509303A1 (en) | 1983-01-14 |
GB2111056B (en) | 1985-03-06 |
GR75996B (en) | 1984-08-03 |
GB2111056A (en) | 1983-06-29 |
FI66366C (en) | 1984-10-10 |
SE8207294D0 (en) | 1982-12-21 |
FI824279L (en) | 1982-12-14 |
IT8220998A0 (en) | 1982-04-29 |
NL8220153A (en) | 1983-03-01 |
IT1190794B (en) | 1988-02-24 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
GR3005315T3 (en) | ||
ES8306759A1 (en) | Cephalosporin derivatives, their preparation and compositions containing them. | |
ES8605506A1 (en) | Piperidine derivatives, their preparation and their therapeutical application. | |
ES8203883A1 (en) | Imidazole derivatives, their preparation and compositions containing them. | |
ES8302001A1 (en) | Cephalosporin derivatives, a process for their preparation and compositions containing them. | |
ES8507090A1 (en) | 1,5-Benzothiazepines with cardiovascular utility, and pharmaceutical compositions containing them | |
ES486824A1 (en) | Neuroleptic-4-(naphthylmethyl)piperidine derivatives | |
ES8205791A1 (en) | 2-(1,4-Benzodioxan-2-ylalkyl) imidazoles, their preparation and pharmaceutical compositions containing them. | |
ES8106289A1 (en) | Derivatives of alpha-phenyl-2-pyrrolidine methanol and their salts, process for their preparation, use as medicines and compositions containing them. | |
ES8401063A1 (en) | Derivatives of substituted N-alkylimidazoles, their preparation and pharmaceutical compositions containing them. | |
ES8307233A1 (en) | Derivatives of 1,4-thiazane-carboxylic acid, preparation and utilization thereof and compositions containing same | |
ES8303397A1 (en) | 1(4-Quinolyl)ethanol or propanol derivatives, pharmaceutical compositions containing them and processes for their preparation. | |
ES8202818A1 (en) | Tetrazolylcoumarin derivatives, process for preparing the same and composition containing the same. | |
ES8104241A1 (en) | 1-((Substituted-naphthyl)ethyl)-imidazole derivatives, pharmaceutical compositions containing them and methods of making them. | |
ES8305359A1 (en) | Bicyclo (3,2,1) octylbenzamides, a process for their preparation and pharmaceutical compositions containing them. | |
ES8400743A1 (en) | 1-Phenylindazol-3-one compounds, process and intermediates for their preparation and medicines containing these compounds. | |
PT80787A (en) | Process for preparing piperidine (or pyrrolidine)-butanamides and compounds relating to them | |
ES8401761A1 (en) | 1-(3,4,5-Trimethoxycinnamoyl)-4-aminocarbonylethyl-substituted piperazine derivatives and a process for the preparation thereof. | |
ES8500742A1 (en) | Phenyl-acetic-acid derivatives, their preparation and pharmaceutical compostions containing them. | |
ES8403891A1 (en) | Furyloxazolylacetic acid derivatives, process for preparing same and pharmaceutical compositions containing same. | |
IE801382L (en) | Piperidines. | |
ES8506011A1 (en) | Derivatives of tetrahydrobenzothiazole and herbicidal compositions containing the same as an active ingredient | |
ES8702909A1 (en) | Tetrahydro-beta-carboline derivatives and process for the preparation thereof. | |
ES8401957A1 (en) | Preparation of thiophene compounds | |
ES8205816A1 (en) | Cardenolide-bis-digitoxoside derivatives, process for their preparation and their utilization as medicines. |