SE7704870L - PROCEDURE FOR PREPARING 4-SUBSTITUTED IMIDAZOLE COMPOUNDS - Google Patents

PROCEDURE FOR PREPARING 4-SUBSTITUTED IMIDAZOLE COMPOUNDS

Info

Publication number
SE7704870L
SE7704870L SE7704870A SE7704870A SE7704870L SE 7704870 L SE7704870 L SE 7704870L SE 7704870 A SE7704870 A SE 7704870A SE 7704870 A SE7704870 A SE 7704870A SE 7704870 L SE7704870 L SE 7704870L
Authority
SE
Sweden
Prior art keywords
preparing
imidazole compounds
procedure
substituted imidazole
formula
Prior art date
Application number
SE7704870A
Other languages
Swedish (sv)
Other versions
SE442199B (en
Inventor
J J Lewis
R L Webb
Original Assignee
Smithkline Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/771,044 external-priority patent/US4119781A/en
Application filed by Smithkline Corp filed Critical Smithkline Corp
Publication of SE7704870L publication Critical patent/SE7704870L/en
Publication of SE442199B publication Critical patent/SE442199B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/84—Sulfur atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88—Nitrogen atoms, e.g. allantoin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
    • C07F9/6503—Five-membered rings
    • C07F9/6506—Five-membered rings having the nitrogen atoms in positions 1 and 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

The imidazole compounds of the general formula II represent valuable intermediates for preparing pharmacologically active compounds. They are obtained by reacting a compound of the formula I in an organic solvent under basic conditions with a compound of formula R<2>-H. The symbols used in the general formulae I and II are defined in Claim 1. <IMAGE>
SE7704870A 1977-02-22 1977-04-27 PROCEDURE FOR PREPARING 4-SUBSTITUTED IMIDAZOLD DERIVATIVES SE442199B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/771,044 US4119781A (en) 1975-10-29 1977-02-22 Process for preparing 4-substituted imidazole compounds

Publications (2)

Publication Number Publication Date
SE7704870L true SE7704870L (en) 1978-08-23
SE442199B SE442199B (en) 1985-12-09

Family

ID=25090518

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7704870A SE442199B (en) 1977-02-22 1977-04-27 PROCEDURE FOR PREPARING 4-SUBSTITUTED IMIDAZOLD DERIVATIVES
SE8008935A SE452887B (en) 1977-02-22 1980-12-18 PHOSPHONIUM METHYLIMIDAZOLE SUBSTANCE USED AS INTERMEDIATE IN THE PREPARATION OF CERTAIN PHARMACOLOGICALLY ACTIVE GUANIDINE AND TIOCHARBAMIDE COMPOUNDS

Family Applications After (1)

Application Number Title Priority Date Filing Date
SE8008935A SE452887B (en) 1977-02-22 1980-12-18 PHOSPHONIUM METHYLIMIDAZOLE SUBSTANCE USED AS INTERMEDIATE IN THE PREPARATION OF CERTAIN PHARMACOLOGICALLY ACTIVE GUANIDINE AND TIOCHARBAMIDE COMPOUNDS

Country Status (22)

Country Link
AR (1) AR217073A1 (en)
AT (1) AT355015B (en)
BE (1) BE853954R (en)
CA (1) CA1084052A (en)
CH (2) CH631167A5 (en)
DE (1) DE2718715A1 (en)
DK (1) DK168277A (en)
ES (1) ES458153A1 (en)
FI (1) FI73208C (en)
FR (1) FR2381031A2 (en)
GB (1) GB1582865A (en)
HU (1) HU174840B (en)
IE (1) IE45035B1 (en)
IL (1) IL51898A (en)
IN (1) IN148285B (en)
IT (1) IT1078449B (en)
LU (1) LU77200A1 (en)
MX (1) MX4663E (en)
NL (1) NL7704617A (en)
NO (1) NO152903C (en)
PT (1) PT66446B (en)
SE (2) SE442199B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL57415A (en) * 1978-05-30 1984-08-31 Smith Kline French Lab Nitropyrrole compounds,process for preparing them and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
IL51898A (en) 1980-07-31
GB1582865A (en) 1981-01-14
NL7704617A (en) 1978-08-24
FR2381031B2 (en) 1982-09-17
FI73208B (en) 1987-05-29
FI73208C (en) 1987-09-10
NO152903C (en) 1985-12-11
AR217073A1 (en) 1980-02-29
NO771453L (en) 1978-08-23
LU77200A1 (en) 1977-08-17
ES458153A1 (en) 1978-04-01
NO152903B (en) 1985-09-02
IT1078449B (en) 1985-05-08
IE45035B1 (en) 1982-06-02
FR2381031A2 (en) 1978-09-15
IN148285B (en) 1981-01-03
DK168277A (en) 1978-08-23
CH631167A5 (en) 1982-07-30
SE442199B (en) 1985-12-09
IE45035L (en) 1978-08-22
CH631168A5 (en) 1982-07-30
MX4663E (en) 1982-07-21
AT355015B (en) 1980-02-11
DE2718715A1 (en) 1978-08-31
IL51898A0 (en) 1977-06-30
FI771291A (en) 1978-08-23
ATA289577A (en) 1979-07-15
PT66446A (en) 1977-05-01
HU174840B (en) 1980-03-28
SE8008935L (en) 1980-12-18
SE452887B (en) 1987-12-21
CA1084052A (en) 1980-08-19
BE853954R (en) 1977-10-26
PT66446B (en) 1978-09-22

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