SE7701845L - PROCEDURE FOR THE PREPARATION OF L-SULFONYL-5 (6) -Substituted BENSIMIDAZOLES - Google Patents
PROCEDURE FOR THE PREPARATION OF L-SULFONYL-5 (6) -Substituted BENSIMIDAZOLESInfo
- Publication number
- SE7701845L SE7701845L SE7701845A SE7701845A SE7701845L SE 7701845 L SE7701845 L SE 7701845L SE 7701845 A SE7701845 A SE 7701845A SE 7701845 A SE7701845 A SE 7701845A SE 7701845 L SE7701845 L SE 7701845L
- Authority
- SE
- Sweden
- Prior art keywords
- image
- bensimidazoles
- sulfonyl
- substituted
- procedure
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Virology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
Abstract
Sulphonylbenzimidazole derivatives of formula <IMAGE> wherein R2 represents <IMAGE> and the substituents R, R5 and R6 are defined in Claim 1, are prepared by reacting a corresponding sulphonylbenzimidazole which instead of the substituent R2 has a group <IMAGE> with a C1-C7-alkyl-magnesium halide or C1-C7-alkyl-lithium and then performing a hydrolysis. Dehydration of the compounds of formula I gives compounds which contain the group <IMAGE> The compounds prepared may be used for the control of viruses.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US05/750,991 US4118742A (en) | 1975-08-28 | 1976-12-15 | Carbonyl-substituted 1-sulfonylbenzimidazoles |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| SE7701845L true SE7701845L (en) | 1978-06-16 |
| SE433351B SE433351B (en) | 1984-05-21 |
Family
ID=25019992
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE7701845A SE433351B (en) | 1976-12-15 | 1977-02-18 | PROCEDURE FOR PREPARING SULPHONYL BENZIMIDAZOLES |
| SE8008090A SE433352B (en) | 1976-12-15 | 1980-11-18 | PROCEDURE FOR PREPARING SULPHONYL BENZIMIDAZOLES |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SE8008090A SE433352B (en) | 1976-12-15 | 1980-11-18 | PROCEDURE FOR PREPARING SULPHONYL BENZIMIDAZOLES |
Country Status (26)
| Country | Link |
|---|---|
| JP (1) | JPS5377062A (en) |
| AR (1) | AR225397A1 (en) |
| AT (1) | AT347937B (en) |
| AU (1) | AU509374B2 (en) |
| BE (1) | BE851630A (en) |
| BG (1) | BG27742A3 (en) |
| CA (1) | CA1079737A (en) |
| CH (1) | CH630368A5 (en) |
| CS (1) | CS190339B2 (en) |
| DD (1) | DD129445A6 (en) |
| DE (1) | DE2706227A1 (en) |
| DK (1) | DK145645C (en) |
| ES (1) | ES456090A1 (en) |
| FR (1) | FR2374311A2 (en) |
| GB (1) | GB1568543A (en) |
| GR (1) | GR66420B (en) |
| HU (1) | HU175361B (en) |
| IE (1) | IE44863B1 (en) |
| IL (1) | IL51445A (en) |
| MX (1) | MX4495E (en) |
| NL (1) | NL187396C (en) |
| PL (1) | PL106887B1 (en) |
| RO (1) | RO71886A (en) |
| SE (2) | SE433351B (en) |
| SU (1) | SU680645A3 (en) |
| ZA (1) | ZA77691B (en) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4420479A (en) * | 1982-04-08 | 1983-12-13 | Eli Lilly And Company | Olefinic benzimidazoles, formulations, and antiviral methods |
| FR2593177B1 (en) * | 1986-01-20 | 1988-04-01 | Novapharme | NEW BENZIMIDAZO |
| US5693661A (en) * | 1995-06-07 | 1997-12-02 | Eli Lilly And Company | Anti-viral compounds |
| JP7226480B2 (en) | 2020-07-30 | 2023-02-21 | 大日本印刷株式会社 | Antiviral article and antiviral resin composition |
| WO2022059676A1 (en) | 2020-09-18 | 2022-03-24 | 大日本印刷株式会社 | Antiviral article and antiviral resin composition |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS51125078A (en) * | 1974-07-01 | 1976-11-01 | Lilly Co Eli | Production of substituted 11sulphonylbenzimidazole |
-
1977
- 1977-02-07 ZA ZA00770691A patent/ZA77691B/en unknown
- 1977-02-07 GR GR52736A patent/GR66420B/el unknown
- 1977-02-08 CA CA271,307A patent/CA1079737A/en not_active Expired
- 1977-02-08 IE IE259/77A patent/IE44863B1/en not_active IP Right Cessation
- 1977-02-09 GB GB5254/77A patent/GB1568543A/en not_active Expired
- 1977-02-14 IL IL51445A patent/IL51445A/en unknown
- 1977-02-14 DE DE19772706227 patent/DE2706227A1/en active Granted
- 1977-02-17 NL NLAANVRAGE7701715,A patent/NL187396C/en not_active IP Right Cessation
- 1977-02-17 RO RO7789438A patent/RO71886A/en unknown
- 1977-02-18 HU HU77EI729A patent/HU175361B/en unknown
- 1977-02-18 AR AR266611A patent/AR225397A1/en active
- 1977-02-18 FR FR7704799A patent/FR2374311A2/en active Granted
- 1977-02-18 ES ES456090A patent/ES456090A1/en not_active Expired
- 1977-02-18 DD DD7700197445A patent/DD129445A6/en unknown
- 1977-02-18 JP JP1769877A patent/JPS5377062A/en active Granted
- 1977-02-18 BG BG7735460A patent/BG27742A3/en unknown
- 1977-02-18 SE SE7701845A patent/SE433351B/en not_active IP Right Cessation
- 1977-02-18 CS CS771093A patent/CS190339B2/en unknown
- 1977-02-18 DK DK73277A patent/DK145645C/en not_active IP Right Cessation
- 1977-02-18 SU SU772452269A patent/SU680645A3/en active
- 1977-02-18 MX MX775442U patent/MX4495E/en unknown
- 1977-02-18 AU AU22440/77A patent/AU509374B2/en not_active Expired
- 1977-02-18 CH CH207577A patent/CH630368A5/en not_active IP Right Cessation
- 1977-02-18 AT AT111277A patent/AT347937B/en not_active IP Right Cessation
- 1977-02-18 BE BE1007954A patent/BE851630A/en not_active IP Right Cessation
- 1977-02-19 PL PL1977196131A patent/PL106887B1/en unknown
-
1980
- 1980-11-18 SE SE8008090A patent/SE433352B/en not_active IP Right Cessation
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