SE7514459L - ALIFATIC SULFAMAT - Google Patents

ALIFATIC SULFAMAT

Info

Publication number
SE7514459L
SE7514459L SE7514459A SE7514459A SE7514459L SE 7514459 L SE7514459 L SE 7514459L SE 7514459 A SE7514459 A SE 7514459A SE 7514459 A SE7514459 A SE 7514459A SE 7514459 L SE7514459 L SE 7514459L
Authority
SE
Sweden
Prior art keywords
radicals
formula
compounds
reacting
aralkyl
Prior art date
Application number
SE7514459A
Other languages
Swedish (sv)
Inventor
A F Hirsch
Original Assignee
Ortho Pharma Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/537,613 external-priority patent/US3997585A/en
Priority claimed from US05/618,998 external-priority patent/US4061663A/en
Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp
Publication of SE7514459L publication Critical patent/SE7514459L/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C307/00—Amides of sulfuric acids, i.e. compounds having singly-bound oxygen atoms of sulfate groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C307/02—Monoamides of sulfuric acids or esters thereof, e.g. sulfamic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Bis-O-sulphamylglycols of the general formula I <IMAGE> are prepared by reacting a glycol of the formula II <IMAGE> with a sulphamyl chloride of the formula III (Hal)-SO2NR1R2 (III> in a solvent in the presence of a strong base. In these compounds, n is zero or an integer from 1 to 8, X and Y denote hydrogen, and if n is 1 additionally denotes lower alkyl radicals, aryl radicals, aralkyl radicals or cyclohexyl radicals. R1 and R2, independently of one another, are hydrogen atoms, alkyl, aryl, aralkyl or cycloalkyl radicals, or they form, together with the nitrogen atom to which they are bonded, a pyrrolidinyl ring or piperidinyl ring. Those compounds of the formula I in which all the radicals R1 and R2 are hydrogen atoms are also prepared by reacting a sulphamoyl halide of the formula III carrying a protective group on its nitrogen atom and, after the reaction, removing this protective group using an acid. The compounds of the formula I are suitable for regulation of the fertility of male animals.
SE7514459A 1974-12-30 1975-12-19 ALIFATIC SULFAMAT SE7514459L (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/537,613 US3997585A (en) 1974-12-30 1974-12-30 Aliphatic sulfamates
US05/618,998 US4061663A (en) 1975-10-02 1975-10-02 Process for preparation of aliphatic primary sulfamates

Publications (1)

Publication Number Publication Date
SE7514459L true SE7514459L (en) 1976-07-01

Family

ID=27065556

Family Applications (1)

Application Number Title Priority Date Filing Date
SE7514459A SE7514459L (en) 1974-12-30 1975-12-19 ALIFATIC SULFAMAT

Country Status (11)

Country Link
JP (1) JPS5198217A (en)
AT (1) AT357998B (en)
CA (1) CA1082194A (en)
CH (1) CH617184A5 (en)
DE (1) DE2559210A1 (en)
DK (1) DK579975A (en)
FR (1) FR2296410A1 (en)
GB (1) GB1524727A (en)
NL (1) NL7514794A (en)
NO (1) NO141607C (en)
SE (1) SE7514459L (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PT94305B (en) * 1989-06-12 1997-02-28 Robins Co Inc A H METHOD FOR PREPARING COMPOUNDS HAVING ONE OR MORE USED AMINOSULFONYLOXIDE RADIATIONS AS PHARMACEUTICAL PRODUCTS
US5194446A (en) * 1989-06-12 1993-03-16 A. H. Robins Company, Incorporated Compounds having one or more aminosulfaonyloxy radicals useful as pharmaceuticals
US5273993A (en) * 1989-06-12 1993-12-28 A. H. Robins Company, Incorporated Compounds having one or more aminosulfonyloxy radicals useful as pharmaceuticals
US6011024A (en) 1991-08-28 2000-01-04 Imperial College Of Science Technology & Medicine Steroid sulphatase inhibitors
US6476011B1 (en) 1991-08-28 2002-11-05 Sterix Limited Methods for introducing an estrogenic compound
US6903084B2 (en) 1991-08-29 2005-06-07 Sterix Limited Steroid sulphatase inhibitors
CA2209229C (en) * 1995-11-02 2007-10-16 Yukong Limited Novel sulfamate compound containing n-substituted carbamoyl group and method for preparing the same
KR970027051A (en) * 1995-11-02 1997-06-24 조규향 Novel Sulfamate Compounds Containing Carbamoyl Groups
US7335650B2 (en) 2000-01-14 2008-02-26 Sterix Limited Composition

Also Published As

Publication number Publication date
NO141607B (en) 1980-01-02
JPS5198217A (en) 1976-08-30
FR2296410A1 (en) 1976-07-30
ATA986175A (en) 1980-01-15
NL7514794A (en) 1976-07-02
CH617184A5 (en) 1980-05-14
DK579975A (en) 1976-07-01
NO754009L (en) 1976-07-01
AT357998B (en) 1980-08-11
CA1082194A (en) 1980-07-22
GB1524727A (en) 1978-09-13
DE2559210A1 (en) 1976-07-01
NO141607C (en) 1980-04-09
FR2296410B1 (en) 1979-09-21

Similar Documents

Publication Publication Date Title
ES2051693T3 (en) PROCEDURE FOR PREPARING SULFONAMIDE BICYCLE COMPOUNDS.
NO792792L (en) IMMUNOMODULATORS AND ANTIVIRAL AGENTS
SE8104783L (en) Heterocyclic Associations
SE7514459L (en) ALIFATIC SULFAMAT
DK399386D0 (en) INDOLINO DERIVATIVES, THEIR PREPARATION AND USE AS PHARMACEUTICALS
KR830005110A (en) Method for preparing fluorene derivative
JPS5771602A (en) Novel carried metallic ion sealing agent, its manufacture and its use to organic synthesis and metal extraction
ATE14428T1 (en) PROCESS FOR THE PREPARATION OF BROMINATED 1,3DIOXOLEN-2-ONES.
ATE90682T1 (en) PROCESS FOR THE MANUFACTURE OF CEFODIZIME.
SE7714656L (en) SULFAMOYLBENZOIC ACIDS
ES428400A1 (en) Pheno aldehydes
KR900018067A (en) Method for preparing cyclic sulfate
KR840004089A (en) Method for preparing guanidino heterocyclic phenylamidine
GB917078A (en) Improvements in or relating to piperidine derivatives
KR840007564A (en) Method for preparing substituted benzylcycloalkenylurea derivatives
GB1312211A (en) Phosphorus-containing dibromoeopentyl glycol ester derivatives
KR840002821A (en) Method for preparing N- (2,3-epoxypropylene) -N-aralkylsulfonamide derivative
KR850003389A (en) Novel benzoylurea derivatives and methods for preparing these intermediates
GB1482388A (en) Method of producing 6-beta-amidinopenicillanic acid derivatives
KR840001150A (en) Method for preparing substituted phenyl (thioo) carbamate
SE8302084L (en) NEW BENZIMIDAZOLD DERIVATIVES
KR860000285A (en) Method for preparing 1,4-dihydropyridine derivative
KR850004588A (en) Method for preparing 2-thiocyanato-benzamide
GB1071815A (en) Phenothiazine derivatives
CH608797A5 (en) Process for the preparation of heterocyclic compounds